BG102282A - Derivatives of 4-(cycloalkyl) piperidines and 4-(cycloalkylalkyl) piperidines, their preparation and application in medicine - Google Patents

Derivatives of 4-(cycloalkyl) piperidines and 4-(cycloalkylalkyl) piperidines, their preparation and application in medicine

Info

Publication number: BG102282A
Authority: BG; Bulgaria
Prior art keywords: piperidines; medicine; cycloalkyl; cycloalkylalkyl; derivatives
Prior art date: 1995-09-08

Application number

BG102282A

Other languages

Bulgarian (bg)

English (en)

Inventor

Patrick Lardenois

Jonathan Frost

Patrick Pasau

Pascal George

Maria RENONES

Regine Bartsch

Wai - Tak LI

Pascale Magat

Regis Dupont

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-09-08

Filing date

1998-02-26

Publication date

1998-09-30

1995-09-08 Priority claimed from FR9510513A external-priority patent/FR2738566B1/fr

1995-09-08 Priority claimed from FR9510512A external-priority patent/FR2738568B1/fr

1998-02-26 Application filed by Synthelabo filed Critical Synthelabo

1998-09-30 Publication of BG102282A publication Critical patent/BG102282A/xx

Links

239000003814 drug Substances 0.000 title abstract 3
150000003053 piperidines Chemical class 0.000 title 2
125000005843 halogen group Chemical group 0.000 abstract 2
WCYWZMWISLQXQU-UHFFFAOYSA-N methyl Chemical compound [CH3] WCYWZMWISLQXQU-UHFFFAOYSA-N 0.000 abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical group [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
125000004429 atom Chemical group 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
-1 cycloalkyl radical Chemical group 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
230000000508 neurotrophic effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/12—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with only hydrogen atoms attached to the ring nitrogen atom

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

BG102282A 1995-09-08 1998-02-26 Derivatives of 4-(cycloalkyl) piperidines and 4-(cycloalkylalkyl) piperidines, their preparation and application in medicine BG102282A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR9510513A FR2738566B1 (fr)	1995-09-08	1995-09-08	Derives de 4-(cycloalkyl)piperidines et de 4-(cycloalkylalkyl)piperidines, leur preparation et leur application en therapeutique
FR9510512A FR2738568B1 (fr)	1995-09-08	1995-09-08	Derives de 4-(cycloalkyl)piperidines et 4-(cycloalkylalkyl) piperidines, leur preparation et leur application en therapeutique
PCT/FR1996/001362 WO1997009309A1 (fr)	1995-09-08	1996-09-05	Derives de 4-(cycloalkyl)piperidines et de 4-(cycloalkylalkyl)pi peridines, leur preparation et leur application en therapeutique

Publications (1)

Publication Number	Publication Date
BG102282A true BG102282A (en)	1998-09-30

Family

ID=26232195

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG102282A BG102282A (en)	1995-09-08	1998-02-26	Derivatives of 4-(cycloalkyl) piperidines and 4-(cycloalkylalkyl) piperidines, their preparation and application in medicine

Country Status (25)

Country	Link
EP (1)	EP0848707B1 (de)
JP (1)	JPH11514975A (de)
KR (1)	KR19990044479A (de)
CN (1)	CN1201453A (de)
AR (1)	AR003530A1 (de)
AT (1)	ATE182885T1 (de)
AU (1)	AU703776B2 (de)
BG (1)	BG102282A (de)
BR (1)	BR9610408A (de)
CA (1)	CA2231326A1 (de)
CO (1)	CO4750660A1 (de)
CZ (1)	CZ66598A3 (de)
DE (1)	DE69603613T2 (de)
EE (1)	EE9800064A (de)
ES (1)	ES2137015T3 (de)
GR (1)	GR3031513T3 (de)
HU (1)	HUP9802938A2 (de)
IL (1)	IL123557A0 (de)
NO (1)	NO981000L (de)
NZ (1)	NZ316981A (de)
PL (1)	PL325421A1 (de)
SI (1)	SI0848707T1 (de)
SK (1)	SK31198A3 (de)
TR (1)	TR199800407T1 (de)
WO (1)	WO1997009309A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU727080B2 (en)	1997-06-30	2000-11-30	Allergan, Inc.	Calcium blockers to treat proliferative vitreoretinopathy
JP2002528416A (ja)	1998-10-27	2002-09-03	アルコンラボラトリーズ，インコーポレーテッド	外網膜の疾患の治療
CN1964627B (zh) *	2004-06-04	2011-10-19	华盛顿大学	治疗神经病变的方法和组合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4028366A (en) *	1975-01-20	1977-06-07	Sterling Drug Inc.	2-Naphthyl-lower-alkanoylamines
FR2640266B2 (fr) *	1988-07-12	1992-07-10	Synthelabo	Derives de (hydroxy-1 piperidinyl-2 alkyl) indolones-2, quinoleinones-2, benzo(b)azepinones-2 et benzimidazolones-2, leur preparation et leur application en therapeutique
FR2684379B1 (fr) *	1991-12-02	1995-04-28	Synthelabo	Derives de piperidine, leur preparation et leur application en therapeutique.
WO1994018172A1 (fr) *	1993-02-01	1994-08-18	Yoshitomi Pharmaceutical Industries, Ltd.	Compose d'imidazolylbenzene et son utilisation comme medicament

1996
- 1996-09-05 SI SI9630106T patent/SI0848707T1/xx unknown
- 1996-09-05 TR TR1998/00407T patent/TR199800407T1/xx unknown
- 1996-09-05 DE DE69603613T patent/DE69603613T2/de not_active Expired - Fee Related
- 1996-09-05 CA CA002231326A patent/CA2231326A1/en not_active Abandoned
- 1996-09-05 PL PL96325421A patent/PL325421A1/xx unknown
- 1996-09-05 EE EE9800064A patent/EE9800064A/xx unknown
- 1996-09-05 KR KR1019980701727A patent/KR19990044479A/ko not_active Withdrawn
- 1996-09-05 ES ES96930216T patent/ES2137015T3/es not_active Expired - Lifetime
- 1996-09-05 NZ NZ316981A patent/NZ316981A/xx unknown
- 1996-09-05 AU AU69344/96A patent/AU703776B2/en not_active Ceased
- 1996-09-05 CZ CZ98665A patent/CZ66598A3/cs unknown
- 1996-09-05 HU HU9802938A patent/HUP9802938A2/hu unknown
- 1996-09-05 JP JP9510910A patent/JPH11514975A/ja active Pending
- 1996-09-05 IL IL12355796A patent/IL123557A0/xx unknown
- 1996-09-05 CO CO96047348A patent/CO4750660A1/es unknown
- 1996-09-05 BR BR9610408A patent/BR9610408A/pt not_active Application Discontinuation
- 1996-09-05 AT AT96930216T patent/ATE182885T1/de active
- 1996-09-05 CN CN96198170A patent/CN1201453A/zh active Pending
- 1996-09-05 EP EP96930216A patent/EP0848707B1/de not_active Expired - Lifetime
- 1996-09-05 WO PCT/FR1996/001362 patent/WO1997009309A1/fr not_active Ceased
- 1996-09-05 SK SK311-98A patent/SK31198A3/sk unknown
- 1996-09-06 AR ARP960104270A patent/AR003530A1/es unknown
1998
- 1998-02-26 BG BG102282A patent/BG102282A/xx unknown
- 1998-03-06 NO NO981000A patent/NO981000L/no unknown
1999
- 1999-10-13 GR GR990402608T patent/GR3031513T3/el unknown

Also Published As

Publication number	Publication date
EP0848707A1 (de)	1998-06-24
KR19990044479A (ko)	1999-06-25
CO4750660A1 (es)	1999-03-31
EE9800064A (et)	1998-08-17
HUP9802938A2 (hu)	1999-10-28
MX9801838A (es)	1998-08-30
SI0848707T1 (en)	2000-02-29
AU6934496A (en)	1997-03-27
DE69603613T2 (de)	2000-03-02
NZ316981A (en)	1998-12-23
SK31198A3 (en)	1998-08-05
JPH11514975A (ja)	1999-12-21
ES2137015T3 (es)	1999-12-01
DE69603613D1 (de)	1999-09-09
PL325421A1 (en)	1998-07-20
NO981000L (no)	1998-05-08
EP0848707B1 (de)	1999-08-04
CN1201453A (zh)	1998-12-09
WO1997009309A1 (fr)	1997-03-13
ATE182885T1 (de)	1999-08-15
GR3031513T3 (en)	2000-01-31
BR9610408A (pt)	1999-07-06
AR003530A1 (es)	1998-08-05
IL123557A0 (en)	1998-10-30
CZ66598A3 (cs)	1998-06-17
NO981000D0 (no)	1998-03-06
AU703776B2 (en)	1999-04-01
CA2231326A1 (en)	1997-03-13
TR199800407T1 (xx)	1998-05-21

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