ATE7393T1 - Imidazo(1,2-a)pyridinderivate, verfahren zu ihrer herstellung und ihre therapeutische anwendung. - Google Patents

Imidazo(1,2-a)pyridinderivate, verfahren zu ihrer herstellung und ihre therapeutische anwendung.

Info

Publication number
ATE7393T1
ATE7393T1 AT81401606T AT81401606T ATE7393T1 AT E7393 T1 ATE7393 T1 AT E7393T1 AT 81401606 T AT81401606 T AT 81401606T AT 81401606 T AT81401606 T AT 81401606T AT E7393 T1 ATE7393 T1 AT E7393T1
Authority
AT
Austria
Prior art keywords
imidazo
production
pyridine derivatives
therapeutic application
pyridine
Prior art date
Application number
AT81401606T
Other languages
English (en)
Inventor
Jean-Pierre Kaplan
Pascal George
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9247171&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE7393(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Synthelabo filed Critical Synthelabo
Application granted granted Critical
Publication of ATE7393T1 publication Critical patent/ATE7393T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AT81401606T 1980-10-22 1981-10-15 Imidazo(1,2-a)pyridinderivate, verfahren zu ihrer herstellung und ihre therapeutische anwendung. ATE7393T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8022537A FR2492382A1 (fr) 1980-10-22 1980-10-22 Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
EP81401606A EP0050563B1 (de) 1980-10-22 1981-10-15 Imidazo(1,2-a)pyridinderivate, Verfahren zu ihrer Herstellung und ihre therapeutische Anwendung

Publications (1)

Publication Number Publication Date
ATE7393T1 true ATE7393T1 (de) 1984-05-15

Family

ID=9247171

Family Applications (1)

Application Number Title Priority Date Filing Date
AT81401606T ATE7393T1 (de) 1980-10-22 1981-10-15 Imidazo(1,2-a)pyridinderivate, verfahren zu ihrer herstellung und ihre therapeutische anwendung.

Country Status (22)

Country Link
US (2) US4382938A (de)
EP (1) EP0050563B1 (de)
JP (1) JPS5798283A (de)
AT (1) ATE7393T1 (de)
AU (1) AU544345B2 (de)
CA (1) CA1157470A (de)
DE (1) DE3163524D1 (de)
DK (1) DK154429C (de)
ES (1) ES8207537A1 (de)
FI (1) FI71143C (de)
FR (1) FR2492382A1 (de)
GR (1) GR74701B (de)
IE (1) IE51686B1 (de)
IL (1) IL64091A (de)
LU (1) LU88228I2 (de)
MX (1) MX6463E (de)
NL (1) NL930044I2 (de)
NO (1) NO155664C (de)
NZ (1) NZ198722A (de)
OA (1) OA07076A (de)
PT (1) PT73863B (de)
ZA (1) ZA817297B (de)

Families Citing this family (92)

* Cited by examiner, † Cited by third party
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FR2525602A1 (fr) * 1982-04-21 1983-10-28 Synthelabo Imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
FR2525601A1 (fr) * 1982-04-21 1983-10-28 Synthelabo Derives d'imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2581646B1 (fr) * 1985-05-07 1987-09-18 Synthelabo Derives d'imidazopyridine, leur preparation et leur application en therapeutique
FR2593179B1 (fr) * 1986-01-22 1988-04-01 Synthelabo Derives d'imidazo(1,2-a)quinoleines, leur preparation et leur application en therapeutique
ES2032455T3 (es) * 1986-01-22 1993-02-16 Synthelabo Procedimiento para preparar derivados de 3-acilaminometil-imidazo (-1,2-a)piridinas.
FR2593817B1 (fr) * 1986-01-31 1988-04-15 Synthelabo Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
FR2599368B1 (fr) * 1986-06-02 1988-08-05 Synthelabo Derives hydroxyles d'imidazopyridines, leur preparation et leur application en therapeutique
FR2600650B1 (fr) * 1986-06-27 1988-09-09 Synthelabo Procede de preparation d'imidazopyridines et composes intermediaires
FR2606410B1 (fr) * 1986-11-07 1989-02-24 Synthelabo Imidazopyridines, leur preparation et leur application en therapeutique
FR2606411B1 (fr) * 1986-11-07 1989-04-07 Synthelabo Imidazopyridine-acetamides, leur preparation et leur application en therapeutique
FR2606409B1 (fr) * 1986-11-07 1989-05-05 Synthelabo Derives d'imidazopyridine, leur preparation et leur application en therapeutique
FR2612927B1 (fr) * 1987-03-27 1989-06-09 Synthelabo Derives d'imidazopyridines, leur preparation et leur application en therapeutique
ES2026666T3 (es) * 1987-03-27 1992-05-01 Synthelabo Procedimiento para preparar derivados de imidazopiridinas.
FR2612928B1 (fr) * 1987-03-27 1989-06-16 Synthelabo Derives hydroxyles d'imidazopyridines, leur preparation et leur application en therapeutique
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US12077512B2 (en) 2019-03-25 2024-09-03 President And Fellows Of Harvard College Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment
JP2021050161A (ja) 2019-09-25 2021-04-01 武田薬品工業株式会社 複素環化合物及びその用途

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Also Published As

Publication number Publication date
DE3163524D1 (en) 1984-06-14
FR2492382B1 (de) 1983-07-29
ZA817297B (en) 1982-09-29
US4382938A (en) 1983-05-10
FI71143B (fi) 1986-08-14
NO155664B (no) 1987-01-26
EP0050563B1 (de) 1984-05-09
GR74701B (de) 1984-07-04
DK154429C (da) 1989-04-17
FI813288L (fi) 1982-04-23
IE812470L (en) 1982-04-22
NO813551L (no) 1982-04-23
ES506412A0 (es) 1982-09-16
NL930044I2 (nl) 1993-09-16
FR2492382A1 (fr) 1982-04-23
NZ198722A (en) 1984-10-19
OA07076A (fr) 1984-01-31
AU7668781A (en) 1983-04-28
JPS5798283A (en) 1982-06-18
FI71143C (fi) 1986-11-24
MX6463E (es) 1985-06-06
AU544345B2 (en) 1985-05-23
NO155664C (no) 1987-05-06
NL930044I1 (nl) 1993-08-02
IL64091A (en) 1984-12-31
CA1157470A (en) 1983-11-22
ES8207537A1 (es) 1982-09-16
EP0050563A1 (de) 1982-04-28
PT73863A (fr) 1981-11-01
IE51686B1 (en) 1987-02-04
IL64091A0 (en) 1982-01-31
PT73863B (fr) 1983-11-07
DK154429B (da) 1988-11-14
DK465181A (da) 1982-04-23
LU88228I2 (de) 1994-02-03
JPS637545B2 (de) 1988-02-17
US4460592A (en) 1984-07-17

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