ATE455118T1 - Chemisches zwischenprodukt - Google Patents
Chemisches zwischenproduktInfo
- Publication number
- ATE455118T1 ATE455118T1 AT03751697T AT03751697T ATE455118T1 AT E455118 T1 ATE455118 T1 AT E455118T1 AT 03751697 T AT03751697 T AT 03751697T AT 03751697 T AT03751697 T AT 03751697T AT E455118 T1 ATE455118 T1 AT E455118T1
- Authority
- AT
- Austria
- Prior art keywords
- aryl
- optionally substituted
- chemical intermediate
- halo
- cyano
- Prior art date
Links
- 125000003118 aryl group Chemical group 0.000 abstract 3
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000004104 aryloxy group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Extraction Or Liquid Replacement (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0223712.1A GB0223712D0 (en) | 2002-10-14 | 2002-10-14 | Chemical intermediate |
| PCT/SE2003/001594 WO2004035592A1 (en) | 2002-10-14 | 2003-10-13 | Chemical intermediate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE455118T1 true ATE455118T1 (de) | 2010-01-15 |
Family
ID=9945773
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT03751697T ATE455118T1 (de) | 2002-10-14 | 2003-10-13 | Chemisches zwischenprodukt |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US7314931B2 (de) |
| EP (1) | EP1554285B1 (de) |
| JP (1) | JP4476810B2 (de) |
| KR (1) | KR20050056239A (de) |
| CN (1) | CN1319976C (de) |
| AT (1) | ATE455118T1 (de) |
| AU (1) | AU2003269768B2 (de) |
| BR (1) | BR0315112A (de) |
| CA (1) | CA2501413A1 (de) |
| DE (1) | DE60330982D1 (de) |
| DK (1) | DK1554285T3 (de) |
| ES (1) | ES2337998T3 (de) |
| GB (1) | GB0223712D0 (de) |
| IL (1) | IL167778A (de) |
| IS (1) | IS7841A (de) |
| MX (1) | MXPA05003812A (de) |
| NO (1) | NO20051627L (de) |
| NZ (1) | NZ539371A (de) |
| PL (1) | PL375100A1 (de) |
| PT (1) | PT1554285E (de) |
| RU (1) | RU2326122C2 (de) |
| SI (1) | SI1554285T1 (de) |
| UA (1) | UA79986C2 (de) |
| WO (1) | WO2004035592A1 (de) |
| ZA (1) | ZA200502579B (de) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR030756A1 (es) * | 2000-10-02 | 2003-09-03 | Astrazeneca Ab | Compuesto de oxabispidina util en el tratamiento de arritmias cardiacas |
| GB0223712D0 (en) * | 2002-10-14 | 2002-11-20 | Astrazeneca Ab | Chemical intermediate |
| SE0401539D0 (sv) | 2004-06-15 | 2004-06-15 | Astrazeneca Ab | New compounds |
| JP2008543750A (ja) * | 2005-06-13 | 2008-12-04 | アストラゼネカ アクチボラグ | 心不整脈の処置用の新規オキサビスピジン化合物 |
| US20100222335A1 (en) * | 2005-06-20 | 2010-09-02 | Astrazeneca Ab | Process For The Preparation Of N,N'-Disubstituted Oxabispidines |
| WO2006137772A1 (en) * | 2005-06-20 | 2006-12-28 | Astrazeneca Ab | New physical form of n,n´- disubstituted oxabispidines |
| CA2610093A1 (en) * | 2005-06-20 | 2006-12-28 | Astrazeneca Ab | Process for the preparation of sulfonic acid salts of oxabispidines |
| AR054391A1 (es) * | 2005-06-20 | 2007-06-20 | Astrazeneca Ab | Procedimiento para la preparacion de 3,7- dihidroxi-1,5-diazaciclooctanos |
| TW200734342A (en) * | 2005-12-15 | 2007-09-16 | Astrazeneca Ab | New compounds for the treatment of cardiac arrhythmias |
| SG10201802911RA (en) | 2013-03-15 | 2018-05-30 | Global Blood Therapeutics Inc | Compounds and uses thereof for the modulation of hemoglobin |
| EA202092627A1 (ru) | 2013-11-18 | 2021-09-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
| TWI773657B (zh) | 2015-12-18 | 2022-08-11 | 美商亞德利克斯公司 | 作爲非全身tgr5促效劑之經取代之4-苯基吡啶化合物 |
| US12084472B2 (en) | 2015-12-18 | 2024-09-10 | Ardelyx, Inc. | Substituted 4-phenyl pyridine compounds as non-systemic TGR5 agonists |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9903759D0 (sv) | 1999-10-18 | 1999-10-18 | Astra Ab | Pharmaceutically active compounds |
| AR030756A1 (es) * | 2000-10-02 | 2003-09-03 | Astrazeneca Ab | Compuesto de oxabispidina util en el tratamiento de arritmias cardiacas |
| SE0101324D0 (sv) | 2001-04-12 | 2001-04-12 | Astrazeneca Ab | New process |
| GB0223712D0 (en) * | 2002-10-14 | 2002-11-20 | Astrazeneca Ab | Chemical intermediate |
-
2002
- 2002-10-14 GB GBGB0223712.1A patent/GB0223712D0/en not_active Ceased
-
2003
- 2003-10-13 KR KR1020057006247A patent/KR20050056239A/ko not_active Ceased
- 2003-10-13 JP JP2004545133A patent/JP4476810B2/ja not_active Expired - Lifetime
- 2003-10-13 WO PCT/SE2003/001594 patent/WO2004035592A1/en not_active Ceased
- 2003-10-13 DE DE60330982T patent/DE60330982D1/de not_active Expired - Lifetime
- 2003-10-13 SI SI200331761T patent/SI1554285T1/sl unknown
- 2003-10-13 EP EP03751697A patent/EP1554285B1/de not_active Expired - Lifetime
- 2003-10-13 CA CA002501413A patent/CA2501413A1/en not_active Abandoned
- 2003-10-13 CN CNB2003801013511A patent/CN1319976C/zh not_active Expired - Fee Related
- 2003-10-13 BR BR0315112-3A patent/BR0315112A/pt not_active IP Right Cessation
- 2003-10-13 AU AU2003269768A patent/AU2003269768B2/en not_active Ceased
- 2003-10-13 NZ NZ539371A patent/NZ539371A/en unknown
- 2003-10-13 US US10/532,223 patent/US7314931B2/en not_active Expired - Fee Related
- 2003-10-13 MX MXPA05003812A patent/MXPA05003812A/es active IP Right Grant
- 2003-10-13 PT PT03751697T patent/PT1554285E/pt unknown
- 2003-10-13 DK DK03751697.8T patent/DK1554285T3/da active
- 2003-10-13 UA UAA200502926A patent/UA79986C2/uk unknown
- 2003-10-13 ES ES03751697T patent/ES2337998T3/es not_active Expired - Lifetime
- 2003-10-13 AT AT03751697T patent/ATE455118T1/de not_active IP Right Cessation
- 2003-10-13 PL PL03375100A patent/PL375100A1/xx not_active Application Discontinuation
- 2003-10-13 RU RU2005109158/04A patent/RU2326122C2/ru not_active IP Right Cessation
-
2005
- 2005-03-30 ZA ZA200502579A patent/ZA200502579B/en unknown
- 2005-03-31 IL IL167778A patent/IL167778A/en not_active IP Right Cessation
- 2005-04-01 NO NO20051627A patent/NO20051627L/no not_active Application Discontinuation
- 2005-05-12 IS IS7841A patent/IS7841A/is unknown
-
2007
- 2007-11-19 US US11/942,013 patent/US20090062532A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1319976C (zh) | 2007-06-06 |
| US20060199814A1 (en) | 2006-09-07 |
| EP1554285B1 (de) | 2010-01-13 |
| JP4476810B2 (ja) | 2010-06-09 |
| UA79986C2 (en) | 2007-08-10 |
| EP1554285A1 (de) | 2005-07-20 |
| IL167778A (en) | 2010-04-29 |
| HK1078861A1 (en) | 2006-03-24 |
| HK1082498A1 (en) | 2006-06-09 |
| GB0223712D0 (en) | 2002-11-20 |
| US7314931B2 (en) | 2008-01-01 |
| MXPA05003812A (es) | 2005-06-08 |
| SI1554285T1 (sl) | 2010-04-30 |
| BR0315112A (pt) | 2005-08-16 |
| DK1554285T3 (da) | 2010-04-19 |
| ZA200502579B (en) | 2006-02-22 |
| KR20050056239A (ko) | 2005-06-14 |
| RU2326122C2 (ru) | 2008-06-10 |
| DE60330982D1 (de) | 2010-03-04 |
| ES2337998T3 (es) | 2010-05-03 |
| WO2004035592A1 (en) | 2004-04-29 |
| NZ539371A (en) | 2006-10-27 |
| US20090062532A1 (en) | 2009-03-05 |
| IS7841A (is) | 2005-05-12 |
| CN1705671A (zh) | 2005-12-07 |
| AU2003269768A1 (en) | 2004-05-04 |
| JP2006505565A (ja) | 2006-02-16 |
| NO20051627L (no) | 2005-05-06 |
| CA2501413A1 (en) | 2004-04-29 |
| PT1554285E (pt) | 2010-03-08 |
| RU2005109158A (ru) | 2006-01-20 |
| AU2003269768B2 (en) | 2007-08-23 |
| PL375100A1 (en) | 2005-11-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1554285 Country of ref document: EP |
|
| REN | Ceased due to non-payment of the annual fee |