BE818990A - Nouvelles pyrimidines - Google Patents

Nouvelles pyrimidines

Info

Publication number
BE818990A
BE818990A BE147737A BE147737A BE818990A BE 818990 A BE818990 A BE 818990A BE 147737 A BE147737 A BE 147737A BE 147737 A BE147737 A BE 147737A BE 818990 A BE818990 A BE 818990A
Authority
BE
Belgium
Prior art keywords
new pyrimidines
pyrimidines
new
Prior art date
Application number
BE147737A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE818990A publication Critical patent/BE818990A/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A63—SPORTS; GAMES; AMUSEMENTS
    • A63C—SKATES; SKIS; ROLLER SKATES; DESIGN OR LAYOUT OF COURTS, RINKS OR THE LIKE
    • A63C19/00—Design or layout of playing courts, rinks, bowling greens or areas for water-skiing; Covers therefor
    • A63C19/02—Shaping of the surface of courts according to the necessities of the different games

Landscapes

  • Engineering & Computer Science (AREA)
  • Architecture (AREA)
  • Civil Engineering (AREA)
  • Structural Engineering (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE147737A 1973-08-20 1974-08-19 Nouvelles pyrimidines BE818990A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19732341925 DE2341925A1 (de) 1973-08-20 1973-08-20 Neue pyrimidinderivate und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
BE818990A true BE818990A (fr) 1975-02-19

Family

ID=5890167

Family Applications (1)

Application Number Title Priority Date Filing Date
BE147737A BE818990A (fr) 1973-08-20 1974-08-19 Nouvelles pyrimidines

Country Status (4)

Country Link
JP (1) JPS5049288A (fr)
BE (1) BE818990A (fr)
DE (1) DE2341925A1 (fr)
ZA (1) ZA745305B (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5075305A (en) * 1991-03-18 1991-12-24 Warner-Lambert Company Compound, composition and use
US5098902A (en) * 1991-03-18 1992-03-24 Warner-Lambert Company Method of treating neurodegenerative diseases

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1172255A (fr) * 1980-12-11 1984-08-07 Robert R. Covington Methode de preparation de buspirone
JPH0635450B2 (ja) * 1984-03-16 1994-05-11 三井東圧化学株式会社 チオシアノピリミジン誘導体、その製造法および農園芸用殺菌剤
US5658923A (en) * 1992-09-18 1997-08-19 Asahi Kasei Kogyo Kabushiki Kaisha Azepine derivatives and use thereof
KR0147732B1 (ko) * 1992-09-18 1998-08-17 유미꾸라 레이이찌 아제핀 유도체, 그의 제조방법 및 용도
CA2208900C (fr) * 1996-07-18 2006-08-01 Lonza Ag Methode de preparation de pyrimidine-2-carboxylates
ATE245641T1 (de) 1998-02-17 2003-08-15 Tularik Inc Antivirale pyrimidinderivate
US6410726B1 (en) 2000-01-12 2002-06-25 Tularik Inc. Arylsulfonic acid salts of pyrimidine-based antiviral
DK2316831T3 (da) * 2002-11-21 2013-06-10 Novartis Ag 2-(Morpholin-4-yl)pyrimidiner som phosphotidylinositol (PI)-3-kinaseinhibitorer samt deres anvendelse ved behandling af cancer
RS20050532A (sr) 2003-01-14 2007-12-31 Arena Pharmaceuticals Inc., Derivati 1,2,3-trisupstituisanog arila i heteroarila kao modulatori metabolizma za profilaksu i tretman poremećaja povezanih sa njim, kao što su dijebetes i hiperglikemija
SI1599468T1 (sl) * 2003-01-14 2008-02-29 Arena Pharm Inc 1,2,3-trisubstituirani arilni in heteroarilni derivati kot modulatorji metabolizma ter profilaksa in zdravljenje motenj v zvezi z njim, kot diabetesain hiperglikemije
CA2531061A1 (fr) 2003-07-02 2005-01-13 Vertex Pharmaceuticals Incorporated Pyrimidines utilisees comme modulateurs des canaux ioniques sensibles au voltage
AR045047A1 (es) 2003-07-11 2005-10-12 Arena Pharm Inc Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos
EP2316827B1 (fr) 2003-07-30 2016-01-27 Xenon Pharmaceuticals Inc. Derives de piperazine et leurs utilisations en tant qu'agents therapeutiques
KR20060037409A (ko) * 2003-07-30 2006-05-03 제논 파마슈티칼스 인크. 피페라진 유도체 및 그의 치료제로서의 용도
HUP0400405A3 (en) * 2004-02-10 2009-03-30 Sanofi Synthelabo Pyrimidine derivatives, process for producing them, their use, pharmaceutical compositions containing them and their intermediates
JP2007217282A (ja) * 2004-03-04 2007-08-30 Astellas Pharma Inc 置換ピリミジン誘導体
EP2289510A1 (fr) 2004-09-20 2011-03-02 Xenon Pharmaceuticals Inc. Dérivés hétérocycliques pour le traitement des maladies induites par des enzymes stearoyl-coa desaturase
US7767677B2 (en) 2004-09-20 2010-08-03 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors
EP2316458A1 (fr) 2004-09-20 2011-05-04 Xenon Pharmaceuticals Inc. Derives de pyridazine destines a l'inhibition du desaturase-coa-stearoyl de l'humain
EP1799667B1 (fr) 2004-09-20 2013-03-20 Xenon Pharmaceuticals Inc. Derives heterocycliques et leur utilisation comme agents therapeutiques
EP1804799B1 (fr) 2004-09-20 2013-08-21 Xenon Pharmaceuticals Inc. Dérivés hétérocycliques et leur utilisation en tant qu'agents thérapeutiques
CA2580856A1 (fr) 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Derives heterocycliques et leur utilisation en tant qu'inhibiteurs de la stearoyl-coa desaturase
US7951805B2 (en) 2004-09-20 2011-05-31 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase
MY148521A (en) 2005-01-10 2013-04-30 Arena Pharm Inc Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto
DOP2006000010A (es) 2005-01-10 2006-07-31 Arena Pharm Inc Procedimiento para preparar eteres aromáticos
EP1904491A2 (fr) 2005-05-31 2008-04-02 Vertex Pharmaceuticals Incorporated Heterocycles utiles comme modulateurs de canaux ioniques
EP2029138A1 (fr) 2005-06-03 2009-03-04 Xenon Pharmaceuticals Inc. Derives aminothiazole utilises en tant qu'inhibiteurs de la stearoyle-coa desaturase humaine
GB0512844D0 (en) * 2005-06-23 2005-08-03 Novartis Ag Organic compounds
JO2660B1 (en) 2006-01-20 2012-06-17 نوفارتيس ايه جي Pi-3 inhibitors and methods of use
CA2675558A1 (fr) 2007-02-06 2008-08-14 Novartis Ag Inhibiteurs de la pi3-kinase et procedes de leur utilisation
ES2499018T3 (es) 2007-09-20 2014-09-26 Irm Llc Compuestos y composiciones como moduladores de la actividad de GPR119
CA2720049A1 (fr) * 2008-03-31 2009-10-08 Zenyaku Kogyo Kabushikikaisha Derive de pyrimidine presentant une activite de protection cellulaire et son utilisation
UY32306A (es) * 2008-12-09 2010-07-30 Gilead Sciences Inc Derivados de pteridinona y pirimidinodiazepinona y composiciones farmacéuticas que modulan en forma selectiva los receptores tipo toll, métodos y usos
CN103221410B (zh) 2010-09-22 2017-09-15 艾尼纳制药公司 Gpr119受体调节剂和对与其相关的障碍的治疗
MX342326B (es) 2011-09-27 2016-09-26 Novartis Ag 3-pirimidin-4-il-oxazolidin-2-onas como inhibidoras de idh mutante.
CN103204816B (zh) 2012-01-16 2016-04-27 中国人民解放军军事医学科学院毒物药物研究所 哌嗪基嘧啶类衍生物及其制备方法和用途
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
CA2903979A1 (fr) 2013-03-14 2014-09-18 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones comme inhibiteurs d'idh mutante
CA3002540C (fr) 2015-01-06 2023-11-07 Arena Pharmaceuticals, Inc. Utilisation de (r)-2-(7-(4-cyclopentyl-3(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acide acetique pour le traitement de conditions liees au recepteur s1p1
JP6838744B2 (ja) 2015-06-22 2021-03-03 アリーナ ファーマシューティカルズ, インコーポレイテッド S1P1レセプター関連障害における使用のための(R)−2−(7−(4−シクロペンチル−3−(トリフルオロメチル)ベンジルオキシ)−1,2,3,4−テトラヒドロシクロペンタ[b]インドール−3−イル)酢酸(化合物1)の結晶性L−アルギニン塩
CN110520124A (zh) 2017-02-16 2019-11-29 艾尼纳制药公司 用于治疗原发性胆汁性胆管炎的化合物和方法
JP7397011B2 (ja) 2018-06-06 2023-12-12 アリーナ ファーマシューティカルズ, インコーポレイテッド S1p1受容体に関連する状態を治療する方法

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5075305A (en) * 1991-03-18 1991-12-24 Warner-Lambert Company Compound, composition and use
US5098902A (en) * 1991-03-18 1992-03-24 Warner-Lambert Company Method of treating neurodegenerative diseases

Also Published As

Publication number Publication date
ZA745305B (en) 1976-04-28
JPS5049288A (en) 1975-05-01
DE2341925A1 (de) 1975-03-06

Similar Documents

Publication Publication Date Title
AT338352B (de) Ohrstuck
BE813158A (fr) Nouvelles benzoquinolizines
ATA1023274A (de) Osteotom
FI56432B (fi) Gaskolv i skjutvapen
HU171312B (hu) Sposob poluchenija slozhnykh efirov n-fosfonometilglicina i karboksialkanolov
BE814229A (fr) Nouvelles azolylamidines
BE813142A (fr) Nouvelles piperazines disubstituees
AT325408B (de) Stoffloser
ATA446774A (de) Monoschi
BE819773A (fr) Nouvelles benzylpyrimidines
FR2295005A1 (fr) Nouvelles substances odoriferantes
DOP1974002166A (es) Antilidas heterociclicas
AT342382B (de) Flussmittel
BE793744A (fr) Gewapend bouwpaneel
BE817294A (fr) Nouvelles sulfonyloxyphenylurees
BE813677A (fr) Nouvelles triazolo-1
AT354042B (de) Raffstore
HU173131B (hu) Sposob i ustrojstvo poluchenija maleinovogo angidrida
BE813947A (fr) Nouvelles dichlorothiazolylurees
BE810364A (fr) Nouvelles benzoylphenylguanidines
BE818131A (fr) Nouvelles benzylpyrimidines
HU173009B (hu) Upakovka dlja obluchaemykh tovarov i sposob izgotovlenija takoj upakovki
BE821477A (fr) Nouvelles penicillines
IT1054123B (it) Fosfoserinato di piridossina
AT323390B (de) Türstock