ATE349459T1 - Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters - Google Patents

Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters

Info

Publication number: ATE349459T1
Authority: AT; Austria
Prior art keywords: ntrenyl; dodecahydrocyclopenta; polymorpho; phen; ester
Prior art date: 2002-07-29

Application number

AT03766325T

Other languages

English (en)

Inventor

Guido Jordine

Michael Mutz

Original Assignee

Novartis Pharma Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-07-29

Filing date

2003-07-28

Publication date

2007-01-15

2003-07-28 Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh

2007-01-15 Application granted granted Critical

2007-01-15 Publication of ATE349459T1 publication Critical patent/ATE349459T1/de

Links

YNPNZTXNASCQKK-UHFFFAOYSA-N Phenanthrene Natural products C1=CC=C2C3=CC=CC=C3C=CC2=C1 YNPNZTXNASCQKK-UHFFFAOYSA-N 0.000 title 1
DGEZNRSVGBDHLK-UHFFFAOYSA-N [1,10]phenanthroline Chemical compound C1=CN=C2C3=NC=CC=C3C=CC2=C1 DGEZNRSVGBDHLK-UHFFFAOYSA-N 0.000 title 1
150000002148 esters Chemical class 0.000 title 1
QERYCTSHXKAMIS-UHFFFAOYSA-N thiophene-2-carboxylic acid Chemical compound OC(=O)C1=CC=CS1 QERYCTSHXKAMIS-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pulmonology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Steroid Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT03766325T 2002-07-29 2003-07-28 Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters ATE349459T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0217504.0A GB0217504D0 (en)	2002-07-29	2002-07-29	Organic compounds

Publications (1)

Publication Number	Publication Date
ATE349459T1 true ATE349459T1 (de)	2007-01-15

Family

ID=9941275

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03766325T ATE349459T1 (de)	2002-07-29	2003-07-28	Polymorph b eines bekannten thiophencarbonsäuredodecahydrocyclopenta(a)phen ntrenylesters

Country Status (30)

Country	Link
US (1)	US7683048B2 (de)
EP (2)	EP1676854A1 (de)
JP (1)	JP2006501207A (de)
KR (1)	KR100688371B1 (de)
CN (1)	CN1305892C (de)
AR (1)	AR040692A1 (de)
AT (1)	ATE349459T1 (de)
AU (1)	AU2003251651B2 (de)
BR (1)	BR0313044A (de)
CA (1)	CA2493330C (de)
CY (1)	CY1106406T1 (de)
DE (1)	DE60310747T2 (de)
DK (1)	DK1554303T3 (de)
EC (1)	ECSP055579A (de)
ES (1)	ES2279970T3 (de)
GB (1)	GB0217504D0 (de)
HK (1)	HK1080484B (de)
IL (2)	IL166287A0 (de)
MX (1)	MXPA05001173A (de)
MY (1)	MY136407A (de)
NO (1)	NO20050806L (de)
NZ (2)	NZ537868A (de)
PE (1)	PE20040722A1 (de)
PL (1)	PL209409B1 (de)
PT (1)	PT1554303E (de)
RU (2)	RU2348646C1 (de)
SI (1)	SI1554303T1 (de)
TW (1)	TWI309164B (de)
WO (1)	WO2004013156A1 (de)
ZA (1)	ZA200500370B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0019172D0 (en)	2000-08-05	2000-09-27	Glaxo Group Ltd	Novel compounds
PT1305329E (pt)	2000-08-05	2007-12-24	Glaxo Group Ltd	Éster s-fluorometílico do ácido 6.alfa.,9.alfa.-difluoro- 17.alfa.-(2-furanilcarboxil)oxi-11.beta.-hidroxi-16.alfa.-metil- 3-oxo-androsta-1,4-dieno-17-carbotióico como um agente antiinflamatório
US6777399B2 (en)	2000-08-05	2004-08-17	Smithkline Beecham Corporation	Anti-inflammatory androstane derivative compositions
US6858596B2 (en)	2000-08-05	2005-02-22	Smithkline Beecham Corporation	Formulation containing anti-inflammatory androstane derivative
MY137522A (en)	2001-04-30	2009-02-27	Glaxo Group Ltd	Novel anti-inflammatory androstane derivatives.
GB2389530B (en)	2002-06-14	2007-01-10	Cipla Ltd	Pharmaceutical compositions
GB0523656D0 (en) *	2005-11-21	2005-12-28	Novartis Ag	Organic compounds
GB0523654D0 (en) *	2005-11-21	2005-12-28	Novartis Ag	Organic compounds
GB0603783D0 (en) *	2006-02-24	2006-04-05	Novartis Ag	Organic compounds
JP2011513203A (ja) *	2008-03-14	2011-04-28	大塚製薬株式会社	Ｍｍｐ−２及び／又はｍｍｐ−９阻害剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU550939A1 (ru) *	1975-05-19	1994-07-15	Институт химии древесины АН ЛатвССР	1,2,3,4,4а,4в,5,6,10,10а -декагидро -6- хлорацетоксиметил -1,4а-диметил -7- (1-метилэтил) -1- фенантренкарбоновая кислота или ее соли
JPH08291073A (ja) *	1995-04-22	1996-11-05	Kissei Pharmaceut Co Ltd	医薬品組成物及びその製造方法
GB0015876D0 (en) *	2000-06-28	2000-08-23	Novartis Ag	Organic compounds

2002
- 2002-07-29 GB GBGB0217504.0A patent/GB0217504D0/en not_active Ceased
2003
- 2003-07-25 PE PE2003000741A patent/PE20040722A1/es not_active Application Discontinuation
- 2003-07-25 AR AR20030102680A patent/AR040692A1/es unknown
- 2003-07-28 PL PL373140A patent/PL209409B1/pl not_active IP Right Cessation
- 2003-07-28 NZ NZ537868A patent/NZ537868A/en unknown
- 2003-07-28 TW TW092120513A patent/TWI309164B/zh not_active IP Right Cessation
- 2003-07-28 MY MYPI20032832A patent/MY136407A/en unknown
- 2003-07-28 DK DK03766325T patent/DK1554303T3/da active
- 2003-07-28 JP JP2004525343A patent/JP2006501207A/ja active Pending
- 2003-07-28 SI SI200330721T patent/SI1554303T1/sl unknown
- 2003-07-28 DE DE60310747T patent/DE60310747T2/de not_active Expired - Lifetime
- 2003-07-28 EP EP06005390A patent/EP1676854A1/de not_active Withdrawn
- 2003-07-28 PT PT03766325T patent/PT1554303E/pt unknown
- 2003-07-28 RU RU2007143025/04A patent/RU2348646C1/ru not_active IP Right Cessation
- 2003-07-28 EP EP03766325A patent/EP1554303B1/de not_active Expired - Lifetime
- 2003-07-28 CA CA2493330A patent/CA2493330C/en not_active Expired - Fee Related
- 2003-07-28 US US10/522,358 patent/US7683048B2/en not_active Expired - Fee Related
- 2003-07-28 MX MXPA05001173A patent/MXPA05001173A/es active IP Right Grant
- 2003-07-28 KR KR1020057001581A patent/KR100688371B1/ko not_active Expired - Fee Related
- 2003-07-28 HK HK06100247.5A patent/HK1080484B/en not_active IP Right Cessation
- 2003-07-28 AT AT03766325T patent/ATE349459T1/de active
- 2003-07-28 AU AU2003251651A patent/AU2003251651B2/en not_active Ceased
- 2003-07-28 BR BR0313044-4A patent/BR0313044A/pt not_active IP Right Cessation
- 2003-07-28 ES ES03766325T patent/ES2279970T3/es not_active Expired - Lifetime
- 2003-07-28 RU RU2005105688/04A patent/RU2330043C2/ru not_active IP Right Cessation
- 2003-07-28 NZ NZ549713A patent/NZ549713A/en unknown
- 2003-07-28 WO PCT/EP2003/008314 patent/WO2004013156A1/en not_active Ceased
- 2003-07-28 CN CNB038180596A patent/CN1305892C/zh not_active Expired - Fee Related
2005
- 2005-01-13 IL IL16628705A patent/IL166287A0/xx unknown
- 2005-01-14 ZA ZA200500370A patent/ZA200500370B/en unknown
- 2005-01-26 EC EC2005005579A patent/ECSP055579A/es unknown
- 2005-02-15 NO NO20050806A patent/NO20050806L/no unknown
2007
- 2007-03-22 CY CY20071100400T patent/CY1106406T1/el unknown
- 2007-07-26 IL IL184848A patent/IL184848A0/en unknown

Also Published As

Publication number	Publication date
EP1554303A1 (de)	2005-07-20
HK1080484A1 (en)	2006-04-28
RU2348646C1 (ru)	2009-03-10
NO20050806L (no)	2005-02-15
GB0217504D0 (en)	2002-09-04
EP1676854A1 (de)	2006-07-05
SI1554303T1 (sl)	2007-06-30
TW200401633A (en)	2004-02-01
HK1080484B (en)	2007-08-03
CY1106406T1 (el)	2011-10-12
PE20040722A1 (es)	2004-11-29
MXPA05001173A (es)	2005-05-16
ECSP055579A (es)	2005-04-18
AU2003251651B2 (en)	2007-07-12
CN1671731A (zh)	2005-09-21
ZA200500370B (en)	2006-07-26
ES2279970T3 (es)	2007-09-01
DE60310747T2 (de)	2007-10-11
BR0313044A (pt)	2005-06-14
DK1554303T3 (da)	2007-04-30
US20060166954A1 (en)	2006-07-27
CA2493330C (en)	2011-08-23
RU2330043C2 (ru)	2008-07-27
RU2005105688A (ru)	2005-10-10
KR20050033632A (ko)	2005-04-12
KR100688371B1 (ko)	2007-03-02
CN1305892C (zh)	2007-03-21
EP1554303B1 (de)	2006-12-27
JP2006501207A (ja)	2006-01-12
RU2007143025A (ru)	2009-01-20
AU2003251651A1 (en)	2004-02-23
TWI309164B (en)	2009-05-01
NZ537868A (en)	2006-11-30
PL209409B1 (pl)	2011-08-31
IL184848A0 (en)	2007-12-03
PL373140A1 (en)	2005-08-22
DE60310747D1 (en)	2007-02-08
NZ549713A (en)	2008-04-30
CA2493330A1 (en)	2004-02-12
IL166287A0 (en)	2006-01-15
MY136407A (en)	2008-09-30
US7683048B2 (en)	2010-03-23
WO2004013156A1 (en)	2004-02-12
PT1554303E (pt)	2007-03-30
AR040692A1 (es)	2005-04-13

Legal Events

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Title

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2007-07-15

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