ATE487693T1 - Verfahren zur herstellung von (r)-(-)-5-(2- aminopropyl)-2-methoxybenzolsulfonamid - Google Patents

Verfahren zur herstellung von (r)-(-)-5-(2- aminopropyl)-2-methoxybenzolsulfonamid

Info

Publication number: ATE487693T1
Authority: AT; Austria
Prior art keywords: formula; methoxybenzenesulfonamide; aminopropyl; producing; resulting
Prior art date: 2004-02-05

Application number

AT05700507T

Other languages

English (en)

Inventor

Josef Hajicek

Marketa Slavikova

Original Assignee

Zentiva Ks

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-02-05

Filing date

2005-02-03

Publication date

2010-11-15

2005-02-03 Application filed by Zentiva Ks filed Critical Zentiva Ks

2010-11-15 Application granted granted Critical

2010-11-15 Publication of ATE487693T1 publication Critical patent/ATE487693T1/de

Links

IORITYIZDHJCGT-SSDOTTSWSA-N 5-[(2r)-2-aminopropyl]-2-methoxybenzenesulfonamide Chemical compound COC1=CC=C(C[C@@H](C)N)C=C1S(N)(=O)=O IORITYIZDHJCGT-SSDOTTSWSA-N 0.000 title abstract 2
238000004519 manufacturing process Methods 0.000 title abstract 2
DRHKJLXJIQTDTD-OAHLLOKOSA-N Tamsulosine Chemical compound CCOC1=CC=CC=C1OCCN[C@H](C)CC1=CC=C(OC)C(S(N)(=O)=O)=C1 DRHKJLXJIQTDTD-OAHLLOKOSA-N 0.000 abstract 1
150000001408 amides Chemical class 0.000 abstract 1
150000001412 amines Chemical class 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
238000005984 hydrogenation reaction Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
125000006239 protecting group Chemical group 0.000 abstract 1
229940124530 sulfonamide Drugs 0.000 abstract 1
150000003456 sulfonamides Chemical class 0.000 abstract 1
XTHPWXDJESJLNJ-UHFFFAOYSA-N sulfurochloridic acid Chemical compound OS(Cl)(=O)=O XTHPWXDJESJLNJ-UHFFFAOYSA-N 0.000 abstract 1
229960002613 tamsulosin Drugs 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
- C07C311/46—Y being a hydrogen or a carbon atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
- C07C303/38—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids by reaction of ammonia or amines with sulfonic acids, or with esters, anhydrides, or halides thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AT05700507T 2004-02-05 2005-02-03 Verfahren zur herstellung von (r)-(-)-5-(2- aminopropyl)-2-methoxybenzolsulfonamid ATE487693T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CZ2004197A CZ2004197A3 (cs)	2004-02-05	2004-02-05	Způsob výroby (R)-(-)-5-(2-aminopropyl)-2-methoxybenzensulfonamidu
PCT/CZ2005/000010 WO2005075415A1 (en)	2004-02-05	2005-02-03	A method of preparation of (r)-(-)-5(2-aminopropyl)-2-methoxybenzenesulfonamide

Publications (1)

Publication Number	Publication Date
ATE487693T1 true ATE487693T1 (de)	2010-11-15

Family

ID=34832120

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT05700507T ATE487693T1 (de)	2004-02-05	2005-02-03	Verfahren zur herstellung von (r)-(-)-5-(2- aminopropyl)-2-methoxybenzolsulfonamid

Country Status (12)

Country	Link
US (1)	US7638649B2 (de)
EP (1)	EP1996544B1 (de)
AT (1)	ATE487693T1 (de)
CA (1)	CA2554851A1 (de)
CZ (1)	CZ2004197A3 (de)
DE (1)	DE602005024728D1 (de)
EA (1)	EA010131B1 (de)
ES (1)	ES2354615T3 (de)
PL (1)	PL1996544T3 (de)
PT (1)	PT1996544E (de)
UA (1)	UA85581C2 (de)
WO (1)	WO2005075415A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT103216B (pt) *	2004-12-06	2010-05-19	Hovione Farmaciencia S A	Preparação de tamsulosin
US8273918B2 (en) *	2005-09-12	2012-09-25	Avrobindo Pharma Ltd.	Process for preparing tamsulosin hydrochloride
AR058165A1 (es) *	2005-10-28	2008-01-23	Medichem Sa	Proceso para la preparacion de tamsulosina y compestos relacionados

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS62114952A (ja)	1985-11-13	1987-05-26	Yamanouchi Pharmaceut Co Ltd	置換フエネチルアミン誘導体の製造法
JPH066565B2 (ja) *	1986-07-21	1994-01-26	山之内製薬株式会社	光学活性なベンゼンスルホンアミド誘導体の製造法
KR100525493B1 (ko)	2001-02-23	2005-11-02	연성정밀화학(주)	설파모일 치환 페네틸아민 유도체의 제조 방법

2004
- 2004-02-05 CZ CZ2004197A patent/CZ2004197A3/cs not_active IP Right Cessation
2005
- 2005-02-03 CA CA002554851A patent/CA2554851A1/en not_active Abandoned
- 2005-02-03 PL PL05700507T patent/PL1996544T3/pl unknown
- 2005-02-03 PT PT05700507T patent/PT1996544E/pt unknown
- 2005-02-03 AT AT05700507T patent/ATE487693T1/de not_active IP Right Cessation
- 2005-02-03 US US10/588,515 patent/US7638649B2/en not_active Expired - Fee Related
- 2005-02-03 ES ES05700507T patent/ES2354615T3/es not_active Expired - Lifetime
- 2005-02-03 EA EA200601393A patent/EA010131B1/ru not_active IP Right Cessation
- 2005-02-03 DE DE602005024728T patent/DE602005024728D1/de not_active Expired - Lifetime
- 2005-02-03 UA UAA200609600A patent/UA85581C2/ru unknown
- 2005-02-03 EP EP05700507A patent/EP1996544B1/de not_active Expired - Lifetime
- 2005-02-03 WO PCT/CZ2005/000010 patent/WO2005075415A1/en not_active Ceased

Also Published As

Publication number	Publication date
EA010131B1 (ru)	2008-06-30
CA2554851A1 (en)	2005-08-18
WO2005075415A1 (en)	2005-08-18
CZ295583B6 (cs)	2005-08-17
DE602005024728D1 (de)	2010-12-23
UA85581C2 (en)	2009-02-10
US7638649B2 (en)	2009-12-29
US20080319225A1 (en)	2008-12-25
EP1996544B1 (de)	2010-11-10
EA200601393A1 (ru)	2006-12-29
CZ2004197A3 (cs)	2005-08-17
PT1996544E (pt)	2011-01-19
PL1996544T3 (pl)	2011-04-29
EP1996544A1 (de)	2008-12-03
ES2354615T3 (es)	2011-03-16

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Legal Events

Date	Code	Title	Description
2011-05-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties