ATE319703T1 - Piperidinverbindungen, die sich als modulatoren der chemokinrezeptoraktivität eignen - Google Patents

Piperidinverbindungen, die sich als modulatoren der chemokinrezeptoraktivität eignen

Info

Publication number: ATE319703T1
Authority: AT; Austria
Prior art keywords: modulators; chemokine receptor; receptor activity; compounds suitable; piperidine compounds
Prior art date: 2001-07-02

Application number

AT02747793T

Other languages

English (en)

Inventor

Richard Evans

Matthew Perry

Brian Springthorpe

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-07-02

Filing date

2002-07-01

Publication date

2006-03-15

2001-07-02 Priority claimed from GB0116179A external-priority patent/GB0116179D0/en

2001-09-25 Priority claimed from GB0123037A external-priority patent/GB0123037D0/en

2002-07-01 Application filed filed Critical

2006-03-15 Application granted granted Critical

2006-03-15 Publication of ATE319703T1 publication Critical patent/ATE319703T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
- C07D211/96—Sulfur atom
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
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Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Virology (AREA)
Oncology (AREA)
Neurology (AREA)
Dermatology (AREA)
Communicable Diseases (AREA)
Immunology (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Hematology (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Molecular Biology (AREA)
Urology & Nephrology (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Obesity (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Heart & Thoracic Surgery (AREA)
AIDS & HIV (AREA)
Tropical Medicine & Parasitology (AREA)
Hospice & Palliative Care (AREA)

AT02747793T 2001-07-02 2002-07-01 Piperidinverbindungen, die sich als modulatoren der chemokinrezeptoraktivität eignen ATE319703T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0116179A GB0116179D0 (en)	2001-07-02	2001-07-02	Chemical compounds
GB0123037A GB0123037D0 (en)	2001-09-25	2001-09-25	Chemical compounds

Publications (1)

Publication Number	Publication Date
ATE319703T1 true ATE319703T1 (de)	2006-03-15

Family

ID=26246268

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT02747793T ATE319703T1 (de)	2001-07-02	2002-07-01	Piperidinverbindungen, die sich als modulatoren der chemokinrezeptoraktivität eignen

Country Status (25)

Country	Link
US (1)	US7307090B2 (de)
EP (2)	EP1604982A1 (de)
JP (1)	JP3857270B2 (de)
KR (1)	KR20040013090A (de)
CN (1)	CN1545509A (de)
AR (1)	AR042401A1 (de)
AT (1)	ATE319703T1 (de)
BR (1)	BR0210733A (de)
CA (1)	CA2452597A1 (de)
CO (1)	CO5540307A2 (de)
CY (1)	CY1106095T1 (de)
DE (1)	DE60209736T2 (de)
DK (1)	DK1404667T3 (de)
ES (1)	ES2258642T3 (de)
HU (1)	HUP0401886A2 (de)
IL (1)	IL159256A0 (de)
IS (1)	IS7094A (de)
MX (1)	MXPA03011722A (de)
NO (1)	NO20035729L (de)
NZ (1)	NZ530202A (de)
PL (1)	PL368041A1 (de)
PT (1)	PT1404667E (de)
RU (1)	RU2004100839A (de)
SA (1)	SA02230184B1 (de)
WO (1)	WO2003004487A1 (de)

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ATE372330T1 (de) *	2002-03-21	2007-09-15	Abbott Lab	N-sulfonylurea-apoptosis-förderer
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SE0202838D0 (sv) *	2002-09-24	2002-09-24	Astrazeneca Ab	Chemical compounds
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SE0302956D0 (sv) *	2003-11-07	2003-11-07	Astrazeneca Ab	Chemical compounds
SE0400925D0 (sv) *	2004-04-06	2004-04-06	Astrazeneca Ab	Chemical compounds
SE0403003D0 (sv) *	2004-12-09	2004-12-09	Astrazeneca Ab	Chemical compound 1
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RU2008136391A (ru) *	2006-02-10	2010-03-20	Янссен Фармацевтика Н.В. (Be)	Пиперидиновые производные в качестве антагонистов рецептора cхcr3
EA200870246A1 (ru) *	2006-02-10	2009-02-27	Янссен Фармацевтика Н.В.	Производные пиперидина в качестве антагонистов cxcr3-рецептора
ES2499018T3 (es) *	2007-09-20	2014-09-26	Irm Llc	Compuestos y composiciones como moduladores de la actividad de GPR119
AU2009322346B2 (en)	2008-12-03	2015-07-02	The Scripps Research Institute	Stem cell cultures
RU2726206C2 (ru)	2015-05-21	2020-07-09	Кемосентрикс, Инк.	Модуляторы ccr2
EP3687525B1 (de)	2017-09-25	2025-10-29	ChemoCentryx, Inc.	Kombinationstherapie mit einem chemokinrezeptor-2 (ccr2)-antagonist und einem pd-1/pd-l1-inhibitor
CN112105353B (zh)	2018-01-08	2024-04-19	凯莫森特里克斯股份有限公司	Ccr2拮抗剂治疗实体瘤的方法
US20190269664A1 (en)	2018-01-08	2019-09-05	Chemocentryx, Inc.	Methods of treating solid tumors with ccr2 antagonists
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- 2002-07-01 CN CNA028162714A patent/CN1545509A/zh active Pending
- 2002-07-01 DK DK02747793T patent/DK1404667T3/da active
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Publication number	Publication date
SA02230184B1 (ar)	2007-03-25
PT1404667E (pt)	2006-07-31
EP1404667B1 (de)	2006-03-08
EP1404667A1 (de)	2004-04-07
BR0210733A (pt)	2004-07-20
IS7094A (is)	2003-12-30
EP1604982A1 (de)	2005-12-14
NO20035729L (no)	2004-02-23
RU2004100839A (ru)	2005-06-20
NO20035729D0 (no)	2003-12-19
DK1404667T3 (da)	2006-07-10
US20040235894A1 (en)	2004-11-25
PL368041A1 (en)	2005-03-21
ES2258642T3 (es)	2006-09-01
KR20040013090A (ko)	2004-02-11
US7307090B2 (en)	2007-12-11
CN1545509A (zh)	2004-11-10
HK1062559A1 (en)	2004-11-12
HUP0401886A2 (hu)	2004-12-28
WO2003004487A1 (en)	2003-01-16
AR042401A1 (es)	2005-06-22
JP2004536112A (ja)	2004-12-02
CY1106095T1 (el)	2011-06-08
JP3857270B2 (ja)	2006-12-13
IL159256A0 (en)	2004-06-01
CO5540307A2 (es)	2005-07-29
MXPA03011722A (es)	2004-03-19
DE60209736D1 (de)	2006-05-04
CA2452597A1 (en)	2003-01-16
DE60209736T2 (de)	2006-11-02
NZ530202A (en)	2005-06-24

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