ATE397930T1 - Verwendung von oxazolidinon-chinolin-hybrid- antibiotika zur behandlung von anthrax und anderen infektionen - Google Patents

Verwendung von oxazolidinon-chinolin-hybrid- antibiotika zur behandlung von anthrax und anderen infektionen

Info

Publication number
ATE397930T1
ATE397930T1 AT04725909T AT04725909T ATE397930T1 AT E397930 T1 ATE397930 T1 AT E397930T1 AT 04725909 T AT04725909 T AT 04725909T AT 04725909 T AT04725909 T AT 04725909T AT E397930 T1 ATE397930 T1 AT E397930T1
Authority
AT
Austria
Prior art keywords
oxazolidinone
infections
hybrid antibiotics
anthrax
quinoline
Prior art date
Application number
AT04725909T
Other languages
English (en)
Inventor
Christian Hubschwerlen
Jean-Luc Specklin
Daniel Baeschlin
Hans Locher
Christine Sigwalt
Original Assignee
Morphochem Ag Komb Chemie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Morphochem Ag Komb Chemie filed Critical Morphochem Ag Komb Chemie
Application granted granted Critical
Publication of ATE397930T1 publication Critical patent/ATE397930T1/de

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT04725909T 2003-04-30 2004-04-06 Verwendung von oxazolidinon-chinolin-hybrid- antibiotika zur behandlung von anthrax und anderen infektionen ATE397930T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46694503P 2003-04-30 2003-04-30
US53082203P 2003-12-18 2003-12-18

Publications (1)

Publication Number Publication Date
ATE397930T1 true ATE397930T1 (de) 2008-07-15

Family

ID=33423632

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04725909T ATE397930T1 (de) 2003-04-30 2004-04-06 Verwendung von oxazolidinon-chinolin-hybrid- antibiotika zur behandlung von anthrax und anderen infektionen

Country Status (15)

Country Link
US (3) US20070155714A1 (de)
EP (1) EP1620098B1 (de)
JP (2) JP4805139B2 (de)
KR (1) KR101101982B1 (de)
AT (1) ATE397930T1 (de)
AU (2) AU2004233557B2 (de)
BR (1) BRPI0409955A (de)
CA (1) CA2529347C (de)
DE (1) DE602004014361D1 (de)
ES (1) ES2308171T3 (de)
IL (1) IL171546A (de)
MX (1) MXPA05011654A (de)
NZ (1) NZ543757A (de)
RU (1) RU2351335C2 (de)
WO (1) WO2004096221A1 (de)

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CA2549675C (en) † 2003-12-18 2012-11-20 Morphochem Aktiengesellschaft Fur Kombinatorische Chemie Oxazolidinone-quinolone hybrid antibiotics
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JP5796412B2 (ja) 2011-08-26 2015-10-21 三菱電機株式会社 半導体素子の製造方法
JP6030146B2 (ja) * 2011-11-08 2016-11-24 アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ ２−オキソ−オキサゾリジン−３，５−ジイル抗生物質誘導体
CN105025929A (zh) 2013-03-08 2015-11-04 阿勒根公司 环孢菌素a-类固醇缀合物
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CN105246476B (zh) * 2013-05-28 2019-11-15 莫弗凯姆联合化学股份公司 含噁唑烷酮-喹诺酮的联合疗法在治疗细菌感染中的应用
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DE10340485B4 (de) * 2003-09-03 2015-05-13 Morphochem AG Aktiengesellschaft für kombinatorische Chemie Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden
CA2549675C (en) 2003-12-18 2012-11-20 Morphochem Aktiengesellschaft Fur Kombinatorische Chemie Oxazolidinone-quinolone hybrid antibiotics
AR054608A1 (es) 2005-08-08 2007-06-27 Actelion Pharmaceuticals Ltd Derivados de oxazolidinona enlazados a quinolonas como antibacterianos
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ATE544764T1 (de) 2006-11-10 2012-02-15 Actelion Pharmaceuticals Ltd 5-hydroxymethyloxazolidin-2-onderivate
CL2007003332A1 (es) 2006-11-24 2008-06-20 Actelion Pharmaceuticals Ltd Compuestos derivados de heterociclos condensados; compuestos intermediarios; composicion farmaceutica; y uso en la prevencion o tratamiento de infecciones bacterianas.
RU2527769C2 (ru) 2008-05-09 2014-09-10 Актелион Фармасьютиклз Лтд Производные 5-гидроксиметилоксазолидин-2-она для лечения бактериальных кишечных заболеваний

Also Published As

Publication number Publication date
JP4805139B2 (ja) 2011-11-02
BRPI0409955A (pt) 2006-04-25
US20070155714A1 (en) 2007-07-05
WO2004096221A1 (en) 2004-11-11
JP5536706B2 (ja) 2014-07-02
DE602004014361D1 (de) 2008-07-24
MXPA05011654A (es) 2005-12-15
US8513231B2 (en) 2013-08-20
AU2010201659A1 (en) 2010-05-20
US20120135961A1 (en) 2012-05-31
RU2351335C2 (ru) 2009-04-10
US8268812B2 (en) 2012-09-18
JP2011184441A (ja) 2011-09-22
US20120322766A1 (en) 2012-12-20
NZ543757A (en) 2009-02-28
EP1620098A1 (de) 2006-02-01
HK1078806A1 (en) 2006-03-24
IL171546A (en) 2014-06-30
CA2529347C (en) 2011-09-06
CA2529347A1 (en) 2004-11-11
EP1620098B1 (de) 2008-06-11
KR101101982B1 (ko) 2012-01-02
KR20060025525A (ko) 2006-03-21
AU2004233557A1 (en) 2004-11-11
RU2005137032A (ru) 2007-06-10
AU2004233557B2 (en) 2010-02-18
ES2308171T3 (es) 2008-12-01
JP2006526577A (ja) 2006-11-24

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