ATE350102T1 - 7-amino-2-alkylthiopteridin-4-yl-amine zur behandlung von chemokinassoziierten erkrankungen - Google Patents

7-amino-2-alkylthiopteridin-4-yl-amine zur behandlung von chemokinassoziierten erkrankungen

Info

Publication number
ATE350102T1
ATE350102T1 AT01977001T AT01977001T ATE350102T1 AT E350102 T1 ATE350102 T1 AT E350102T1 AT 01977001 T AT01977001 T AT 01977001T AT 01977001 T AT01977001 T AT 01977001T AT E350102 T1 ATE350102 T1 AT E350102T1
Authority
AT
Austria
Prior art keywords
diseases
treatment
psoriasis
compounds
skin
Prior art date
Application number
AT01977001T
Other languages
English (en)
Inventor
Roger Bonnert
Iain Walters
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of ATE350102T1 publication Critical patent/ATE350102T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT01977001T 2000-10-20 2001-10-16 7-amino-2-alkylthiopteridin-4-yl-amine zur behandlung von chemokinassoziierten erkrankungen ATE350102T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0003828A SE0003828D0 (sv) 2000-10-20 2000-10-20 Novel compounds

Publications (1)

Publication Number Publication Date
ATE350102T1 true ATE350102T1 (de) 2007-01-15

Family

ID=20281519

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01977001T ATE350102T1 (de) 2000-10-20 2001-10-16 7-amino-2-alkylthiopteridin-4-yl-amine zur behandlung von chemokinassoziierten erkrankungen

Country Status (9)

Country Link
US (1) US7071193B2 (de)
EP (1) EP1328319B1 (de)
JP (1) JP4250416B2 (de)
AT (1) ATE350102T1 (de)
AU (1) AU2001296151A1 (de)
DE (1) DE60125801T2 (de)
ES (1) ES2276836T3 (de)
SE (1) SE0003828D0 (de)
WO (1) WO2002032507A1 (de)

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SE9903544D0 (sv) * 1999-10-01 1999-10-01 Astra Pharma Prod Novel compounds
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ATE369861T1 (de) * 2003-09-12 2007-09-15 4 Aza Ip Nv Pteridin-derivate zur behandlung von erkrankungen im zusammenhang mit tnf-alpha
US20070032477A1 (en) * 2003-10-17 2007-02-08 Waer Mark J A Pteridine derivatives useful for making pharmaceutical compositions
DE602004008312T2 (de) * 2003-10-17 2008-04-17 4 Aza Ip Nv Heterocyclus-substituierte pteridin-derivate und ihre verwendung in der therapie
GB0328243D0 (en) * 2003-12-05 2004-01-07 Astrazeneca Ab Methods
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WO2016029077A1 (en) * 2014-08-22 2016-02-25 Janus Biotherapeutics, Inc. Novel n2, n4, n7, 6-tetrasubstituted pteridine-2,4,7-triamine and 2, 4, 6, 7-tetrasubstituted pteridine compounds and methods of synthesis and use thereof
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TW202212339A (zh) 2019-04-17 2022-04-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
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Also Published As

Publication number Publication date
JP4250416B2 (ja) 2009-04-08
SE0003828D0 (sv) 2000-10-20
WO2002032507A1 (en) 2002-04-25
DE60125801T2 (de) 2007-10-11
JP2004511532A (ja) 2004-04-15
AU2001296151A1 (en) 2002-04-29
DE60125801D1 (de) 2007-02-15
EP1328319A1 (de) 2003-07-23
EP1328319B1 (de) 2007-01-03
ES2276836T3 (es) 2007-07-01
US7071193B2 (en) 2006-07-04
US20040102447A1 (en) 2004-05-27

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