ATE507219T1 - Malatsalze und polymorphe von (3s,5s)-7-ä3-amino- 5-methyl-piperidinylü-1-cyclopropyl-1,4-dihydro 8-methoxy-4-oxo-3-chinolincarbonsäure - Google Patents

Malatsalze und polymorphe von (3s,5s)-7-ä3-amino- 5-methyl-piperidinylü-1-cyclopropyl-1,4-dihydro 8-methoxy-4-oxo-3-chinolincarbonsäure

Info

Publication number
ATE507219T1
ATE507219T1 AT07735261T AT07735261T ATE507219T1 AT E507219 T1 ATE507219 T1 AT E507219T1 AT 07735261 T AT07735261 T AT 07735261T AT 07735261 T AT07735261 T AT 07735261T AT E507219 T1 ATE507219 T1 AT E507219T1
Authority
AT
Austria
Prior art keywords
piperidinylü
polymorphs
cyclopropyl
dihydro
oxo
Prior art date
Application number
AT07735261T
Other languages
English (en)
Inventor
Nancy Redman-Furey
Jane Godlewski
Michael Dicks
Original Assignee
Warner Chilcott Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38441484&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE507219(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Chilcott Co Llc filed Critical Warner Chilcott Co Llc
Application granted granted Critical
Publication of ATE507219T1 publication Critical patent/ATE507219T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT07735261T 2006-03-28 2007-03-26 Malatsalze und polymorphe von (3s,5s)-7-ä3-amino- 5-methyl-piperidinylü-1-cyclopropyl-1,4-dihydro 8-methoxy-4-oxo-3-chinolincarbonsäure ATE507219T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78648306P 2006-03-28 2006-03-28
PCT/IB2007/051055 WO2007110834A2 (en) 2006-03-28 2007-03-26 Malate salts, and polymorphs of (3s,5s)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid

Publications (1)

Publication Number Publication Date
ATE507219T1 true ATE507219T1 (de) 2011-05-15

Family

ID=38441484

Family Applications (1)

Application Number Title Priority Date Filing Date
AT07735261T ATE507219T1 (de) 2006-03-28 2007-03-26 Malatsalze und polymorphe von (3s,5s)-7-ä3-amino- 5-methyl-piperidinylü-1-cyclopropyl-1,4-dihydro 8-methoxy-4-oxo-3-chinolincarbonsäure

Country Status (27)

Country Link
US (1) US8039485B2 (de)
EP (1) EP2001862B1 (de)
JP (1) JP5097967B2 (de)
KR (1) KR101102288B1 (de)
AR (2) AR060189A1 (de)
AT (1) ATE507219T1 (de)
AU (1) AU2007230630B2 (de)
BR (1) BRPI0709772B8 (de)
CA (1) CA2647346C (de)
CY (1) CY1111683T1 (de)
DE (1) DE602007014191D1 (de)
DK (1) DK2001862T3 (de)
ES (1) ES2366150T3 (de)
HR (1) HRP20110558T1 (de)
IL (1) IL193990A (de)
MA (1) MA30554B1 (de)
MX (1) MX2008012328A (de)
MY (1) MY148393A (de)
NZ (1) NZ570494A (de)
PE (1) PE20080175A1 (de)
PL (1) PL2001862T3 (de)
PT (1) PT2001862E (de)
SI (1) SI2001862T1 (de)
SM (1) SMP200800058B (de)
TW (1) TWI364419B (de)
WO (1) WO2007110834A2 (de)
ZA (1) ZA200807158B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2647454A1 (en) * 2006-03-28 2007-10-04 The Procter & Gamble Company A coupling process for preparing quinolone intermediates
US8658183B2 (en) * 2007-08-09 2014-02-25 Taigen Biotechnology Company, Ltd. Antimicrobial parenteral formulation
AU2008358909B2 (en) * 2008-07-01 2012-12-13 Taigen Biotechnology Co., Ltd. Treatment of antibiotic-resistant bacteria infection
CN101618039B (zh) * 2008-07-02 2012-04-11 太景生物科技股份有限公司 肺炎的治疗药物
US8553466B2 (en) 2010-03-04 2013-10-08 Samsung Electronics Co., Ltd. Non-volatile memory device, erasing method thereof, and memory system including the same
CZ304983B6 (cs) * 2012-10-12 2015-03-11 Zentiva, K.S. Způsob výroby a nové intermediáty syntézy elvitegraviru
CZ304984B6 (cs) 2012-10-12 2015-03-11 Zentiva, K.S. Zlepšený způsob výroby a nové intermediáty syntézy elvitegraviru
CN103145615B (zh) * 2013-03-20 2015-07-29 浙江医药股份有限公司 一种奈诺沙星螯合物的后处理方法
CN114437026A (zh) * 2021-10-26 2022-05-06 浙江医药股份有限公司新昌制药厂 一种低组合物杂质的苹果酸奈诺沙星原料药及其制备方法
CN116332831B (zh) * 2023-03-15 2025-10-28 浙江医药股份有限公司新昌制药厂 氨基被Boc保护的3-氨基-5-甲基哌啶的提纯方法

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Also Published As

Publication number Publication date
TW200808759A (en) 2008-02-16
ES2366150T3 (es) 2011-10-17
MX2008012328A (es) 2008-10-09
WO2007110834A2 (en) 2007-10-04
AU2007230630B2 (en) 2012-12-20
CY1111683T1 (el) 2015-10-07
PL2001862T3 (pl) 2011-09-30
KR101102288B1 (ko) 2012-01-03
HRP20110558T1 (hr) 2011-09-30
AR060189A1 (es) 2008-05-28
NZ570494A (en) 2011-09-30
KR20090004887A (ko) 2009-01-12
EP2001862A2 (de) 2008-12-17
US20070232650A1 (en) 2007-10-04
JP2009531417A (ja) 2009-09-03
AR060377A1 (es) 2008-06-11
EP2001862B1 (de) 2011-04-27
JP5097967B2 (ja) 2012-12-12
MY148393A (en) 2013-04-15
ZA200807158B (en) 2009-09-30
SMP200800058B (it) 2009-09-07
MA30554B1 (fr) 2009-07-01
AU2007230630A1 (en) 2007-10-04
SMAP200800058A (it) 2008-10-29
DK2001862T3 (da) 2011-08-08
CA2647346A1 (en) 2007-10-04
BRPI0709772B8 (pt) 2021-05-25
PT2001862E (pt) 2011-07-20
BRPI0709772B1 (pt) 2019-10-15
TWI364419B (en) 2012-05-21
PE20080175A1 (es) 2008-03-14
RU2417222C2 (ru) 2011-04-27
US8039485B2 (en) 2011-10-18
WO2007110834A3 (en) 2007-12-06
CA2647346C (en) 2011-07-19
DE602007014191D1 (en) 2011-06-09
SI2001862T1 (sl) 2011-10-28
IL193990A (en) 2014-12-31
BRPI0709772A2 (pt) 2011-07-26
RU2008134544A (ru) 2010-05-10

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