ATE551342T1 - Heterocyclische verbindungen und zusammensetzungen als c-kit- und pdgfr- kinasehemmer - Google Patents

Heterocyclische verbindungen und zusammensetzungen als c-kit- und pdgfr- kinasehemmer

Info

Publication number
ATE551342T1
ATE551342T1 AT09711557T AT09711557T ATE551342T1 AT E551342 T1 ATE551342 T1 AT E551342T1 AT 09711557 T AT09711557 T AT 09711557T AT 09711557 T AT09711557 T AT 09711557T AT E551342 T1 ATE551342 T1 AT E551342T1
Authority
AT
Austria
Prior art keywords
kit
compositions
kinase inhibitors
heterocyclic compounds
pdgfr kinase
Prior art date
Application number
AT09711557T
Other languages
English (en)
Inventor
Xiaolin Li
Xiaodong Liu
Jon Loren
Valentina Molteni
Juliet Nabakka
Vince Yeh
Donatella Chianelli
Original Assignee
Irm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40577860&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE551342(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Irm Llc filed Critical Irm Llc
Application granted granted Critical
Publication of ATE551342T1 publication Critical patent/ATE551342T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Virology (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Otolaryngology (AREA)
  • Molecular Biology (AREA)
AT09711557T 2008-02-22 2009-02-20 Heterocyclische verbindungen und zusammensetzungen als c-kit- und pdgfr- kinasehemmer ATE551342T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3091208P 2008-02-22 2008-02-22
PCT/US2009/034778 WO2009105712A1 (en) 2008-02-22 2009-02-20 Heterocyclic compounds and compositions as c-kit and pdgfr kinase inhibitors

Publications (1)

Publication Number Publication Date
ATE551342T1 true ATE551342T1 (de) 2012-04-15

Family

ID=40577860

Family Applications (1)

Application Number Title Priority Date Filing Date
AT09711557T ATE551342T1 (de) 2008-02-22 2009-02-20 Heterocyclische verbindungen und zusammensetzungen als c-kit- und pdgfr- kinasehemmer

Country Status (17)

Country Link
US (1) US8278452B2 (de)
EP (1) EP2252612B1 (de)
JP (1) JP5230755B2 (de)
KR (1) KR101216323B1 (de)
CN (1) CN102083828B (de)
AR (1) AR070469A1 (de)
AT (1) ATE551342T1 (de)
AU (1) AU2009217356B2 (de)
BR (1) BRPI0908849A2 (de)
CA (1) CA2714700C (de)
CL (1) CL2009000400A1 (de)
EA (1) EA018551B1 (de)
ES (1) ES2383331T3 (de)
MX (1) MX2010009207A (de)
PE (1) PE20091492A1 (de)
TW (1) TW200940538A (de)
WO (1) WO2009105712A1 (de)

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RS58326B1 (sr) 2011-05-04 2019-03-29 Rhizen Pharmaceuticals S A Nova jedinjenja kao modulatori proteinskih kinaza
HK1200459A1 (en) * 2011-09-19 2015-08-07 Gencia Corporation Modified creatine compounds
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WO2013174962A1 (en) 2012-05-25 2013-11-28 Janssen R&D Ireland Uracyl spirooxetane nucleosides
SMT202000302T1 (it) * 2012-06-07 2020-07-08 Deciphera Pharmaceuticals Llc Diidronaftiridine e composti correlati utili come chinasi inibitori per il trattamento di malattie proliferative
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KR101988079B1 (ko) 2012-07-04 2019-06-11 리젠 파마슈티컬스 소시에떼 아노님 선택적 pi3k 델타 억제제
CN110684067A (zh) 2012-12-21 2020-01-14 艾丽奥斯生物制药有限公司 取代的核苷和核苷酸
CU24362B1 (es) 2013-09-06 2018-10-04 Aurigene Discovery Tech Ltd Derivados de 1,2,4-oxadiazol como inmunomoduladores
CN104458675A (zh) * 2013-09-12 2015-03-25 中国药科大学 一种筛选干细胞因子受体激酶抑制剂高通量筛选方法
CN104458674A (zh) * 2013-09-12 2015-03-25 中国药科大学 一种筛选血管内皮生长因子1激酶抑制剂高通量筛选方法
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KR20200083503A (ko) 2017-11-03 2020-07-08 오리진 디스커버리 테크놀로지스 리미티드 Tim-3 경로와 pd-1 경로의 이중 저해제
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