BE1002966A5 - Compositions pharmaceutiques. - Google Patents
Compositions pharmaceutiques. Download PDFInfo
- Publication number
- BE1002966A5 BE1002966A5 BE8901158A BE8901158A BE1002966A5 BE 1002966 A5 BE1002966 A5 BE 1002966A5 BE 8901158 A BE8901158 A BE 8901158A BE 8901158 A BE8901158 A BE 8901158A BE 1002966 A5 BE1002966 A5 BE 1002966A5
- Authority
- BE
- Belgium
- Prior art keywords
- pharmaceutical compositions
- pharmaceutically acceptable
- composition
- hypertensions
- alanyl
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 206010020772 Hypertension Diseases 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000002671 adjuvant Substances 0.000 abstract 1
- 150000001408 amides Chemical class 0.000 abstract 1
- 239000002775 capsule Substances 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 238000004806 packaging method and process Methods 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000007493 shaping process Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Abstract
Composition pharmaceutique qui comprend de l'acide 5-t-butyl-3-[N-(1-(S)-éthoxycarbonyl-3-phénylpropyl)-L-alanyl]-2,3-dihydro-1,3,4-thiadiazole-2-(S)-carboxylique, ou un sel, ester ou amide pharmaceutiquement acceptable de celui-ci, en mélange avec un adjuvant, diluant ou excipient pharmaceutiquement acceptable. Avantageusement, la composition sa prête au façonnage en comprimés ou au conditionnement dans des capsules et permet le traitement d'hypertensions de diverses origines.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB888825541A GB8825541D0 (en) | 1988-11-01 | 1988-11-01 | Formulation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE1002966A5 true BE1002966A5 (fr) | 1991-10-08 |
Family
ID=10646121
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE8901158A BE1002966A5 (fr) | 1988-11-01 | 1989-10-31 | Compositions pharmaceutiques. |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0367509A3 (fr) |
| JP (1) | JPH02172917A (fr) |
| BE (1) | BE1002966A5 (fr) |
| CA (1) | CA2001906A1 (fr) |
| CH (1) | CH679554A5 (fr) |
| DK (1) | DK541789A (fr) |
| FR (1) | FR2638642A1 (fr) |
| GB (2) | GB8825541D0 (fr) |
| GR (1) | GR1000437B (fr) |
| IE (1) | IE893502L (fr) |
| LU (1) | LU87616A1 (fr) |
| PT (1) | PT92167A (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19544507B4 (de) | 1995-11-29 | 2007-11-15 | Novartis Ag | Cyclosporin enthaltende Präparate |
| SE9700135D0 (sv) † | 1997-01-20 | 1997-01-20 | Astra Ab | New formulation |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2838387A1 (de) * | 1978-05-16 | 1979-10-31 | Lilly Industries Ltd | Zusammensetzung zum fuellen von kapseln |
| US4178374A (en) * | 1974-08-16 | 1979-12-11 | Merck & Co., Inc. | Novel pharmaceutical compositions of β-blockers with diuretics |
| EP0105996A1 (fr) * | 1982-10-15 | 1984-04-25 | Merck & Co. Inc. | Compositions ophtalmiques pour le traitement de la pression intraoculaire élevée |
| EP0217519A1 (fr) * | 1985-08-31 | 1987-04-08 | FISONS plc | Inhibiteurs de l'enzyme de conversion de l'angiotensine hétérocycliques à 5 chaînons |
-
1988
- 1988-11-01 GB GB888825541A patent/GB8825541D0/en active Pending
-
1989
- 1989-10-27 GB GB8924207A patent/GB2224206B/en not_active Expired - Fee Related
- 1989-10-27 EP EP19890311096 patent/EP0367509A3/fr not_active Withdrawn
- 1989-10-30 LU LU87616A patent/LU87616A1/fr unknown
- 1989-10-31 DK DK541789A patent/DK541789A/da not_active Application Discontinuation
- 1989-10-31 BE BE8901158A patent/BE1002966A5/fr not_active IP Right Cessation
- 1989-10-31 FR FR8914314A patent/FR2638642A1/fr not_active Withdrawn
- 1989-10-31 CA CA002001906A patent/CA2001906A1/fr not_active Abandoned
- 1989-10-31 GR GR890100710A patent/GR1000437B/el unknown
- 1989-10-31 IE IE893502A patent/IE893502L/xx unknown
- 1989-10-31 PT PT92167A patent/PT92167A/pt unknown
- 1989-11-01 JP JP1283162A patent/JPH02172917A/ja active Pending
- 1989-11-01 CH CH3944/89A patent/CH679554A5/fr not_active IP Right Cessation
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4178374A (en) * | 1974-08-16 | 1979-12-11 | Merck & Co., Inc. | Novel pharmaceutical compositions of β-blockers with diuretics |
| DE2838387A1 (de) * | 1978-05-16 | 1979-10-31 | Lilly Industries Ltd | Zusammensetzung zum fuellen von kapseln |
| EP0105996A1 (fr) * | 1982-10-15 | 1984-04-25 | Merck & Co. Inc. | Compositions ophtalmiques pour le traitement de la pression intraoculaire élevée |
| EP0217519A1 (fr) * | 1985-08-31 | 1987-04-08 | FISONS plc | Inhibiteurs de l'enzyme de conversion de l'angiotensine hétérocycliques à 5 chaînons |
Also Published As
| Publication number | Publication date |
|---|---|
| CH679554A5 (fr) | 1992-03-13 |
| GB8924207D0 (en) | 1989-12-13 |
| GR890100710A (en) | 1990-12-31 |
| DK541789D0 (da) | 1989-10-31 |
| GB2224206A (en) | 1990-05-02 |
| EP0367509A2 (fr) | 1990-05-09 |
| DK541789A (da) | 1990-05-02 |
| PT92167A (pt) | 1990-05-31 |
| GR1000437B (el) | 1992-07-30 |
| CA2001906A1 (fr) | 1990-05-01 |
| GB2224206B (en) | 1992-12-09 |
| FR2638642A1 (fr) | 1990-05-11 |
| IE893502L (en) | 1990-05-01 |
| JPH02172917A (ja) | 1990-07-04 |
| GB8825541D0 (en) | 1988-12-07 |
| EP0367509A3 (fr) | 1991-05-15 |
| LU87616A1 (fr) | 1991-07-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: FISONS PLC. Effective date: 19931031 |