ATE514778T1 - G-protein-gekoppelte rezeptor-antagonisten - Google Patents

G-protein-gekoppelte rezeptor-antagonisten

Info

Publication number
ATE514778T1
ATE514778T1 AT99944181T AT99944181T ATE514778T1 AT E514778 T1 ATE514778 T1 AT E514778T1 AT 99944181 T AT99944181 T AT 99944181T AT 99944181 T AT99944181 T AT 99944181T AT E514778 T1 ATE514778 T1 AT E514778T1
Authority
AT
Austria
Prior art keywords
protein
coupled receptor
receptor antagonists
receptor
tocolytics
Prior art date
Application number
AT99944181T
Other languages
English (en)
Inventor
Sylvain Chemtob
Krishna Peri
Original Assignee
Chu Sainte Justine
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chu Sainte Justine filed Critical Chu Sainte Justine
Application granted granted Critical
Publication of ATE514778T1 publication Critical patent/ATE514778T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
    • C07K14/72—Receptors; Cell surface antigens; Cell surface determinants for hormones
    • C07K14/723—G protein coupled receptor, e.g. TSHR-thyrotropin-receptor, LH/hCG receptor, FSH receptor
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06—Antiabortive agents; Labour repressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Endocrinology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Pregnancy & Childbirth (AREA)
  • Gynecology & Obstetrics (AREA)
  • Cell Biology (AREA)
  • Immunology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
AT99944181T 1998-09-17 1999-09-15 G-protein-gekoppelte rezeptor-antagonisten ATE514778T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15462798A 1998-09-17 1998-09-17
PCT/CA1999/000844 WO2000017348A1 (en) 1998-09-17 1999-09-15 G protein-coupled receptor agonists or antagonists

Publications (1)

Publication Number Publication Date
ATE514778T1 true ATE514778T1 (de) 2011-07-15

Family

ID=22552099

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99944181T ATE514778T1 (de) 1998-09-17 1999-09-15 G-protein-gekoppelte rezeptor-antagonisten

Country Status (8)

Country Link
EP (1) EP1114151B1 (de)
JP (1) JP4431280B2 (de)
AT (1) ATE514778T1 (de)
AU (1) AU5722499A (de)
CA (2) CA2689373A1 (de)
ES (1) ES2369470T3 (de)
MX (1) MXPA01002798A (de)
WO (1) WO2000017348A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1138692A1 (de) 2000-03-29 2001-10-04 Erasmus Universiteit Rotterdam Fragmente des menschlichen Choriongonadotropins als Immunoregulatoren
US7358330B2 (en) 2001-03-29 2008-04-15 Biotempt B.V. Immunoregulatory compositions
EP1300418A1 (de) * 2001-10-04 2003-04-09 Erasmus Universiteit Rotterdam Genregulation durch Oligopeptide
USRE43279E1 (en) 2000-03-29 2012-03-27 Biotemp B.V. Compositions capable of reducing elevated blood urea concentration
AU2002248322B2 (en) * 2001-01-24 2005-06-09 The Arizona Board Of Regents, On Behalf Of, The University Of Arizona Methods for screening for substances which inhibit FP prostanoid receptor interaction with a compound having PGF2alphaalphaactivity and methods of treating cancer
AU2002331064B2 (en) * 2001-08-10 2007-08-23 Palatin Technologies, Inc. Peptidomimetics of biologically active metallopeptides
US7560433B2 (en) 2001-12-21 2009-07-14 Biotempt B.V. Treatment of multiple sclerosis (MS)
JP2005532295A (ja) * 2002-04-17 2005-10-27 メディカル リサーチ カウンシル 月経過多を治療するためのＦＰレセプターアンタゴニスト又はＰＧＦ２αアンタゴニスト
GB0208785D0 (en) * 2002-04-17 2002-05-29 Medical Res Council Treatment methtods
US7521530B2 (en) * 2002-06-11 2009-04-21 Universite De Montreal Peptides and peptidomimetics useful for inhibiting the activity of prostaglandin F2α receptor

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5688938A (en) 1991-08-23 1997-11-18 The Brigham & Women's Hospital, Inc. Calcium receptor-active molecules
EP0613472A1 (de) 1991-11-05 1994-09-07 G.D. Searle & Co. 10-acyl-dibenz(b,f)(1,4)-oxazepine und ihre thiazepine analoge verwendbar als prostaglandinantagonisten
US5869281A (en) 1993-06-25 1999-02-09 Merck Frosst Canada Inc. DNA encoding prostaglandin receptor FP
CA2211176A1 (en) 1995-01-25 1996-08-01 Cor Therapeutics, Inc. Recombinant c140 receptor, its agonists and antagonists, and nucleic acids encoding the receptor

Also Published As

Publication number Publication date
WO2000017348A1 (en) 2000-03-30
CA2689373A1 (en) 2000-03-30
AU5722499A (en) 2000-04-10
MXPA01002798A (es) 2003-06-06
CA2342960C (en) 2010-03-09
JP4431280B2 (ja) 2010-03-10
EP1114151B1 (de) 2011-06-29
EP1114151A1 (de) 2001-07-11
JP2002526509A (ja) 2002-08-20
ES2369470T3 (es) 2011-12-01
CA2342960A1 (en) 2000-03-30

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