ATE546459T1 - Verfahren zur herstellung von kristallinem ciclesonid mit definierter teilchengrösse - Google Patents

Verfahren zur herstellung von kristallinem ciclesonid mit definierter teilchengrösse

Info

Publication number: ATE546459T1
Authority: AT; Austria
Prior art keywords: particle size; producing crystalline; defined particle; crystalline ciclesonide; ciclesonide
Prior art date: 2003-03-27

Application number

AT04723609T

Other languages

English (en)

Inventor

Beate Schmidt

Klaus Eistetter

Stefan Kaupp

Ernst Sturm

Original Assignee

Nycomed Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-03-27

Filing date

2004-03-26

Publication date

2012-03-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33099298&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE546459(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-03-26 Application filed by Nycomed Gmbh filed Critical Nycomed Gmbh

2012-03-15 Application granted granted Critical

2012-03-15 Publication of ATE546459T1 publication Critical patent/ATE546459T1/de

Links

LUKZNWIVRBCLON-GXOBDPJESA-N Ciclesonide Chemical compound C1([C@H]2O[C@@]3([C@H](O2)C[C@@H]2[C@@]3(C[C@H](O)[C@@H]3[C@@]4(C)C=CC(=O)C=C4CC[C@H]32)C)C(=O)COC(=O)C(C)C)CCCCC1 LUKZNWIVRBCLON-GXOBDPJESA-N 0.000 title 1
229960003728 ciclesonide Drugs 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
239000002245 particle Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01F—MIXING, e.g. DISSOLVING, EMULSIFYING OR DISPERSING
- B01F21/00—Dissolving

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Pulmonology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT04723609T 2003-03-27 2004-03-26 Verfahren zur herstellung von kristallinem ciclesonid mit definierter teilchengrösse ATE546459T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP03007007		2003-03-27
DE10314097		2003-03-27
PCT/EP2004/050373 WO2004085460A1 (en)	2003-03-27	2004-03-26	Process for preparing crystalline ciclesonide with defined particle size

Publications (1)

Publication Number	Publication Date
ATE546459T1 true ATE546459T1 (de)	2012-03-15

Family

ID=33099298

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04723609T ATE546459T1 (de)	2003-03-27	2004-03-26	Verfahren zur herstellung von kristallinem ciclesonid mit definierter teilchengrösse

Country Status (27)

Country	Link
US (1)	US9422327B2 (de)
EP (1)	EP1611150B1 (de)
JP (1)	JP4746535B2 (de)
KR (1)	KR101102709B1 (de)
AR (1)	AR043579A1 (de)
AT (1)	ATE546459T1 (de)
AU (1)	AU2004224092B2 (de)
BR (1)	BRPI0408569B1 (de)
CA (1)	CA2519752C (de)
CL (1)	CL2004000636A1 (de)
CY (1)	CY1112970T1 (de)
DK (1)	DK1611150T3 (de)
EA (1)	EA011157B1 (de)
ES (1)	ES2382928T3 (de)
HR (1)	HRP20050917B1 (de)
IL (1)	IL170746A (de)
MX (1)	MXPA05010041A (de)
MY (1)	MY143936A (de)
NO (1)	NO331984B1 (de)
NZ (1)	NZ542827A (de)
PE (1)	PE20050388A1 (de)
PL (1)	PL1611150T3 (de)
PT (1)	PT1611150E (de)
RS (1)	RS52549B (de)
SI (1)	SI1611150T1 (de)
TW (1)	TWI328589B (de)
WO (1)	WO2004085460A1 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PE20050941A1 (es)	2003-12-16	2005-11-08	Nycomed Gmbh	Suspensiones acuosas de ciclesonida para nebulizacion
WO2007056181A2 (en) *	2005-11-02	2007-05-18	Sicor, Inc.	Process for the preparation of ciclesonide
EP1904514A2 (de) *	2006-02-08	2008-04-02	Sicor, Inc.	Kristalline formen von ciclesonide
WO2008015696A2 (en) *	2006-05-23	2008-02-07	Cadila Healthcare Limited	Process for preparing ciclesonide
WO2008062450A2 (en) *	2006-09-18	2008-05-29	Cadila Healthcare Limited	Crystalline polymorphs of ciclesonide
EP2064227A2 (de) *	2006-09-19	2009-06-03	Cipla Ltd.	Verfahren zur herstellung von ciclesonid und dessen kristallform
IT1397499B1 (it) *	2009-01-09	2013-01-16	Farmabios Spa	Processo per la preparazione di ciclesonide
JP2011513469A (ja) *	2008-03-13	2011-04-28	ファルマビオスソシエタペルアチオニ	プレグナン誘導体の製造法
US20100120733A1 (en) *	2008-11-07	2010-05-13	Auspex Pharmaceuticals, Inc.	Steroid modulators of glucocorticoid receptor
US9109005B2 (en)	2012-02-23	2015-08-18	Boehringer Ingelheim International Gmbh	Method for manufacturing of ciclesonide
WO2014007770A2 (en)	2012-07-05	2014-01-09	Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi	Inhalation compositions comprising corticosteroid and sorbitol
WO2014007781A2 (en)	2012-07-05	2014-01-09	Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi	Inhalation compositions
US10111957B2 (en)	2012-07-05	2018-10-30	Arven Ilac Snayi ve Ticaret A.S.	Inhalation compositions comprising glucose anhydrous
RS62040B1 (sr)	2016-06-02	2021-07-30	Abbvie Inc	Agonist receptora glukokortikoida i njegovi imunokonjugati
EP3658192B1 (de)	2017-12-01	2021-04-28	AbbVie Inc.	Glucocorticoid-rezeptoragonist und immunkonjugate davon

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8328929D0 (en) *	1983-10-29	1983-11-30	Sterwin Ag	Steroid compounds
DE68907062T2 (de)	1988-10-05	1993-10-07	Upjohn Co	Feinverteiltes feste kristalline pulver durch niederschlag in einem anti-lösungsmittel.
DE407028T1 (de)	1989-05-31	1994-03-17	Fisons Plc	Medikament und Inhalationsvorrichtung dafür.
GR1001529B (el)	1990-09-07	1994-03-31	Elmuquimica Farm Sl	Μέ?οδος για την λήψη νέων 21-εστέρων της 16-17-ακετάλης της πρ να-1,4-διενο-3,20-διόνης.
FR2668945B1 (fr)	1990-11-12	1993-02-19	Theramex	Nouveau procede de cristallisation des substances organiques et les composes ainsi obtenus.
AU650953B2 (en)	1991-03-21	1994-07-07	Novartis Ag	Inhaler
GB9213874D0 (en)	1992-06-30	1992-08-12	Fisons Plc	Process to novel medicament form
GB9306703D0 (en)	1993-03-31	1993-05-26	Fisons Plc	Inhalation device
CZ287877B6 (cs)	1993-04-02	2001-03-14	Byk Gulden Lomberg Chemische Fabrik Gmbh	Prednisolonové deriváty a farmaceutické prostředky s jejich obsahem
IL111194A (en)	1993-10-08	1998-02-08	Fisons Plc	Process for the production of medicament formulations
WO1995024416A1 (de)	1994-03-09	1995-09-14	Byk Gulden Lomberg Chemische Fabrik Gmbh	Neue silylverbindungen und ihre verwendung
DE19541689A1 (de)	1994-11-14	1996-05-15	Byk Gulden Lomberg Chem Fab	Kombinationsarzneimittel
DE19635498A1 (de)	1996-09-03	1998-03-26	Byk Gulden Lomberg Chem Fab	Verfahren zur Epimerenanreicherung
US6120752A (en)	1997-05-21	2000-09-19	3M Innovative Properties Company	Medicinal aerosol products containing formulations of ciclesonide and related steroids
GB9722285D0 (en)	1997-10-23	1997-12-17	Rhone Poulenc Rorer Ltd	Inhalation device
US6264923B1 (en)	1998-05-13	2001-07-24	3M Innovative Properties Company	Medicinal aerosol formulation of ciclesonide and related compounds
NZ509328A (en) *	1998-07-24	2002-11-26	Jago Res A	Medicinal aerosol formulations
GB9828721D0 (en)	1998-12-24	1999-02-17	Glaxo Group Ltd	Novel apparatus and process
CA2376818A1 (en) *	1999-06-25	2001-01-04	Cognis Deutschland Gmbh & Co. Kg	Use of nanoscale sterols and sterol esters
AR026073A1 (es)	1999-10-20	2002-12-26	Nycomed Gmbh	Composicion farmaceutica acuosa que contiene ciclesonida
AR026072A1 (es)	1999-10-20	2002-12-26	Nycomed Gmbh	Composicion farmaceutica que contiene ciclesonida para aplicacion a la mucosa
DE60142920D1 (de)	2000-11-10	2010-10-07	Nycomed Gmbh	Verfahren zur herstellung von 16,17-ä(cyclohexylmethylen)bis(oxy)ü -11,21-dihydroxy-pregna-1,4-dien-3,20-dion oder ihre 21-isobutyrat durch transketalisation

2004
- 2004-02-13 MY MYPI20040475A patent/MY143936A/en unknown
- 2004-02-19 TW TW093104136A patent/TWI328589B/zh not_active IP Right Cessation
- 2004-03-12 AR ARP040100815A patent/AR043579A1/es unknown
- 2004-03-25 PE PE2004000317A patent/PE20050388A1/es not_active Application Discontinuation
- 2004-03-25 CL CL200400636A patent/CL2004000636A1/es unknown
- 2004-03-26 ES ES04723609T patent/ES2382928T3/es not_active Expired - Lifetime
- 2004-03-26 PL PL04723609T patent/PL1611150T3/pl unknown
- 2004-03-26 WO PCT/EP2004/050373 patent/WO2004085460A1/en not_active Ceased
- 2004-03-26 CA CA2519752A patent/CA2519752C/en not_active Expired - Fee Related
- 2004-03-26 SI SI200431866T patent/SI1611150T1/sl unknown
- 2004-03-26 NZ NZ542827A patent/NZ542827A/en not_active IP Right Cessation
- 2004-03-26 MX MXPA05010041A patent/MXPA05010041A/es active IP Right Grant
- 2004-03-26 BR BRPI0408569-8A patent/BRPI0408569B1/pt active IP Right Grant
- 2004-03-26 AU AU2004224092A patent/AU2004224092B2/en not_active Expired
- 2004-03-26 JP JP2006505496A patent/JP4746535B2/ja not_active Expired - Lifetime
- 2004-03-26 DK DK04723609.6T patent/DK1611150T3/da active
- 2004-03-26 RS YU20050704A patent/RS52549B/sr unknown
- 2004-03-26 AT AT04723609T patent/ATE546459T1/de active
- 2004-03-26 HR HRP20050917AA patent/HRP20050917B1/hr not_active IP Right Cessation
- 2004-03-26 US US10/549,631 patent/US9422327B2/en active Active
- 2004-03-26 EP EP04723609A patent/EP1611150B1/de not_active Expired - Lifetime
- 2004-03-26 KR KR1020057017580A patent/KR101102709B1/ko not_active Expired - Lifetime
- 2004-03-26 EA EA200501391A patent/EA011157B1/ru not_active IP Right Cessation
- 2004-03-26 PT PT04723609T patent/PT1611150E/pt unknown
2005
- 2005-09-08 IL IL170746A patent/IL170746A/en active IP Right Grant
- 2005-10-19 NO NO20054835A patent/NO331984B1/no unknown
2012
- 2012-05-08 CY CY20121100425T patent/CY1112970T1/el unknown

Also Published As

Publication number	Publication date
WO2004085460A8 (en)	2007-03-15
JP2006521332A (ja)	2006-09-21
KR101102709B1 (ko)	2012-01-05
PL1611150T3 (pl)	2012-07-31
TW200418519A (en)	2004-10-01
CL2004000636A1 (es)	2005-02-04
US20060128954A1 (en)	2006-06-15
DK1611150T3 (da)	2012-05-14
AU2004224092B2 (en)	2010-03-04
TWI328589B (en)	2010-08-11
KR20050114250A (ko)	2005-12-05
EP1611150B1 (de)	2012-02-22
JP4746535B2 (ja)	2011-08-10
EA200501391A1 (ru)	2006-06-30
BRPI0408569A (pt)	2006-03-21
PE20050388A1 (es)	2005-05-30
WO2004085460A1 (en)	2004-10-07
MXPA05010041A (es)	2005-11-17
AU2004224092A1 (en)	2004-10-07
EA011157B1 (ru)	2009-02-27
BRPI0408569B1 (pt)	2017-08-29
NZ542827A (en)	2008-02-29
HRP20050917B1 (hr)	2014-02-14
NO331984B1 (no)	2012-05-21
RS20050704A (sr)	2007-06-04
SI1611150T1 (sl)	2012-06-29
US9422327B2 (en)	2016-08-23
CY1112970T1 (el)	2016-04-13
CA2519752C (en)	2012-05-29
ES2382928T3 (es)	2012-06-14
EP1611150A1 (de)	2006-01-04
HRP20050917A2 (en)	2006-12-31
NO20054835L (no)	2005-10-19
HK1088905A1 (zh)	2006-11-17
RS52549B (sr)	2013-04-30
IL170746A (en)	2012-06-28
MY143936A (en)	2011-07-29
AR043579A1 (es)	2005-08-03
IL170746A0 (en)	2009-02-11
CA2519752A1 (en)	2004-10-07
PT1611150E (pt)	2012-05-07

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