ATE414695T1 - 8-chlor-2,3-benzodiazepinderivate - Google Patents

8-chlor-2,3-benzodiazepinderivate

Info

Publication number: ATE414695T1
Authority: AT; Austria
Prior art keywords: benzodiazepine derivatives; new; chloro; stands; preparation
Prior art date: 2003-08-04

Application number

AT04769081T

Other languages

English (en)

Inventor

Jozsef Barkoczy

Istvan Ling

Gyula Simig

Gabor Szenasi

Gabor Gigler

Szabolcs Kertesz

Gyula Szuecs

Geza Szabo

Miklos Vegh

Laszlo Harsing

Original Assignee

Egyt Gyogyszervegyeszeti Gyar

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-08-04

Filing date

2004-07-29

Publication date

2008-12-15

2004-07-29 Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar

2008-12-15 Application granted granted Critical

2008-12-15 Publication of ATE414695T1 publication Critical patent/ATE414695T1/de

Links

CKISTXXLRVRADV-UHFFFAOYSA-N C1=NNC=C2C=C(Cl)C=CC2=C1 Chemical class C1=NNC=C2C=C(Cl)C=CC2=C1 CKISTXXLRVRADV-UHFFFAOYSA-N 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
MGRVRXRGTBOSHW-UHFFFAOYSA-N (aminomethyl)phosphonic acid Chemical compound NCP(O)(O)=O MGRVRXRGTBOSHW-UHFFFAOYSA-N 0.000 abstract 1
102000003678 AMPA Receptors Human genes 0.000 abstract 1
108090000078 AMPA Receptors Proteins 0.000 abstract 1
102000000079 Kainic Acid Receptors Human genes 0.000 abstract 1
108010069902 Kainic Acid Receptors Proteins 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000000753 cycloalkyl group Chemical group 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/02—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Vascular Medicine (AREA)
Physical Education & Sports Medicine (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Psychology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

AT04769081T 2003-08-04 2004-07-29 8-chlor-2,3-benzodiazepinderivate ATE414695T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
HU0302449A HUP0302449A3 (en)	2003-08-04	2003-08-04	8-chloro-2,3-benzodiazepine derivatives, pharmaceutical compositions containing them and process for producing them

Publications (1)

Publication Number	Publication Date
ATE414695T1 true ATE414695T1 (de)	2008-12-15

Family

ID=89981556

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04769081T ATE414695T1 (de)	2003-08-04	2004-07-29	8-chlor-2,3-benzodiazepinderivate

Country Status (23)

Country	Link
US (1)	US7960375B2 (de)
EP (1)	EP1660462B1 (de)
JP (1)	JP4752011B2 (de)
KR (1)	KR20060120578A (de)
CN (1)	CN100551915C (de)
AT (1)	ATE414695T1 (de)
AU (1)	AU2004261491B2 (de)
BG (1)	BG109462A (de)
CA (1)	CA2534458A1 (de)
CZ (1)	CZ2006131A3 (de)
DE (1)	DE602004017878D1 (de)
DK (1)	DK1660462T3 (de)
EA (1)	EA009373B1 (de)
ES (1)	ES2317038T3 (de)
HU (1)	HUP0302449A3 (de)
IL (1)	IL173476A (de)
PL (2)	PL379245A1 (de)
PT (1)	PT1660462E (de)
SI (1)	SI1660462T1 (de)
SK (1)	SK50212006A3 (de)
UA (1)	UA84159C2 (de)
WO (1)	WO2005012265A1 (de)
ZA (1)	ZA200601698B (de)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU179018B (en) *	1978-10-19	1982-08-28	Gyogyszerkutato Intezet	Process for producing new 5h-2,3-benzodiazepine derivatives
HU191702B (en)	1984-06-27	1987-03-30	Gyogyszerkutato Intezet	New process for preparing 1-aryl-5 h-2,3-benzodiazepines
HU191698B (en) *	1984-07-27	1987-03-30	Gyogyszerkutato Intezet	Process for producing new 1-aryl-5h-2beta-benzodiazepines
HU195788B (en) *	1986-05-21	1988-07-28	Gyogyszerkutato Intezet	Process for producing 1-/hydroxy-stiryl/-5h-2,3-benzobiazepines and pharmaceutical compositions containing them
HU206719B (en)	1990-12-21	1992-12-28	Gyogyszerkutato Intezet	Process for producing 1-/4-acylamino-phenyl/-7,8-methylenedioxy-5h-2,3-benzodiazepine derivatives, acid addicional salts and pharmaceutical compositions containing them
DE19604920A1 (de) *	1996-02-01	1997-08-07	Schering Ag	Neue 2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel
HU9600871D0 (en) *	1996-04-04	1996-05-28	Gyogyszerkutato Intezet	New 2,3-benzodiazepine derivatives
HU225100B1 (hu) *	2000-12-21	2006-06-28	Egyt Gyogyszervegyeszeti Gyar	2,3-Benzodiazepinszármazékok, ilyen hatóanyagot tartalmazó gyógyászati készítmények és alkalmazásuk

2003
- 2003-08-04 HU HU0302449A patent/HUP0302449A3/hu unknown
2004
- 2004-07-29 PT PT04769081T patent/PT1660462E/pt unknown
- 2004-07-29 AT AT04769081T patent/ATE414695T1/de active
- 2004-07-29 SI SI200431033T patent/SI1660462T1/sl unknown
- 2004-07-29 AU AU2004261491A patent/AU2004261491B2/en not_active Ceased
- 2004-07-29 EP EP04769081A patent/EP1660462B1/de not_active Expired - Lifetime
- 2004-07-29 CA CA002534458A patent/CA2534458A1/en not_active Abandoned
- 2004-07-29 ZA ZA200601698A patent/ZA200601698B/en unknown
- 2004-07-29 PL PL379245A patent/PL379245A1/pl not_active Application Discontinuation
- 2004-07-29 EA EA200600373A patent/EA009373B1/ru not_active IP Right Cessation
- 2004-07-29 WO PCT/HU2004/000082 patent/WO2005012265A1/en not_active Ceased
- 2004-07-29 CZ CZ20060131A patent/CZ2006131A3/cs unknown
- 2004-07-29 DK DK04769081T patent/DK1660462T3/da active
- 2004-07-29 UA UAA200602304A patent/UA84159C2/ru unknown
- 2004-07-29 ES ES04769081T patent/ES2317038T3/es not_active Expired - Lifetime
- 2004-07-29 PL PL04769081T patent/PL1660462T3/pl unknown
- 2004-07-29 JP JP2006522422A patent/JP4752011B2/ja not_active Expired - Fee Related
- 2004-07-29 SK SK5021-2006A patent/SK50212006A3/sk unknown
- 2004-07-29 KR KR1020067002464A patent/KR20060120578A/ko not_active Abandoned
- 2004-07-29 CN CNB2004800254093A patent/CN100551915C/zh not_active Expired - Fee Related
- 2004-07-29 US US10/567,598 patent/US7960375B2/en not_active Expired - Fee Related
- 2004-07-29 DE DE602004017878T patent/DE602004017878D1/de not_active Expired - Lifetime
2006
- 2006-01-31 IL IL173476A patent/IL173476A/en not_active IP Right Cessation
- 2006-03-02 BG BG109462A patent/BG109462A/en unknown

Also Published As

Publication number	Publication date
PL1660462T3 (pl)	2009-07-31
EA200600373A1 (ru)	2006-08-25
SK50212006A3 (sk)	2006-08-03
BG109462A (en)	2006-11-30
IL173476A0 (en)	2006-06-11
AU2004261491A1 (en)	2005-02-10
HUP0302449A3 (en)	2005-06-28
SI1660462T1 (sl)	2009-04-30
HUP0302449A2 (hu)	2005-04-28
WO2005012265A1 (en)	2005-02-10
JP4752011B2 (ja)	2011-08-17
ES2317038T3 (es)	2009-04-16
US20080153814A1 (en)	2008-06-26
US7960375B2 (en)	2011-06-14
CA2534458A1 (en)	2005-02-10
CZ2006131A3 (cs)	2006-12-13
KR20060120578A (ko)	2006-11-27
DK1660462T3 (da)	2009-03-16
HU0302449D0 (en)	2003-10-28
AU2004261491B2 (en)	2009-12-17
EA009373B1 (ru)	2007-12-28
CN1871223A (zh)	2006-11-29
EP1660462A1 (de)	2006-05-31
PL379245A1 (pl)	2006-08-07
IL173476A (en)	2013-01-31
JP2007501216A (ja)	2007-01-25
CN100551915C (zh)	2009-10-21
PT1660462E (pt)	2009-02-20
UA84159C2 (en)	2008-09-25
DE602004017878D1 (de)	2009-01-02
EP1660462B1 (de)	2008-11-19
ZA200601698B (en)	2007-05-30

Legal Events

Date

Code

Title

Description

2009-07-15

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Publication of translation of european patent specification

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