ATE94165T1 - Zwischenprodukte fuer antibiotika. - Google Patents
Zwischenprodukte fuer antibiotika.Info
- Publication number
- ATE94165T1 ATE94165T1 AT87306539T AT87306539T ATE94165T1 AT E94165 T1 ATE94165 T1 AT E94165T1 AT 87306539 T AT87306539 T AT 87306539T AT 87306539 T AT87306539 T AT 87306539T AT E94165 T1 ATE94165 T1 AT E94165T1
- Authority
- AT
- Austria
- Prior art keywords
- antibiotics
- intermediate products
- azetidinones
- chlorides
- aldimines
- Prior art date
Links
- 239000003242 anti bacterial agent Substances 0.000 title abstract 2
- 229940088710 antibiotic agent Drugs 0.000 title abstract 2
- 239000013067 intermediate product Substances 0.000 title 1
- -1 2,5-Disubstituted oxazolidin-4-one-3-ylacetyl chlorides Chemical class 0.000 abstract 1
- AODGNVSBNVOVPQ-UHFFFAOYSA-N 2-(5-oxoimidazolidin-1-yl)acetyl chloride Chemical class ClC(=O)CN1CNCC1=O AODGNVSBNVOVPQ-UHFFFAOYSA-N 0.000 abstract 1
- 150000004705 aldimines Chemical class 0.000 abstract 1
- MNFORVFSTILPAW-UHFFFAOYSA-N azetidin-2-one Chemical class O=C1CCN1 MNFORVFSTILPAW-UHFFFAOYSA-N 0.000 abstract 1
- 238000006352 cycloaddition reaction Methods 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Cephalosporin Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/888,895 US4772694A (en) | 1986-07-24 | 1986-07-24 | Chiral 3-(1,2,5-trisubstituted imidazolidinone) azetidinone antibiotic intermediates |
| EP87306539A EP0254578B1 (de) | 1986-07-24 | 1987-07-23 | Zwischenprodukte für Antibiotika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE94165T1 true ATE94165T1 (de) | 1993-09-15 |
Family
ID=25394125
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT87306539T ATE94165T1 (de) | 1986-07-24 | 1987-07-23 | Zwischenprodukte fuer antibiotika. |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4772694A (de) |
| EP (1) | EP0254578B1 (de) |
| JP (1) | JPH0757752B2 (de) |
| KR (1) | KR960000048B1 (de) |
| AT (1) | ATE94165T1 (de) |
| CA (1) | CA1308725C (de) |
| DE (1) | DE3787333T2 (de) |
| ES (1) | ES2059384T3 (de) |
| HU (1) | HU197741B (de) |
| IL (1) | IL83269A (de) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4870169A (en) * | 1985-07-17 | 1989-09-26 | President And Fellows Of Harvard College | Intermediates for beta-lactam antibiotics |
| JPH0733254B2 (ja) * | 1990-02-27 | 1995-04-12 | ソブエクレー株式会社 | 活性水酸化マグネシウムの製造方法 |
| CA2246753C (en) | 1996-02-23 | 2005-05-10 | Eli Lilly And Company | Non-peptidyl vasopressin v1a antagonists |
| US5957712A (en) * | 1997-07-30 | 1999-09-28 | Thomas & Betts International, Inc. | Loadbreak connector assembly which prevents switching flashover |
| AU2002342045C1 (en) * | 2001-10-12 | 2009-07-30 | Azevan Pharmaceuticals, Inc. | Beta-lactamyl vasopressin Vla antagonists |
| WO2006102283A2 (en) | 2005-03-22 | 2006-09-28 | Azevan Pharmaceuticals, Inc. | Beta-lactamylalkanoic acids for treating premenstrual disorders |
| PL1910346T3 (pl) * | 2005-07-19 | 2019-09-30 | Azevan Pharmaceuticals, Inc. | Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny |
| EP2050738B1 (de) * | 2006-07-28 | 2013-07-10 | Kaneka Corporation | Neues imidazolidinonderivat, verfahren zu dessen herstellung und verfahren zur herstellung einer optisch aktiven aminosäure |
| US20100016274A1 (en) * | 2006-09-14 | 2010-01-21 | Koppel Gary A | Beta-lactam cannabinoid receptor modulators |
| RU2623209C9 (ru) | 2010-07-01 | 2018-01-22 | Азеван Фармасьютикалз, Инк. | Способы лечения посттравматического стрессового расстройства |
| BR112016022575A2 (pt) | 2014-03-28 | 2017-08-15 | Azevan Pharmaceuticals Inc | Composições e métodos para o tratamento de doenças neurodegenerativas |
| MX2020002762A (es) | 2017-09-15 | 2020-09-17 | Azevan Pharmaceuticals Inc | Composiciones y métodos para tratar una lesión cerebral. |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3487071A (en) * | 1968-12-23 | 1969-12-30 | Bristol Myers Co | 3-blocked amino-delta**1,4-2-azetidinones |
| US3920696A (en) * | 1973-04-02 | 1975-11-18 | Lilly Co Eli | 2s-carboxyalkylthio-3r-imidoazetidin-4-ones and compounds useful in their preparation |
| US4166816A (en) * | 1975-05-05 | 1979-09-04 | Smithkline Corporation | Methods and intermediates for preparing cis-4-oxoazetidine intermediates |
| US4200572A (en) * | 1975-09-03 | 1980-04-29 | Smithkline Corporation | Substituted azetidinones |
| US4565654A (en) * | 1983-03-28 | 1986-01-21 | University Of Notre Dame Du Lac | N-Acyloxy monocyclic β-lactams |
| US4751299A (en) * | 1983-11-18 | 1988-06-14 | Takeda Chemical Industries, Ltd. | Optically active β-lactams and method of their production |
-
1986
- 1986-07-24 US US06/888,895 patent/US4772694A/en not_active Expired - Lifetime
-
1987
- 1987-07-21 CA CA000542653A patent/CA1308725C/en not_active Expired - Lifetime
- 1987-07-21 IL IL83269A patent/IL83269A/xx not_active IP Right Cessation
- 1987-07-21 KR KR1019870007911A patent/KR960000048B1/ko not_active Expired - Fee Related
- 1987-07-23 ES ES87306539T patent/ES2059384T3/es not_active Expired - Lifetime
- 1987-07-23 EP EP87306539A patent/EP0254578B1/de not_active Expired - Lifetime
- 1987-07-23 DE DE87306539T patent/DE3787333T2/de not_active Expired - Fee Related
- 1987-07-23 JP JP62186497A patent/JPH0757752B2/ja not_active Expired - Fee Related
- 1987-07-23 HU HU873397A patent/HU197741B/hu not_active IP Right Cessation
- 1987-07-23 AT AT87306539T patent/ATE94165T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| KR960000048B1 (ko) | 1996-01-03 |
| US4772694A (en) | 1988-09-20 |
| IL83269A (en) | 1991-12-15 |
| HUT45048A (en) | 1988-05-30 |
| DE3787333T2 (de) | 1994-02-03 |
| JPH0757752B2 (ja) | 1995-06-21 |
| JPS6335571A (ja) | 1988-02-16 |
| EP0254578B1 (de) | 1993-09-08 |
| DE3787333D1 (de) | 1993-10-14 |
| CA1308725C (en) | 1992-10-13 |
| EP0254578A1 (de) | 1988-01-27 |
| KR880001648A (ko) | 1988-04-25 |
| HU197741B (en) | 1989-05-29 |
| ES2059384T3 (es) | 1994-11-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |