ATE549019T1 - 1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung - Google Patents

1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung

Info

Publication number: ATE549019T1
Authority: AT; Austria
Prior art keywords: acetylü; adamant; ylamino; carbonitrile; pyrrolidine
Prior art date: 2005-06-10

Application number

AT09172285T

Other languages

English (en)

Inventor

James Kowalski

Jay Lakshman

Abu Serajuddin

Yatindra Joshi

Original Assignee

Novartis Pharma Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-06-10

Filing date

2006-06-08

Publication date

2012-03-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37532821&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE549019(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-06-08 Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh

2012-03-15 Application granted granted Critical

2012-03-15 Publication of ATE549019T1 publication Critical patent/ATE549019T1/de

Links

-1 3-HYDROXY-ADAMANT-1-YLAMINO Chemical class 0.000 title 1
238000009472 formulation Methods 0.000 title 1
239000000203 mixture Substances 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Diabetes (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Hematology (AREA)
Physical Education & Sports Medicine (AREA)
Obesity (AREA)
Cardiology (AREA)
Rheumatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Urology & Nephrology (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Immunology (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Psychology (AREA)
Child & Adolescent Psychology (AREA)
Inorganic Chemistry (AREA)

AT09172285T 2005-06-10 2006-06-08 1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung ATE549019T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US68971905P	2005-06-10	2005-06-10
US69030905P	2005-06-14	2005-06-14

Publications (1)

Publication Number	Publication Date
ATE549019T1 true ATE549019T1 (de)	2012-03-15

Family

ID=37532821

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AT09172285T ATE549019T1 (de)	2005-06-10	2006-06-08	1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung
AT06772653T ATE444748T1 (de)	2005-06-10	2006-06-08	1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AT06772653T ATE444748T1 (de)	2005-06-10	2006-06-08	1-ä(3-hydroxy-adamant-1-ylamino)-acetylü- pyrrolidin-2(s)-carbonitril-formulierung mit modifizierter freisetzung

Country Status (32)

Country	Link
US (2)	US20100021539A1 (de)
EP (2)	EP2191824B1 (de)
JP (7)	JP5579986B2 (de)
KR (1)	KR101312812B1 (de)
AR (1)	AR054383A1 (de)
AT (2)	ATE549019T1 (de)
AU (1)	AU2006257947B2 (de)
BR (1)	BRPI0613499B8 (de)
CA (1)	CA2610422A1 (de)
CY (1)	CY1109719T1 (de)
DE (1)	DE602006009656D1 (de)
DK (1)	DK1898904T3 (de)
EC (1)	ECSP077987A (de)
ES (2)	ES2385129T3 (de)
GT (1)	GT200600246A (de)
HR (1)	HRP20090680T1 (de)
IL (1)	IL187420A (de)
JO (1)	JO2584B1 (de)
MA (1)	MA29564B1 (de)
MX (1)	MX2007015677A (de)
MY (1)	MY152185A (de)
NO (1)	NO343043B1 (de)
NZ (1)	NZ563447A (de)
PE (3)	PE20110057A1 (de)
PL (2)	PL2191824T3 (de)
PT (2)	PT1898904E (de)
RU (1)	RU2423124C2 (de)
SA (1)	SA06270171B1 (de)
SI (1)	SI1898904T1 (de)
TN (1)	TNSN07464A1 (de)
TW (1)	TWI381835B (de)
WO (1)	WO2006135723A2 (de)

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Also Published As

Publication number	Publication date
KR101312812B1 (ko)	2013-09-27
TW200726467A (en)	2007-07-16
MX2007015677A (es)	2009-02-20
JP2013177428A (ja)	2013-09-09
BRPI0613499B1 (pt)	2020-07-14
WO2006135723A2 (en)	2006-12-21
US20110086096A1 (en)	2011-04-14
JP2016222675A (ja)	2016-12-28
AR054383A1 (es)	2007-06-20
EP1898904B1 (de)	2009-10-07
EP2191824B1 (de)	2012-03-14
JP5579986B2 (ja)	2014-08-27
KR20080028364A (ko)	2008-03-31
CY1109719T1 (el)	2014-08-13
ES2385129T3 (es)	2012-07-18
SI1898904T1 (sl)	2010-01-29
PL2191824T3 (pl)	2012-08-31
ECSP077987A (es)	2008-01-23
JP2008543773A (ja)	2008-12-04
ATE444748T1 (de)	2009-10-15
RU2007148241A (ru)	2009-07-20
NZ563447A (en)	2012-02-24
RU2423124C2 (ru)	2011-07-10
PE20070691A1 (es)	2007-08-06
BRPI0613499A2 (pt)	2011-01-11
PL1898904T3 (pl)	2010-03-31
JP2020055816A (ja)	2020-04-09
MY152185A (en)	2014-08-29
JP2022058771A (ja)	2022-04-12
PE20110057A1 (es)	2011-02-15
NO20080177L (no)	2008-02-15
DK1898904T3 (da)	2009-12-21
CA2610422A1 (en)	2006-12-21
DE602006009656D1 (de)	2009-11-19
JP2015091864A (ja)	2015-05-14
HK1117037A1 (en)	2009-01-09
BRPI0613499A8 (pt)	2019-01-15
JO2584B1 (en)	2011-02-27
JP2018172392A (ja)	2018-11-08
ES2334261T3 (es)	2010-03-08
EP1898904A2 (de)	2008-03-19
PE20150728A1 (es)	2015-06-01
HK1143094A1 (en)	2010-12-24
SA06270171B1 (ar)	2010-03-08
PT2191824E (pt)	2012-06-18
AU2006257947A1 (en)	2006-12-21
NO343043B1 (no)	2018-10-15
US20100021539A1 (en)	2010-01-28
EP2191824A1 (de)	2010-06-02
HRP20090680T1 (hr)	2010-02-28
IL187420A0 (en)	2008-02-09
IL187420A (en)	2013-01-31
TWI381835B (zh)	2013-01-11
BRPI0613499B8 (pt)	2021-05-25
WO2006135723A3 (en)	2007-07-05
TNSN07464A1 (en)	2009-03-17
PT1898904E (pt)	2009-12-23
AU2006257947B2 (en)	2010-06-10
MA29564B1 (fr)	2008-06-02
GT200600246A (es)	2007-03-28

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EP1951275A4 (de)	2010-05-05	Zusammensetzung gegen adipositas
BRPI0618398A2 (pt)	2016-11-16	artigo absorvente
NO20055686D0 (no)	2005-12-01	Sammensetning
DK1688111T3 (da)	2013-09-08	Absorberende artikel
DK1978944T3 (da)	2012-11-05	Blød-gelatine-kapselformulering
TWI370115B (en)	2012-08-11	New formulation
EP1897558A4 (de)	2012-09-12	Feste zubereitung
FR2881643B1 (fr)	2008-12-05	Composition matifiante comprenant de la perlite
ITFI20050094A1 (it)	2006-11-07	Opercolatrice perfezionata
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PL1928232T3 (pl)	2016-12-30	Stała formulacja
ITMI20051971A1 (it)	2007-04-19	Procedimento per la preparazione di - modafinil
ES1060039Y (es)	2006-02-01	Mosquero perfeccionado