ATE414070T1 - Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen - Google Patents

Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen

Info

Publication number
ATE414070T1
ATE414070T1 AT01272539T AT01272539T ATE414070T1 AT E414070 T1 ATE414070 T1 AT E414070T1 AT 01272539 T AT01272539 T AT 01272539T AT 01272539 T AT01272539 T AT 01272539T AT E414070 T1 ATE414070 T1 AT E414070T1
Authority
AT
Austria
Prior art keywords
optically active
dihydrobenzofuran
optionally substituted
dihydrobenzofuran compounds
producing optically
Prior art date
Application number
AT01272539T
Other languages
English (en)
Inventor
Isao Aoki
Mari Adachi
Hiroyuki Tawada
Makoto Yamashita
Misayo Sera
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Application granted granted Critical
Publication of ATE414070T1 publication Critical patent/ATE414070T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
    • C07F9/6574—Esters of oxyacids of phosphorus
    • C07F9/65742—Esters of oxyacids of phosphorus non-condensed with carbocyclic rings or heterocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
AT01272539T 2000-12-28 2001-12-27 Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen ATE414070T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2000400531 2000-12-28

Publications (1)

Publication Number Publication Date
ATE414070T1 true ATE414070T1 (de) 2008-11-15

Family

ID=18865111

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01272539T ATE414070T1 (de) 2000-12-28 2001-12-27 Verfahren zur herstellung von optisch aktiven 2,4-dihydrobenzofuranverbindungen

Country Status (7)

Country Link
US (2) US6878831B2 (de)
EP (1) EP1346988B1 (de)
AT (1) ATE414070T1 (de)
CA (1) CA2432410A1 (de)
DE (1) DE60136566D1 (de)
ES (1) ES2312399T3 (de)
WO (1) WO2002053551A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003074046A1 (en) * 2002-03-01 2003-09-12 Takeda Chemical Industries, Ltd. Antidepressant
JP4227061B2 (ja) * 2004-03-30 2009-02-18 シャープ株式会社 アミン化合物、該アミン化合物を用いた電子写真感光体およびそれを備える画像形成装置
WO2006022311A1 (ja) * 2004-08-27 2006-03-02 Takeda Pharmaceutical Company Limited アゾ化合物とその製造方法
CA2668864A1 (en) * 2006-11-09 2008-05-15 Takeda Pharmaceutical Company Limited Pharmaceutical composition comprising a dihydrobenzofuranyl isoindoline and a lipophilic component
US8604242B2 (en) 2008-10-13 2013-12-10 Interquim, S.A. Process for the preparation of optically active (S)-(−)-2-(N-propylamino)-5-methoxytetraline and (S)-(−)-2-(N-propylamino)-5-hydroxytetraline compounds
CN105384710B (zh) * 2015-11-04 2017-11-10 重庆天春科技有限公司 一种药物中间体呋喃类化合物的合成方法
CN105330621B (zh) * 2015-11-04 2017-11-10 重庆天春科技有限公司 一种呋喃酯类化合物的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8403224A (nl) * 1984-10-24 1986-05-16 Oce Andeno Bv Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen.
TW199152B (de) * 1990-11-01 1993-02-01 Takeda Pharm Industry Co Ltd
US6479536B1 (en) 1998-12-04 2002-11-12 Takeda Chemical Industries, Ltd. Benzofuran derivatives, process for the preparation of the same and uses thereof
WO2001030763A1 (en) 1999-10-22 2001-05-03 Takeda Chemical Industries, Ltd. Process for producing optically active naphthalene derivative and optical resolver therefor

Also Published As

Publication number Publication date
US7420070B2 (en) 2008-09-02
DE60136566D1 (de) 2008-12-24
CA2432410A1 (en) 2002-07-11
US20040077712A1 (en) 2004-04-22
EP1346988A4 (de) 2004-03-17
WO2002053551A1 (en) 2002-07-11
EP1346988A1 (de) 2003-09-24
US6878831B2 (en) 2005-04-12
EP1346988B1 (de) 2008-11-12
US20050171184A1 (en) 2005-08-04
ES2312399T3 (es) 2009-03-01

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