ATE87627T1 - Pyrido(4,3-d>pyrimidin-derivate. - Google Patents

Pyrido(4,3-d>pyrimidin-derivate.

Info

Publication number
ATE87627T1
ATE87627T1 AT87810234T AT87810234T ATE87627T1 AT E87627 T1 ATE87627 T1 AT E87627T1 AT 87810234 T AT87810234 T AT 87810234T AT 87810234 T AT87810234 T AT 87810234T AT E87627 T1 ATE87627 T1 AT E87627T1
Authority
AT
Austria
Prior art keywords
amino
hydroxy
allergic
pyrido
alkylamino group
Prior art date
Application number
AT87810234T
Other languages
English (en)
Inventor
Kouichiro Go
Yoshiyuki Kurimoto
Kinashi Zoki
Norihiko Kitamura
Original Assignee
Nippon Zoki Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Zoki Pharmaceutical Co filed Critical Nippon Zoki Pharmaceutical Co
Application granted granted Critical
Publication of ATE87627T1 publication Critical patent/ATE87627T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
AT87810234T 1986-04-16 1987-04-10 Pyrido(4,3-d>pyrimidin-derivate. ATE87627T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8906586 1986-04-16
EP87810234A EP0244352B1 (de) 1986-04-16 1987-04-10 Pyrido[4,3-d]pyrimidin-Derivate

Publications (1)

Publication Number Publication Date
ATE87627T1 true ATE87627T1 (de) 1993-04-15

Family

ID=13960451

Family Applications (1)

Application Number Title Priority Date Filing Date
AT87810234T ATE87627T1 (de) 1986-04-16 1987-04-10 Pyrido(4,3-d>pyrimidin-derivate.

Country Status (6)

Country Link
US (1) US4808618A (de)
EP (1) EP0244352B1 (de)
JP (1) JPH07116188B2 (de)
AT (1) ATE87627T1 (de)
DE (1) DE3785076T2 (de)
ES (1) ES2053580T3 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9214053D0 (en) * 1992-07-02 1992-08-12 Ici Plc Heterocyclic amides
US5705491A (en) * 1992-10-27 1998-01-06 Nippon Zoki Pharmaceutical Co., Ltd. Adenosine deaminase inhibitor
TR199802192T2 (xx) * 1996-06-07 1999-02-22 Mannesmann Aktiengesellschaft �nce �erit d�k�m tesisi i�in d�k�m ba�l���.
US11091477B2 (en) * 2016-08-12 2021-08-17 Madera Therapeutics, LLC Protein kinase regulators
CN109265457A (zh) * 2018-11-01 2019-01-25 中国药科大学 一种利用氧化芳构化构建吡啶并嘧啶二酮骨架的新方法
CN109336884B (zh) * 2018-11-09 2021-02-05 安庆奇创药业有限公司 一种合成曲美替尼关键中间体的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA762455A (en) * 1962-03-22 1967-07-04 Dr. Karl Thomae Gesellschaft Mit Beschrankter Haftung Pyrido-pyrimidines

Also Published As

Publication number Publication date
JPS6345278A (ja) 1988-02-26
ES2053580T3 (es) 1994-08-01
US4808618A (en) 1989-02-28
DE3785076T2 (de) 1993-07-08
EP0244352A2 (de) 1987-11-04
JPH07116188B2 (ja) 1995-12-13
DE3785076D1 (de) 1993-05-06
EP0244352A3 (en) 1989-05-31
EP0244352B1 (de) 1993-03-31

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties