ATE483721T1 - In 4''- bzw. 4'-position substituierte avermectine mit pestiziden eigenschaften - Google Patents

In 4''- bzw. 4'-position substituierte avermectine mit pestiziden eigenschaften

Info

Publication number
ATE483721T1
ATE483721T1 AT04707515T AT04707515T ATE483721T1 AT E483721 T1 ATE483721 T1 AT E483721T1 AT 04707515 T AT04707515 T AT 04707515T AT 04707515 T AT04707515 T AT 04707515T AT E483721 T1 ATE483721 T1 AT E483721T1
Authority
AT
Austria
Prior art keywords
position substituted
pesticidal properties
substituted avermectins
avermectins
pesticidal
Prior art date
Application number
AT04707515T
Other languages
English (en)
Inventor
Jerome Cassayre
Hans Tobler
Thomas Pitterna
Peter Maienfisch
Kessabi Fiona Murphy
Laura Quaranta
Ottmar Franz Hueter
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Application granted granted Critical
Publication of ATE483721T1 publication Critical patent/ATE483721T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT04707515T 2003-02-04 2004-02-03 In 4''- bzw. 4'-position substituierte avermectine mit pestiziden eigenschaften ATE483721T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0302548.3A GB0302548D0 (en) 2003-02-04 2003-02-04 Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
PCT/EP2004/000972 WO2004069852A1 (en) 2003-02-04 2004-02-03 Avermectins substituted in the 4” and 4’-positions having pesticidal properties

Publications (1)

Publication Number Publication Date
ATE483721T1 true ATE483721T1 (de) 2010-10-15

Family

ID=9952416

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04707515T ATE483721T1 (de) 2003-02-04 2004-02-03 In 4''- bzw. 4'-position substituierte avermectine mit pestiziden eigenschaften

Country Status (11)

Country Link
US (1) US7378399B2 (de)
EP (1) EP1613639B1 (de)
JP (1) JP2006516590A (de)
AR (1) AR043005A1 (de)
AT (1) ATE483721T1 (de)
CL (1) CL2004000160A1 (de)
DE (1) DE602004029452D1 (de)
ES (1) ES2349531T3 (de)
GB (1) GB0302548D0 (de)
TW (1) TW200510444A (de)
WO (1) WO2004069852A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) * 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR040073A1 (es) * 2002-05-07 2005-03-16 Syngenta Participations Ag Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas
GB0302308D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
TWI422328B (zh) * 2006-06-19 2014-01-11 Univ California 結合有殺線蟲之種子塗覆物的生物控制劑
TW201309639A (zh) * 2011-02-17 2013-03-01 Lg Life Sciences Ltd 作為gpr119促效劑之肟衍生物
CN105017358B (zh) * 2015-07-31 2018-07-10 内蒙古嘉宝仕生物科技股份有限公司 一种合成甲胺基阿维菌素苯甲酸盐的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2636880B2 (ja) * 1987-04-29 1997-07-30 三共株式会社 効力の増強された農業用殺虫殺ダニ剤
GB2220856A (en) * 1988-07-18 1990-01-24 Merck & Co Inc Novel synergistic agricultural insecticidal and acaricidal combinations containing avermectin derivatives
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas

Also Published As

Publication number Publication date
EP1613639A1 (de) 2006-01-11
DE602004029452D1 (de) 2010-11-18
WO2004069852A1 (en) 2004-08-19
CL2004000160A1 (es) 2005-01-14
TW200510444A (en) 2005-03-16
GB0302548D0 (en) 2003-03-12
ES2349531T3 (es) 2011-01-04
EP1613639B1 (de) 2010-10-06
AR043005A1 (es) 2005-07-13
US20060154879A1 (en) 2006-07-13
US7378399B2 (en) 2008-05-27
JP2006516590A (ja) 2006-07-06

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Legal Events

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