ATE334121T1 - Verfahren zur herstellung von threo-1,2-epoxy-3- amino-4-phenylbutan-derivaten - Google Patents

Verfahren zur herstellung von threo-1,2-epoxy-3- amino-4-phenylbutan-derivaten

Info

Publication number: ATE334121T1
Authority: AT; Austria
Prior art keywords: amino; epoxy; threo; phenylbutane; derivatives
Prior art date: 1999-01-29

Application number

AT00901998T

Other languages

English (en)

Inventor

Katsuji Maehara

Yukinori Tokuda

Hiroshi Murao

Yasuyoshi Ueda

Original Assignee

Kaneka Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-29

Filing date

2000-01-31

Publication date

2006-08-15

2000-01-31 Application filed by Kaneka Corp filed Critical Kaneka Corp

2006-08-15 Application granted granted Critical

2006-08-15 Publication of ATE334121T1 publication Critical patent/ATE334121T1/de

Links

238000004519 manufacturing process Methods 0.000 title abstract 2
239000003495 polar organic solvent Substances 0.000 abstract 2
239000002904 solvent Substances 0.000 abstract 1
XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D301/00—Preparation of oxiranes
- C07D301/02—Synthesis of the oxirane ring
- C07D301/24—Synthesis of the oxirane ring by splitting off HAL—Y from compounds containing the radical HAL—C—C—OY
- C07D301/26—Y being hydrogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/36—Compounds containing oxirane rings with hydrocarbon radicals, substituted by nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Epoxy Compounds (AREA)

AT00901998T 1999-01-29 2000-01-31 Verfahren zur herstellung von threo-1,2-epoxy-3- amino-4-phenylbutan-derivaten ATE334121T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2164099		1999-01-29
JP23972099		1999-08-26

Publications (1)

Publication Number	Publication Date
ATE334121T1 true ATE334121T1 (de)	2006-08-15

Family

ID=26358729

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00901998T ATE334121T1 (de)	1999-01-29	2000-01-31	Verfahren zur herstellung von threo-1,2-epoxy-3- amino-4-phenylbutan-derivaten

Country Status (8)

Country	Link
US (1)	US6344572B1 (de)
EP (2)	EP1067125B1 (de)
AT (1)	ATE334121T1 (de)
AU (1)	AU2322600A (de)
CA (1)	CA2325919C (de)
DE (1)	DE60029517T2 (de)
ES (1)	ES2267494T3 (de)
WO (1)	WO2000044736A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR100708221B1 (ko)	1999-08-31	2007-04-17	아지노모토 가부시키가이샤	에폭사이드 결정의 제조방법
GB2369356B (en) *	2000-09-18	2004-02-04	Phoenix Chemicals Ltd	Process
JP4651178B2 (ja) *	2000-10-23	2011-03-16	三菱レイヨン株式会社	２−グリシジルオキシエチル（メタ）アクリレートの製造方法
US7122696B2 (en)	2000-11-30	2006-10-17	Ajinomoto Co., Inc.	Processes for preparation of N-protected-β-amino alcohols and N-protected-β-amino epoxides
US6764545B2 (en) *	2000-12-12	2004-07-20	Ajinomoto Co., Inc.	Production method of epoxide crystal
JP4314113B2 (ja) *	2001-07-31	2009-08-12	ウェイン・ステイト・ユニバーシティ	ヘパラン硫酸プロテオグリカンに対する標的化のための、ニューレグリンヘパリン結合ドメインとのハイブリッドタンパク質
PT1725566E (pt)	2003-12-23	2009-09-16	Tibotec Pharm Ltd	Processo para a preparação de (1s,2r)-3-[[(4-aminofenil) sulfonil](isobutil)amino]-1-benzil-2-hidroxipropilcarbamato de (3r,3as,6ar)-hexa-hidrofuro[2,3-b]furan-3-ilo
JP4818124B2 (ja)	2003-12-23	2011-11-16	テイボテク・フアーマシユーチカルズ・リミテツド	（３Ｒ，３ａＳ，６ａＲ）−ヘキサヒドロフロ〔２，３−ｂ〕フラン−３−イル（１Ｓ，１Ｒ）−３−〔〔（４−アミノフェニル）スルホニル〕（イソブチル）アミノ〕−１−ベンジル−２−ヒドロキシプロピルカルバマートの製造方法
US7582468B2 (en) *	2005-05-25	2009-09-01	Bristol-Myers Squibb Company	Process for preparing (2R,3S)-1,2-epoxy-3-(protected)amino-4-substituted butane and intermediates thereof
CN102432621B (zh)	2006-11-09	2016-02-17	爱尔兰詹森科学公司	六氢呋喃并[2,3-b]呋喃-3-醇的制备方法
WO2008132154A1 (en)	2007-04-27	2008-11-06	Tibotec Pharmaceuticals Ltd.	Methods for the preparation of n-isobutyl-n-(2-hydroxy-3-amino-4-phenylbutyl)-p-nitrobenzenesulfonylamide derivatives
MX2009013499A (es) *	2007-06-22	2010-01-18	Bristol Myers Squibb Co	Composiciones comprimidas que contienen atazanavir.
DE602008005316D1 (de) *	2007-06-22	2011-04-14	Bristol Myers Squibb Co	Tablettierte atazanavirhaltige zusammensetzungen
JP2010530892A (ja) *	2007-06-22	2010-09-16	ブリストル−マイヤーズスクイブカンパニー	アタザナビルを含む錠剤組成物
CN101778624A (zh) *	2007-06-22	2010-07-14	百时美施贵宝公司	含有阿扎那韦的压片组合物
US20110178305A1 (en) *	2008-05-08	2011-07-21	Ranbaxy Laboratories Limited	Process for the preparation of 3,4-epoxy-2-amino-1-substituted butane derivatives and intermediate compounds thereof
TWI482775B (zh)	2008-09-01	2015-05-01	Tibotec Pharm Ltd	用於製備（３ｒ，３ａｓ，６ａｒ）－六氫呋喃并〔２，３－ｂ〕呋喃－３－基（１ｓ，２ｒ）－３－〔〔（４－胺基苯基）磺醯基〕（異丁基）胺基〕－１－苯甲基－２－羥基丙基胺基甲酸酯之方法
US8921415B2 (en)	2009-01-29	2014-12-30	Mapi Pharma Ltd.	Polymorphs of darunavir
EP2528923B1 (de)	2010-01-28	2014-07-30	Mapi Pharma Limited	Verfahren zur herstellung von darunavir und darunavir-zwischenprodukten

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH07504654A (ja) *	1992-03-11	1995-05-25	ナルヘックス　リミテッド	オキソ及びヒドロキシ置換炭化水素のアミン誘導体
US5559256A (en) *	1992-07-20	1996-09-24	E. R. Squibb & Sons, Inc.	Aminediol protease inhibitors
US5481011A (en) *	1994-12-13	1996-01-02	Bristol-Myers Squibb Company	Process for preparing N-protected amino acid α-halomethyl ketones and alcohols from N-protected amino acid esters
DE69616446T2 (de) *	1995-02-03	2002-05-16	Kaneka Corp., Osaka	Verfahren zur herstellung von alpha-haloketonen, alpha-halohydrinen und epoxiden
US5767316A (en) *	1995-11-17	1998-06-16	Ajinomoto Co., Inc.	Process for producing 3-amino-2-oxo-1-halogenopropane derivatives
JPH09323960A (ja) *	1996-06-05	1997-12-16	Ajinomoto Co Inc	３−アミノ−１，２−オキシランの製造方法

2000
- 2000-01-31 AU AU23226/00A patent/AU2322600A/en not_active Abandoned
- 2000-01-31 EP EP00901998A patent/EP1067125B1/de not_active Expired - Lifetime
- 2000-01-31 ES ES00901998T patent/ES2267494T3/es not_active Expired - Lifetime
- 2000-01-31 US US09/647,340 patent/US6344572B1/en not_active Expired - Lifetime
- 2000-01-31 AT AT00901998T patent/ATE334121T1/de not_active IP Right Cessation
- 2000-01-31 EP EP06110625A patent/EP1661893A3/de not_active Withdrawn
- 2000-01-31 DE DE60029517T patent/DE60029517T2/de not_active Expired - Lifetime
- 2000-01-31 WO PCT/JP2000/000495 patent/WO2000044736A1/ja not_active Ceased
- 2000-01-31 CA CA002325919A patent/CA2325919C/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US6344572B1 (en)	2002-02-05
CA2325919A1 (en)	2000-08-03
WO2000044736A1 (en)	2000-08-03
EP1067125B1 (de)	2006-07-26
DE60029517T2 (de)	2006-11-23
CA2325919C (en)	2009-07-21
DE60029517D1 (de)	2006-09-07
EP1661893A2 (de)	2006-05-31
ES2267494T3 (es)	2007-03-16
EP1067125A4 (de)	2004-06-16
AU2322600A (en)	2000-08-18
EP1661893A3 (de)	2006-06-07
EP1067125A1 (de)	2001-01-10

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Legal Events

Date	Code	Title	Description
2007-01-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties