BE904059A - Utilisation de derives d'isoquinoleine et de leurs sels pour la production de compositions pharmaceutiques - Google Patents
Utilisation de derives d'isoquinoleine et de leurs sels pour la production de compositions pharmaceutiquesInfo
- Publication number
- BE904059A BE904059A BE0/216148A BE216148A BE904059A BE 904059 A BE904059 A BE 904059A BE 0/216148 A BE0/216148 A BE 0/216148A BE 216148 A BE216148 A BE 216148A BE 904059 A BE904059 A BE 904059A
- Authority
- BE
- Belgium
- Prior art keywords
- production
- salts
- pharmaceutical compositions
- treatment
- release
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 238000000034 method Methods 0.000 abstract 4
- NTYJJOPFIAHURM-UHFFFAOYSA-N Histamine Chemical compound NCCC1=CN=CN1 NTYJJOPFIAHURM-UHFFFAOYSA-N 0.000 abstract 2
- 230000015572 biosynthetic process Effects 0.000 abstract 2
- -1 lipid peroxides Chemical class 0.000 abstract 2
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229960001340 histamine Drugs 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 125000002183 isoquinolinyl group Chemical class C1(=NC=CC2=CC=CC=C12)* 0.000 abstract 1
- 210000004185 liver Anatomy 0.000 abstract 1
- 230000002132 lysosomal effect Effects 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Procédé pour la préparation d'un médicament pour l'emploi dans un traitement inhibant la formation de peroxydes de lipides, la libération des enzymes lysosomiales, la production d'oxygène actif et/ou la libération d'histamine et procédé pour le traitement des affections associées à la formation de peroxydes de lipides et également un procédé perfectionné pour le traitement des affections hépatiques, lesdits procédés comprenant l'administration de quantités efficaces d'un dérivé d'isoquinoléine représenté par la formule générale I.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69230985A | 1985-01-17 | 1985-01-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE904059A true BE904059A (fr) | 1986-07-17 |
Family
ID=24780061
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/216148A BE904059A (fr) | 1985-01-17 | 1986-01-17 | Utilisation de derives d'isoquinoleine et de leurs sels pour la production de compositions pharmaceutiques |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0201359A3 (fr) |
| JP (2) | JPS61165326A (fr) |
| BE (1) | BE904059A (fr) |
| CH (2) | CH677731A5 (fr) |
| FR (1) | FR2578164B1 (fr) |
| IT (1) | IT1213024B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS63270678A (ja) * | 1987-04-30 | 1988-11-08 | Mitsui Petrochem Ind Ltd | 新規含窒素化合物 |
| US20050049278A1 (en) * | 2003-08-27 | 2005-03-03 | Youssef Bennani | Benzo[1,3]dioxole compounds, pharmaceutical compositions thereof, and processes of making and using the same |
| CN101735229A (zh) * | 2009-12-24 | 2010-06-16 | 沈阳药科大学 | 四氢异喹啉类化合物及其制备方法和用途 |
| FR3111071B1 (fr) * | 2020-06-04 | 2023-01-13 | H4 Orphan Pharma | Utilisation de ligands multifonctionnels pour traiter les syndromes de détresse respiratoire et le choc cytokinique liés aux infections virales à coronavirus. |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1206909B (de) * | 1959-08-14 | 1965-12-16 | Maurice Jeanson | Verfahren zur Herstellung von Inhibitoren der Histidindecarboxylase |
| FR2424271A1 (fr) * | 1978-04-28 | 1979-11-23 | Laire Chimie Sa De | Derives de phtalidyl-isoquinoleines, leur preparation et leur application comme medicaments |
| EP0028279B1 (fr) * | 1979-10-22 | 1983-02-16 | Calaire Chimie S.A. | Dérivés de phtalidyl-isoquinoléines, leur préparation et leur application comme médicaments |
-
1986
- 1986-01-14 JP JP61006118A patent/JPS61165326A/ja active Pending
- 1986-01-14 JP JP61006117A patent/JPS61165327A/ja active Pending
- 1986-01-17 EP EP86400095A patent/EP0201359A3/fr not_active Withdrawn
- 1986-01-17 CH CH2174/88A patent/CH677731A5/fr not_active IP Right Cessation
- 1986-01-17 IT IT8619100A patent/IT1213024B/it active
- 1986-01-17 BE BE0/216148A patent/BE904059A/fr not_active IP Right Cessation
- 1986-01-17 CH CH167/86A patent/CH670642A5/fr not_active IP Right Cessation
- 1986-01-17 FR FR868600651A patent/FR2578164B1/fr not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP0201359A3 (fr) | 1989-07-19 |
| FR2578164A1 (fr) | 1986-09-05 |
| JPS61165326A (ja) | 1986-07-26 |
| CH677731A5 (en) | 1991-06-28 |
| JPS61165327A (ja) | 1986-07-26 |
| CH670642A5 (fr) | 1989-06-30 |
| FR2578164B1 (fr) | 1990-08-10 |
| IT1213024B (it) | 1989-12-07 |
| EP0201359A2 (fr) | 1986-11-12 |
| IT8619100A0 (it) | 1986-01-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: MITSUBISHI HASEI CORP. Effective date: 19930131 |