BE696499A - - Google Patents

Info

Publication number
BE696499A
BE696499A BE696499DA BE696499A BE 696499 A BE696499 A BE 696499A BE 696499D A BE696499D A BE 696499DA BE 696499 A BE696499 A BE 696499A
Authority
BE
Belgium
Application number
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE696499A publication Critical patent/BE696499A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/20Two benzimidazolyl-2 radicals linked together directly or via a hydrocarbon or substituted hydrocarbon radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE696499D 1966-04-01 1967-04-03 BE696499A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DEF0048833 1966-04-01

Publications (1)

Publication Number Publication Date
BE696499A true BE696499A (fr) 1967-10-03

Family

ID=7102516

Family Applications (1)

Application Number Title Priority Date Filing Date
BE696499D BE696499A (fr) 1966-04-01 1967-04-03

Country Status (9)

Country Link
US (1) US3538097A (fr)
BE (1) BE696499A (fr)
CH (2) CH533124A (fr)
DE (1) DE1670684A1 (fr)
FR (2) FR1519964A (fr)
GB (1) GB1186723A (fr)
MY (1) MY7100120A (fr)
NL (1) NL6704539A (fr)
OA (1) OA02583A (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996006831A1 (fr) * 1994-08-26 1996-03-07 Auckland Division Cancer Society Of New Zealand Inc. Nouveaux agents d'alkilation cibles sur l'adn
AU695936B2 (en) * 1994-08-26 1998-08-27 Auckland Division Cancer Society Of New Zealand Inc Novel dna-targeted alkylating agents

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4091101A (en) * 1977-06-15 1978-05-23 Merck & Co., Inc. 6-(1-Piperazinyl)quinoxaline
DE3611343A1 (de) * 1986-04-04 1987-10-08 Boehringer Mannheim Gmbh Heterocyclisch substituierte benzimidazole, verfahren zu ihrer herstellung, arzneimittel sowie zwischenprodukte
US5807874A (en) * 1995-05-17 1998-09-15 Rutgers, The State University Of New Jersey Trisbenzimidazoles useful as topoisomerase I inhibitors
US5767142A (en) * 1996-03-20 1998-06-16 Rutgers, The State University Of New Jersey Trisbenzimidazoles useful as topoisomerase I inhibitors
AUPN449295A0 (en) * 1995-07-28 1995-08-24 Inner And Eastern Health Care Network, The Radioprotectors
US5981541A (en) * 1996-09-23 1999-11-09 Rutgers, The State University Of New Jersey Substituted heterocycles as anti-tumor agents
US6140328A (en) * 1997-12-12 2000-10-31 Rutgers, The State University Of New Jersey Heterocyclic cytotoxic agents
IL136911A0 (en) * 1997-12-31 2001-06-14 Univ Rutgers Heterocyclic topoisomerase poisons
US6063801A (en) 1998-02-12 2000-05-16 Rutgers, The State University Of New Jersey Heterocyclic topoisomerase poisons
US6740650B2 (en) 1999-10-29 2004-05-25 Rutgers, The State University Of New Jersey Heterocyclic cytotoxic agents
WO2003041653A2 (fr) * 2001-11-14 2003-05-22 Rutgers, The State University Agents cytotoxiques
JP4789414B2 (ja) * 2001-11-14 2011-10-12 ラトガーズ,ザ ステイト ユニバーシティ 可溶化トポイソメラーゼ毒性剤
CA2467774C (fr) * 2001-11-14 2011-09-20 Rutgers, The State University Poisons de topoisomerase solubilises
DE60225943T2 (de) * 2001-11-14 2009-01-29 Rutgers, The State University Topoisomerase-giftmittel
US20050119251A1 (en) * 2001-12-21 2005-06-02 Jian-Min Fu Nicotinamide derivatives and their use as therapeutic agents
AU2003268075A1 (en) * 2002-08-09 2004-02-25 Edmond J. Lavoie Nitro and amino substituted dibenzonaphthyridines as topoisomerase agents
AU2003265406A1 (en) 2002-08-09 2004-02-25 Edmond J. Lavoie Nitro and amino substituted topoisomerase agents
US6992088B2 (en) * 2002-08-09 2006-01-31 Rutgers, The State University Of New Jersey Nitro and amino substituted heterocycles as topoisomerase I targeting agents
JP4774212B2 (ja) * 2002-11-12 2011-09-14 ラトガーズ、ザ・ステイト・ユニバーシテイ・オブ・ニユー・ジヤージー トポイソメラーゼ−ターゲッティング剤
BRPI0515482A (pt) * 2004-09-20 2008-07-22 Xenon Pharmaceuticals Inc derivados heterocìclicos e seus usos como agentes terapêuticos
US8071603B2 (en) 2004-09-20 2011-12-06 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors
US8541457B2 (en) * 2005-06-03 2013-09-24 Xenon Pharmaceuticals Inc. Aminothiazole derivatives as human stearoyl-CoA desaturase inhibitors
JP5639763B2 (ja) * 2006-12-21 2014-12-10 ピーター・マッカラム・キャンサー・インスティチュート 放射線防護剤および関連する方法
GB0821913D0 (en) 2008-12-02 2009-01-07 Price & Co Antibacterial compounds
WO2010102219A1 (fr) 2009-03-06 2010-09-10 Rutgers, The State University Of New Jersey Dérivés de méthylènedioxybenzo [i] phénanthridine pour traiter le cancer
WO2010127363A1 (fr) 2009-05-01 2010-11-04 Rutgers, The State University Of New Jersey Inhibiteurs de topoisomérase
JP5712524B2 (ja) * 2009-10-28 2015-05-07 Jsr株式会社 液晶配向剤および液晶表示素子
SI2575968T1 (sl) * 2010-06-01 2016-06-30 Summit Therapeutics Plc Spojine za zdravljenje bolezni, ki je povezana s clostridium difficile
WO2012170867A1 (fr) * 2011-06-09 2012-12-13 Rhizen Pharmaceuticals Sa Nouveaux composes utilises comme modulateurs de gpr-119
GB201506660D0 (en) 2015-04-20 2015-06-03 Cellcentric Ltd Pharmaceutical compounds
GB201506658D0 (en) 2015-04-20 2015-06-03 Cellcentric Ltd Pharmaceutical compounds
WO2017125944A1 (fr) * 2016-01-23 2017-07-27 Jawaharlal Nehru University (Jnu) Activité antibactérienne à large spectre de nouveaux bisbenzimidazoles ciblant la topoisomérase ia et composition synergique associant bisbenzimidazole et inhibiteurs de pompes d'efflux pour lutter contre les bactéries pathogènes
WO2017176648A1 (fr) 2016-04-04 2017-10-12 Rutgers, The State University Of New Jersey Poisons de topoisomérase

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3103403A (en) * 1963-09-10 Dyeing of polyester fibers with com-
US2980690A (en) * 1957-08-30 1961-04-18 Ciba Pharm Prod Inc New basically substituted benzylbenzimidazoles
US3072661A (en) * 1960-08-24 1963-01-08 Interchem Corp New process for improved bis-imidazole vat dyestuff pigments
US3133056A (en) * 1961-05-15 1964-05-12 May & Baker Ltd N-phenylpiperazine derivatives of tetrahydrobenzodiazepines
NL128199C (fr) * 1962-04-21
NL135043C (fr) * 1963-10-11
GB1122988A (en) * 1964-10-22 1968-08-07 Fisons Pest Control Ltd Benzimidazole derivatives
US3336191A (en) * 1966-03-11 1967-08-15 Smith Kline French Lab Anthelmintic 2-amidobenzimidazoles
US3362956A (en) * 1965-08-19 1968-01-09 Sterling Drug Inc 1-[(heterocyclyl)-lower-alkyl]-4-substituted-piperazines

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996006831A1 (fr) * 1994-08-26 1996-03-07 Auckland Division Cancer Society Of New Zealand Inc. Nouveaux agents d'alkilation cibles sur l'adn
AU695936B2 (en) * 1994-08-26 1998-08-27 Auckland Division Cancer Society Of New Zealand Inc Novel dna-targeted alkylating agents

Also Published As

Publication number Publication date
GB1186723A (en) 1970-04-02
OA02583A (fr) 1970-05-05
FR1519964A (fr) 1968-04-05
CH525902A (de) 1972-07-31
FR6681M (fr) 1969-02-03
CH533124A (de) 1973-01-31
MY7100120A (en) 1971-12-31
DE1670684A1 (de) 1970-12-03
NL6704539A (fr) 1967-10-02
US3538097A (en) 1970-11-03

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