ATE473215T1 - 4-anilinchinazolinderivate als antiproliferative wirkstoffe - Google Patents

4-anilinchinazolinderivate als antiproliferative wirkstoffe

Info

Publication number
ATE473215T1
ATE473215T1 AT03710015T AT03710015T ATE473215T1 AT E473215 T1 ATE473215 T1 AT E473215T1 AT 03710015 T AT03710015 T AT 03710015T AT 03710015 T AT03710015 T AT 03710015T AT E473215 T1 ATE473215 T1 AT E473215T1
Authority
AT
Austria
Prior art keywords
anilinequinazoline
derivatives
active ingredients
antiproliferative active
antiproliferative
Prior art date
Application number
AT03710015T
Other languages
English (en)
Inventor
Robert Hugh Bradbury
L F A Hennequin
Jason Kettle
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=28678580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE473215(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0207323A external-priority patent/GB0207323D0/en
Priority claimed from GB0230086A external-priority patent/GB0230086D0/en
Priority claimed from GB0301916A external-priority patent/GB0301916D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of ATE473215T1 publication Critical patent/ATE473215T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT03710015T 2002-03-28 2003-03-26 4-anilinchinazolinderivate als antiproliferative wirkstoffe ATE473215T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0207323A GB0207323D0 (en) 2002-03-28 2002-03-28 Compounds
GB0230086A GB0230086D0 (en) 2002-12-24 2002-12-24 Compounds
GB0301916A GB0301916D0 (en) 2003-01-28 2003-01-28 Compounds
PCT/GB2003/001306 WO2003082831A1 (en) 2002-03-28 2003-03-26 4-anilino quinazoline derivatives as antiproliferative agents

Publications (1)

Publication Number Publication Date
ATE473215T1 true ATE473215T1 (de) 2010-07-15

Family

ID=28678580

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03710015T ATE473215T1 (de) 2002-03-28 2003-03-26 4-anilinchinazolinderivate als antiproliferative wirkstoffe

Country Status (28)

Country Link
US (4) US20050215574A1 (de)
EP (1) EP1487806B1 (de)
JP (2) JP3891493B2 (de)
KR (1) KR101006947B1 (de)
CN (1) CN100439344C (de)
AR (1) AR039203A1 (de)
AT (1) ATE473215T1 (de)
AU (1) AU2003214443B8 (de)
BR (1) BR0308670A (de)
CA (1) CA2479642C (de)
CY (1) CY1111039T1 (de)
DE (1) DE60333262D1 (de)
DK (1) DK1487806T3 (de)
ES (1) ES2346135T3 (de)
IL (2) IL164135A0 (de)
IS (1) IS2855B (de)
MX (1) MXPA04009486A (de)
MY (1) MY158054A (de)
NO (1) NO329542B1 (de)
NZ (1) NZ535014A (de)
PL (1) PL214880B1 (de)
PT (1) PT1487806E (de)
SA (1) SA03240080B1 (de)
SI (1) SI1487806T1 (de)
TW (2) TWI324597B (de)
UA (1) UA78302C2 (de)
UY (1) UY27742A1 (de)
WO (1) WO2003082831A1 (de)

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