AU4469201A - Novel crystal form of pyrrolidylthiocarbapenem derivative - Google Patents

Novel crystal form of pyrrolidylthiocarbapenem derivative

Info

Publication number
AU4469201A
AU4469201A AU4469201A AU4469201A AU4469201A AU 4469201 A AU4469201 A AU 4469201A AU 4469201 A AU4469201 A AU 4469201A AU 4469201 A AU4469201 A AU 4469201A AU 4469201 A AU4469201 A AU 4469201A
Authority
AU
Australia
Prior art keywords
novel crystal
crystal form
pyrrolidylthiocarbapenem derivative
pyrrolidylthiocarbapenem
derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU4469201A
Other languages
English (en)
Inventor
Izumi Saitoh
Masayuki Takahira
Toshio Kawakita
Yasuyuki Yoshioka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=18614158&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU4469201(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Publication of AU4469201A publication Critical patent/AU4469201A/xx
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
AU4469201A 2000-03-31 2001-03-30 Novel crystal form of pyrrolidylthiocarbapenem derivative Pending AU4469201A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000099868 2000-03-31
PCT/JP2001/002834 WO2001072750A1 (en) 2000-03-31 2001-03-30 Novel crystal form of pyrrolidylthiocarbapenem derivative

Publications (1)

Publication Number Publication Date
AU4469201A true AU4469201A (en) 2001-10-08

Family

ID=18614158

Family Applications (2)

Application Number Title Priority Date Filing Date
AU4469201A Pending AU4469201A (en) 2000-03-31 2001-03-30 Novel crystal form of pyrrolidylthiocarbapenem derivative
AU2001244692A Ceased AU2001244692B2 (en) 2000-03-31 2001-03-30 Novel crystal form of pyrrolidylthiocarbapenem derivative

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2001244692A Ceased AU2001244692B2 (en) 2000-03-31 2001-03-30 Novel crystal form of pyrrolidylthiocarbapenem derivative

Country Status (17)

Country Link
US (5) US20030153191A1 (2)
EP (1) EP1270575B1 (2)
JP (1) JP3375084B2 (2)
KR (1) KR100472842B1 (2)
CN (1) CN1192030C (2)
AT (1) ATE304014T1 (2)
AU (2) AU4469201A (2)
BR (1) BRPI0109712B8 (2)
CA (1) CA2404703C (2)
CY (2) CY1105674T1 (2)
DE (1) DE60113243T2 (2)
DK (1) DK1270575T3 (2)
ES (1) ES2252205T3 (2)
MX (1) MXPA02009592A (2)
TW (1) TWI293631B (2)
WO (1) WO2001072750A1 (2)
ZA (1) ZA200207675B (2)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030153191A1 (en) * 2000-03-31 2003-08-14 Izumi Saitoh Novel crystal form of pyrrolidylthiocarbapenem derivative
JP5004355B2 (ja) * 2001-05-10 2012-08-22 塩野義製薬株式会社 アセチルチオピロリジン誘導体の製法
HUP0402112A2 (hu) * 2001-11-16 2005-02-28 Ranbaxy Laboratories Limited Eljárás kristályos imipenem előállítására
TWI353855B (en) * 2005-05-26 2011-12-11 Shionogi & Co Method for preparing an aqueous solution of doripe
TW200815442A (en) * 2006-04-28 2008-04-01 Kaneka Corp Improved method for the crystallization of intermediates of carbapenem antibiotics
WO2008006298A1 (en) * 2006-07-03 2008-01-17 Chengdu Di'ao Jiuhong Pharmaceutical Factory Novel crystal form of doripenem, preparation method and uses thereof
CN101191787B (zh) * 2006-11-21 2011-07-27 上海医药工业研究院 高效液相色谱法测定多利培南含量的方法
WO2009118680A1 (en) 2008-03-24 2009-10-01 Ranbaxy Laboratories Limited Process for the preparation of sterile doripenem
US8822445B2 (en) 2010-06-03 2014-09-02 Xuanzhu Pharma Co., Ltd. Crystalline form of carbapenem derivative or its hydrates and preparation methods and uses thereof
CN102977101A (zh) * 2011-09-07 2013-03-20 中国人民解放军军事医学科学院毒物药物研究所 多尼培南一水合物、其药物组合物、其制备方法和用途
CN102285988B (zh) * 2011-09-08 2012-09-05 上海希迈医药科技有限公司 一种多尼培南水合物晶体及其制备方法
WO2013068910A1 (en) * 2011-11-08 2013-05-16 Ranbaxy Laboratories Limited Process for the preparation of polymorphs of doripenem
CN104072497B (zh) * 2013-03-29 2017-10-03 石药集团中奇制药技术（石家庄）有限公司 一种多尼培南新结晶及其制备方法
CN103389347B (zh) * 2013-07-26 2015-12-09 深圳市海滨制药有限公司 高效液相色谱法测定多尼培南的方法
WO2015167148A1 (ko) * 2014-04-28 2015-11-05 제이더블유중외제약 주식회사 도리페넴의 신규한 결정 및 이의 제조방법
KR20160007679A (ko) 2016-01-04 2016-01-20 제일약품주식회사 도리페넴의 신규한 결정형

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5317016A (en) * 1991-08-20 1994-05-31 Shionogi Seiyaku Kabushiki Kaisha Pyrrolidylthiocarbapenem derivative
US5539102A (en) * 1992-02-21 1996-07-23 Shionogi Seiyaku Kabushiki Kaisha Production method for sulfamide
WO1995029913A1 (en) * 1994-05-02 1995-11-09 Shionogi & Co., Ltd. Crystal of pyrrolidylthiocarbapenem derivative, lyophilized preparation containing said crystal, and process for producing the same
JP3558684B2 (ja) * 1994-06-28 2004-08-25 塩野義製薬株式会社 ピロリジルチオカルバペネム誘導体の乾燥方法
US20030153191A1 (en) * 2000-03-31 2003-08-14 Izumi Saitoh Novel crystal form of pyrrolidylthiocarbapenem derivative
BRPI0407480A (pt) * 2003-02-14 2006-02-07 Shionogi & Co Cristal de intermediário sintético de carbapenem
US20120035357A1 (en) 2009-02-26 2012-02-09 Orchid Chemicals & Pharmaceuticals Ltd. Process for the preparation of carbapenem antibiotic

Also Published As

Publication number Publication date
WO2001072750A1 (en) 2001-10-04
DE60113243T2 (de) 2006-02-16
ES2252205T3 (es) 2006-05-16
US20130059831A1 (en) 2013-03-07
CN1432016A (zh) 2003-07-23
BR0109712A (pt) 2003-04-29
CY2009001I1 (el) 2009-11-04
CA2404703A1 (en) 2002-09-26
EP1270575A4 (en) 2004-02-18
JP3375084B2 (ja) 2003-02-10
KR20020087446A (ko) 2002-11-22
DE60113243D1 (de) 2005-10-13
AU2001244692B2 (en) 2004-10-14
CN1192030C (zh) 2005-03-09
MXPA02009592A (es) 2003-03-12
KR100472842B1 (ko) 2005-03-10
US20070060562A1 (en) 2007-03-15
TWI293631B (2) 2008-02-21
ZA200207675B (en) 2003-09-25
DK1270575T3 (da) 2006-01-16
US20150031664A1 (en) 2015-01-29
EP1270575A1 (en) 2003-01-02
US20080207586A1 (en) 2008-08-28
US8247402B2 (en) 2012-08-21
US9221823B2 (en) 2015-12-29
ATE304014T1 (de) 2005-09-15
CA2404703C (en) 2007-06-05
US20030153191A1 (en) 2003-08-14
CY1105674T1 (el) 2010-07-28
EP1270575B1 (en) 2005-09-07
BRPI0109712B1 (pt) 2017-10-24
BRPI0109712B8 (pt) 2021-05-25
CY2009001I2 (el) 2009-11-04

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