ATE88479T1 - Syntheseprodukte aus schwefel oder nichtschwefelhaltigen aminosaeuren mit pregnanderivaten, ihre herstellung und ihre anwendung. - Google Patents

Syntheseprodukte aus schwefel oder nichtschwefelhaltigen aminosaeuren mit pregnanderivaten, ihre herstellung und ihre anwendung.

Info

Publication number: ATE88479T1
Authority: AT; Austria
Prior art keywords: sulfur; pct; amino acids; derivatives; production
Prior art date: 1986-06-24

Application number

AT87440040T

Other languages

English (en)

Inventor

Catherine Milioni

Constantin Efthyimiopoulos

Bernard Koch

Louis Jung

Jean Jung

Original Assignee

Univ Pasteur

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-06-24

Filing date

1987-06-24

Publication date

1993-05-15

1987-06-24 Application filed by Univ Pasteur filed Critical Univ Pasteur

1993-05-15 Application granted granted Critical

1993-05-15 Publication of ATE88479T1 publication Critical patent/ATE88479T1/de

Links

NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 title abstract 2
229910052717 sulfur Inorganic materials 0.000 title abstract 2
239000011593 sulfur Substances 0.000 title abstract 2
239000005864 Sulphur Substances 0.000 title 1
JWMFYGXQPXQEEM-WZBAXQLOSA-N pregnane Chemical class C1CC2CCCC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](CC)[C@@]1(C)CC2 JWMFYGXQPXQEEM-WZBAXQLOSA-N 0.000 title 1
RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical class C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 abstract 1
150000001413 amino acids Chemical class 0.000 abstract 1
230000003110 anti-inflammatory effect Effects 0.000 abstract 1
230000015572 biosynthetic process Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
238000003786 synthesis reaction Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of only two carbon atoms, e.g. pregnane derivatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT87440040T 1986-06-24 1987-06-24 Syntheseprodukte aus schwefel oder nichtschwefelhaltigen aminosaeuren mit pregnanderivaten, ihre herstellung und ihre anwendung. ATE88479T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8609246A FR2600653B1 (fr)	1986-06-24	1986-06-24	Composes de synthese associative d'acides amines soufres ou non soufres avec des derives du d-4 pregnene 3,20-dione ou avec des derives du d-1,4 pregnadiene 3,20-dione aux proprietes glucocorticoides et anti-inflammatoires, procedes d'obtention, compositions pharmaceutiques les contenant. proprietes pharmacologiques et applications
EP87440040A EP0254655B1 (de)	1986-06-24	1987-06-24	Syntheseprodukte aus Schwefel oder nichtschwefelhaltigen Aminosäuren mit Pregnanderivaten, ihre Herstellung und ihre Anwendung

Publications (1)

Publication Number	Publication Date
ATE88479T1 true ATE88479T1 (de)	1993-05-15

Family

ID=9336727

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT87440040T ATE88479T1 (de)	1986-06-24	1987-06-24	Syntheseprodukte aus schwefel oder nichtschwefelhaltigen aminosaeuren mit pregnanderivaten, ihre herstellung und ihre anwendung.

Country Status (7)

Country	Link
US (1)	US4913852A (de)
EP (1)	EP0254655B1 (de)
JP (1)	JP2667418B2 (de)
AT (1)	ATE88479T1 (de)
DE (1)	DE3785505T2 (de)
FR (1)	FR2600653B1 (de)
WO (1)	WO1988000202A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5116829A (en) *	1990-04-23	1992-05-26	Kao Corporation	Steroid compounds
US5420120A (en) *	1993-12-17	1995-05-30	Alcon Laboratories, Inc.	Anti-inflammatory glucocorticoid compounds for topical ophthalmic use
US5632975A (en) *	1995-03-09	1997-05-27	Earles; R. Martin	Composition and method for treatment of dermatitis on the scalp
US6090800A (en) *	1997-05-06	2000-07-18	Imarx Pharmaceutical Corp.	Lipid soluble steroid prodrugs
US20050019266A1 (en) *	1997-05-06	2005-01-27	Unger Evan C.	Novel targeted compositions for diagnostic and therapeutic use
IT1311922B1 (it) *	1999-04-13	2002-03-20	Nicox Sa	Composti farmaceutici.
WO2000063229A1 (en) *	1999-04-19	2000-10-26	Senju Pharmaceutical Co., Ltd.	Steroid derivatives
EP1424998B1 (de) *	2001-08-16	2010-05-26	The Trustees of The University of Pennsylvania	Synthese und verwendung von reagenzien für die verbesserte dna-lipofektion und/oder prodrug- und arzneimitteltherapien mit langsamer freisetzung
CZ309617B6 (cs) *	2019-04-05	2023-05-24	Ústav organické chemie a biochemie AV ČR, v. v. i	3α5ß-Neuroaktivní steroidy pro léčbu epilepsie a záchvatových onemocnění

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1069624B (de) *	1956-08-31	1959-11-26	Chas. Pfizer S. Co., Inc., Brooklyn, N. Y. (V. St. A.)	Verfahren zur Herstellung von nebennierenrindenhormonwirksamen Derivaten des Hydrocortisons
DE1126386B (de) *	1959-11-14	1962-03-29	Hoechst Ag	Verfahren zur Herstellung von Steroid-21-aminosaeureestern
FR2077750B1 (de) *	1970-02-11	1973-03-16	Clin Byla Ets
GB1516095A (en) *	1974-07-31	1978-06-28	Glaxo Lab Ltd	17,21-diesters of 17alpha,21-dihydroxy-steroids of the pregnane series
FR2459249A1 (fr) *	1979-06-14	1981-01-09	Fabre Sa Pierre	Derives de steroides azotes sur l'atome de carbone en positio n 21 de la chaine laterale et leur application comme anti-inflammatoires

1986
- 1986-06-24 FR FR8609246A patent/FR2600653B1/fr not_active Expired
1987
- 1987-06-24 WO PCT/FR1987/000244 patent/WO1988000202A1/fr not_active Ceased
- 1987-06-24 US US07/166,122 patent/US4913852A/en not_active Expired - Fee Related
- 1987-06-24 DE DE87440040T patent/DE3785505T2/de not_active Expired - Fee Related
- 1987-06-24 AT AT87440040T patent/ATE88479T1/de active
- 1987-06-24 EP EP87440040A patent/EP0254655B1/de not_active Expired - Lifetime
- 1987-06-24 JP JP62503786A patent/JP2667418B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
FR2600653A1 (fr)	1987-12-31
DE3785505D1 (de)	1993-05-27
EP0254655B1 (de)	1993-04-21
US4913852A (en)	1990-04-03
DE3785505T2 (de)	1993-10-28
FR2600653B1 (fr)	1988-12-16
WO1988000202A1 (fr)	1988-01-14
EP0254655A1 (de)	1988-01-27
JP2667418B2 (ja)	1997-10-27
JPH01500430A (ja)	1989-02-16

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