ATE487479T1 - Radioaktiv markierte neurokinin-1-rezeptor- antagonisten - Google Patents
Radioaktiv markierte neurokinin-1-rezeptor- antagonistenInfo
- Publication number
- ATE487479T1 ATE487479T1 AT03759348T AT03759348T ATE487479T1 AT E487479 T1 ATE487479 T1 AT E487479T1 AT 03759348 T AT03759348 T AT 03759348T AT 03759348 T AT03759348 T AT 03759348T AT E487479 T1 ATE487479 T1 AT E487479T1
- Authority
- AT
- Austria
- Prior art keywords
- neurokinin
- receptor antagonists
- radioactively labeled
- radioactively
- labeled
- Prior art date
Links
- 239000002742 neurokinin 1 receptor antagonist Substances 0.000 title abstract 2
- 241000124008 Mammalia Species 0.000 abstract 1
- 102000002002 Neurokinin-1 Receptors Human genes 0.000 abstract 1
- 108010040718 Neurokinin-1 Receptors Proteins 0.000 abstract 1
- 238000002059 diagnostic imaging Methods 0.000 abstract 1
- 238000002372 labelling Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41322302P | 2002-09-24 | 2002-09-24 | |
| PCT/US2003/029707 WO2004029024A2 (en) | 2002-09-24 | 2003-09-19 | Radiolabeled neurokinin-1 receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE487479T1 true ATE487479T1 (de) | 2010-11-15 |
Family
ID=32043220
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT03759348T ATE487479T1 (de) | 2002-09-24 | 2003-09-19 | Radioaktiv markierte neurokinin-1-rezeptor- antagonisten |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US7354935B2 (de) |
| EP (1) | EP1545525B1 (de) |
| AT (1) | ATE487479T1 (de) |
| CA (1) | CA2499825C (de) |
| DE (1) | DE60334922D1 (de) |
| ES (1) | ES2354151T3 (de) |
| WO (1) | WO2004029024A2 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2382818T3 (es) * | 2005-09-29 | 2012-06-13 | Merck Sharp & Dohme Corp. | Inhibidores de transportadores glicina radiomarcados |
| JP5580741B2 (ja) | 2008-09-19 | 2014-08-27 | 武田薬品工業株式会社 | 含窒素複素環化合物およびその用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3925662B2 (ja) | 1995-01-12 | 2007-06-06 | グラクソ，グループ，リミテッド | タキキニンアンタゴニスト活性を有するピペリジン誘導体 |
| AU1309100A (en) * | 1998-09-29 | 2000-04-17 | Merck & Co., Inc. | Radiolabeled neurokinin-1 receptor antagonists |
| GB0222426D0 (en) * | 2002-09-27 | 2002-11-06 | Imaging Res Solutions Ltd | Chemical process |
-
2003
- 2003-09-19 ES ES03759348T patent/ES2354151T3/es not_active Expired - Lifetime
- 2003-09-19 CA CA2499825A patent/CA2499825C/en not_active Expired - Fee Related
- 2003-09-19 WO PCT/US2003/029707 patent/WO2004029024A2/en not_active Ceased
- 2003-09-19 AT AT03759348T patent/ATE487479T1/de not_active IP Right Cessation
- 2003-09-19 US US10/528,888 patent/US7354935B2/en not_active Expired - Fee Related
- 2003-09-19 EP EP03759348A patent/EP1545525B1/de not_active Expired - Lifetime
- 2003-09-19 DE DE60334922T patent/DE60334922D1/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| CA2499825C (en) | 2011-11-01 |
| US20050214204A1 (en) | 2005-09-29 |
| EP1545525A2 (de) | 2005-06-29 |
| EP1545525A4 (de) | 2009-07-01 |
| ES2354151T3 (es) | 2011-03-10 |
| DE60334922D1 (de) | 2010-12-23 |
| US7354935B2 (en) | 2008-04-08 |
| EP1545525B1 (de) | 2010-11-10 |
| CA2499825A1 (en) | 2004-04-08 |
| WO2004029024A2 (en) | 2004-04-08 |
| WO2004029024A3 (en) | 2004-07-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |