ATE334679T1 - Feste oral anzuwendende arzneizubereitung mit gesteuerter wirkstoffabgabe enthaltend eine säureempfindliche benzimidazolverbindung - Google Patents

Feste oral anzuwendende arzneizubereitung mit gesteuerter wirkstoffabgabe enthaltend eine säureempfindliche benzimidazolverbindung

Info

Publication number
ATE334679T1
ATE334679T1 AT00500203T AT00500203T ATE334679T1 AT E334679 T1 ATE334679 T1 AT E334679T1 AT 00500203 T AT00500203 T AT 00500203T AT 00500203 T AT00500203 T AT 00500203T AT E334679 T1 ATE334679 T1 AT E334679T1
Authority
AT
Austria
Prior art keywords
acid
solid oral
medicinal preparation
benzimidazole compound
active release
Prior art date
Application number
AT00500203T
Other languages
English (en)
Inventor
Cabrera Antonio Lopez
Vincent Mancinelli
Ibarra Pedro Juan Solanas
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Application granted granted Critical
Publication of ATE334679T1 publication Critical patent/ATE334679T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
AT00500203T 1999-09-13 2000-09-13 Feste oral anzuwendende arzneizubereitung mit gesteuerter wirkstoffabgabe enthaltend eine säureempfindliche benzimidazolverbindung ATE334679T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES009902027A ES2168043B1 (es) 1999-09-13 1999-09-13 Forma farmaceutica solida oral de liberacion modificada que contiene un compuesto de bencimidazol labil en medio acido.

Publications (1)

Publication Number Publication Date
ATE334679T1 true ATE334679T1 (de) 2006-08-15

Family

ID=8309905

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00500203T ATE334679T1 (de) 1999-09-13 2000-09-13 Feste oral anzuwendende arzneizubereitung mit gesteuerter wirkstoffabgabe enthaltend eine säureempfindliche benzimidazolverbindung

Country Status (12)

Country Link
US (1) US6780436B1 (de)
EP (1) EP1086694B1 (de)
JP (1) JP4885347B2 (de)
KR (1) KR100724201B1 (de)
AT (1) ATE334679T1 (de)
AU (1) AU777322B2 (de)
CA (1) CA2318008C (de)
CY (1) CY1106219T1 (de)
DE (1) DE60029712T2 (de)
DK (1) DK1086694T3 (de)
ES (2) ES2168043B1 (de)
PT (1) PT1086694E (de)

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CN104586809A (zh) * 2015-01-08 2015-05-06 浙江亚太药业股份有限公司 一种埃索美拉唑镁微丸肠溶片及制备方法
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WO2017145146A1 (en) 2016-02-25 2017-08-31 Dexcel Pharma Technologies Ltd. Compositions comprising proton pump inhibitors
US10076494B2 (en) 2016-06-16 2018-09-18 Dexcel Pharma Technologies Ltd. Stable orally disintegrating pharmaceutical compositions
PT3512530T (pt) * 2016-09-15 2021-01-13 Stichting Het Nederlands Kanker Inst Antoni Van Leeuwenhoek Ziekenhuis Pirofosfato oral para utilização na redução de calcificação de tecido
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Also Published As

Publication number Publication date
DK1086694T3 (da) 2006-12-04
KR100724201B1 (ko) 2007-05-31
DE60029712D1 (de) 2006-09-14
PT1086694E (pt) 2006-12-29
DE60029712T2 (de) 2007-08-02
AU5791900A (en) 2001-03-15
US6780436B1 (en) 2004-08-24
CA2318008A1 (en) 2001-03-13
EP1086694A2 (de) 2001-03-28
EP1086694A3 (de) 2002-09-25
JP2001199878A (ja) 2001-07-24
EP1086694B1 (de) 2006-08-02
CY1106219T1 (el) 2011-06-08
CA2318008C (en) 2010-08-17
ES2269088T3 (es) 2007-04-01
AU777322B2 (en) 2004-10-14
JP4885347B2 (ja) 2012-02-29
ES2168043B1 (es) 2003-04-01
KR20020020974A (ko) 2002-03-18
ES2168043A1 (es) 2002-05-16

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