ATE487479T1 - Radioaktiv markierte neurokinin-1-rezeptor- antagonisten - Google Patents

Radioaktiv markierte neurokinin-1-rezeptor- antagonisten

Info

Publication number
ATE487479T1
ATE487479T1 AT03759348T AT03759348T ATE487479T1 AT E487479 T1 ATE487479 T1 AT E487479T1 AT 03759348 T AT03759348 T AT 03759348T AT 03759348 T AT03759348 T AT 03759348T AT E487479 T1 ATE487479 T1 AT E487479T1
Authority
AT
Austria
Prior art keywords
neurokinin
receptor antagonists
radioactively labeled
radioactively
labeled
Prior art date
Application number
AT03759348T
Other languages
English (en)
Inventor
H Donald Burns
Wai-Si Eng
Raymond Gibson
Terence Hamill
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Application granted granted Critical
Publication of ATE487479T1 publication Critical patent/ATE487479T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT03759348T 2002-09-24 2003-09-19 Radioaktiv markierte neurokinin-1-rezeptor- antagonisten ATE487479T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41322302P 2002-09-24 2002-09-24
PCT/US2003/029707 WO2004029024A2 (en) 2002-09-24 2003-09-19 Radiolabeled neurokinin-1 receptor antagonists

Publications (1)

Publication Number Publication Date
ATE487479T1 true ATE487479T1 (de) 2010-11-15

Family

ID=32043220

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03759348T ATE487479T1 (de) 2002-09-24 2003-09-19 Radioaktiv markierte neurokinin-1-rezeptor- antagonisten

Country Status (7)

Country Link
US (1) US7354935B2 (de)
EP (1) EP1545525B1 (de)
AT (1) ATE487479T1 (de)
CA (1) CA2499825C (de)
DE (1) DE60334922D1 (de)
ES (1) ES2354151T3 (de)
WO (1) WO2004029024A2 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7834031B2 (en) * 2005-09-29 2010-11-16 Merck Sharp & Dohme Corp. Radiolabeled glycine transporter inhibitors
US8592454B2 (en) * 2008-09-19 2013-11-26 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound and use of same

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0802912B1 (de) 1995-01-12 2004-10-13 Glaxo Group Limited Piperidinderivate mit tachykinin-antagonistischer wirkung
EP1119356B1 (de) * 1998-09-29 2009-08-19 Merck & Co., Inc. Radiomarkierte neurokinin-1 rezeptor antagonisten
GB0222426D0 (en) * 2002-09-27 2002-11-06 Imaging Res Solutions Ltd Chemical process

Also Published As

Publication number Publication date
DE60334922D1 (de) 2010-12-23
US20050214204A1 (en) 2005-09-29
EP1545525B1 (de) 2010-11-10
EP1545525A4 (de) 2009-07-01
CA2499825A1 (en) 2004-04-08
EP1545525A2 (de) 2005-06-29
CA2499825C (en) 2011-11-01
WO2004029024A2 (en) 2004-04-08
US7354935B2 (en) 2008-04-08
ES2354151T3 (es) 2011-03-10
WO2004029024A3 (en) 2004-07-08

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties