ATE345329T1 - Pyridinderivate als modulatoren des cb2-rezeptors - Google Patents

Pyridinderivate als modulatoren des cb2-rezeptors

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Publication number
ATE345329T1
ATE345329T1 AT03798193T AT03798193T ATE345329T1 AT E345329 T1 ATE345329 T1 AT E345329T1 AT 03798193 T AT03798193 T AT 03798193T AT 03798193 T AT03798193 T AT 03798193T AT E345329 T1 ATE345329 T1 AT E345329T1
Authority
AT
Austria
Prior art keywords
pyridine derivatives
receptor
modulators
diseases
indirectly
Prior art date
Application number
AT03798193T
Other languages
English (en)
Inventor
Andrew John Eatherton
Gerard Martin Paul Giblin
Richard Howard Green
Karamjit Singh Jandu
William Leonard Mitchell
Alan Naylor
Giovanni Palombi
Bollate
Derek Anthony Rawlings
Brian Peter Slingsby
Andrew Richard Whittington
Road Wood
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE345329T1 publication Critical patent/ATE345329T1/de

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
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AT03798193T 2002-09-27 2003-09-25 Pyridinderivate als modulatoren des cb2-rezeptors ATE345329T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0222495.4A GB0222495D0 (en) 2002-09-27 2002-09-27 Compounds

Publications (1)

Publication Number Publication Date
ATE345329T1 true ATE345329T1 (de) 2006-12-15

Family

ID=9944906

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03798193T ATE345329T1 (de) 2002-09-27 2003-09-25 Pyridinderivate als modulatoren des cb2-rezeptors

Country Status (9)

Country Link
US (1) US20070129367A1 (de)
EP (1) EP1562907B1 (de)
JP (1) JP2006508065A (de)
AT (1) ATE345329T1 (de)
AU (1) AU2003276028A1 (de)
DE (1) DE60309739T2 (de)
ES (1) ES2277149T3 (de)
GB (1) GB0222495D0 (de)
WO (1) WO2004029027A1 (de)

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UY27939A1 (es) 2002-08-21 2004-03-31 Glaxo Group Ltd Compuestos
TW200505902A (en) * 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
US7932272B2 (en) 2003-09-30 2011-04-26 Eisai R&D Management Co., Ltd. Antifungal agent containing heterocyclic compound
GB0402357D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402356D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402355D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
WO2006106711A1 (ja) 2005-03-30 2006-10-12 Eisai R & D Management Co., Ltd. ピリジン誘導体を含有する抗真菌剤
WO2006129609A1 (ja) * 2005-05-30 2006-12-07 Shionogi & Co., Ltd. ２－ナフチルイミノ－５，５－ジ置換－１，３－チアジン誘導体
TWI385169B (zh) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
US20090275611A1 (en) * 2006-04-07 2009-11-05 Boehringer Ingelheim International Gmbh Compounds Which Modulate The CB2 Receptor
CA2657247A1 (en) 2006-07-28 2008-01-31 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
WO2008035726A1 (en) 2006-09-21 2008-03-27 Eisai R & D Management Co., Ltd. Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same
WO2008039645A1 (en) 2006-09-25 2008-04-03 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
FR2907784B1 (fr) * 2006-10-27 2009-02-13 Sod Conseils Rech Applic Derives phenyliques et leur utilisation comme medicament
EP2139852A1 (de) 2006-12-19 2010-01-06 Pharmos Corporation Sulfonamidderivate mit therapeutischen indikationen
TW200841879A (en) 2007-04-27 2008-11-01 Eisai R&D Man Co Ltd Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
EP2143723A4 (de) 2007-04-27 2011-05-18 Eisai R&D Man Co Ltd Salz eines heterocyclus-substituierten pyridinderivats oder kristall davon
JP5300225B2 (ja) 2007-08-03 2013-09-25 バイエル・クロップサイエンス・アーゲー 除草剤トリアゾリルピリジンケトン類
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JP2006508065A (ja) 2006-03-09
AU2003276028A1 (en) 2004-04-19
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US20070129367A1 (en) 2007-06-07
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