BG102484A - Method for the preparation of dioxoazabicyclohexanes - Google Patents

Method for the preparation of dioxoazabicyclohexanes

Info

Publication number: BG102484A
Authority: BG; Bulgaria
Prior art keywords: formulawhere; alkyl; potassium; benzyl; dioxoazabicyclohexanes
Prior art date: 1995-11-30

Application number

BG102484A

Other languages

Bulgarian (bg)

English (en)

Inventor

Stephen Ray

John RUMPUS

Original Assignee

Pfizer Research And Development Company, N.V./S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-11-30

Filing date

1998-05-25

Publication date

1999-03-31

1998-05-25 Application filed by Pfizer Research And Development Company, N.V./S.A. filed Critical Pfizer Research And Development Company, N.V./S.A.

1999-03-31 Publication of BG102484A publication Critical patent/BG102484A/xx

Links

HGCBTXNRSHFSOF-UHFFFAOYSA-N 1-cyclohexylpiperidine-2,3-dione Chemical class O=C1C(=O)CCCN1C1CCCCC1 HGCBTXNRSHFSOF-UHFFFAOYSA-N 0.000 title 1
WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 abstract 3
ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 abstract 3
CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 abstract 2
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
FJDQFPXHSGXQBY-UHFFFAOYSA-L caesium carbonate Chemical compound [Cs+].[Cs+].[O-]C([O-])=O FJDQFPXHSGXQBY-UHFFFAOYSA-L 0.000 abstract 2
239000003960 organic solvent Substances 0.000 abstract 2
NROKBHXJSPEDAR-UHFFFAOYSA-M potassium fluoride Chemical compound [F-].[K+] NROKBHXJSPEDAR-UHFFFAOYSA-M 0.000 abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
XTHFKEDIFFGKHM-UHFFFAOYSA-N Dimethoxyethane Chemical compound COCCOC XTHFKEDIFFGKHM-UHFFFAOYSA-N 0.000 abstract 1
IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 abstract 1
DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 abstract 1
ZLMJMSJWJFRBEC-UHFFFAOYSA-N Potassium Chemical compound [K] ZLMJMSJWJFRBEC-UHFFFAOYSA-N 0.000 abstract 1
229910000024 caesium carbonate Inorganic materials 0.000 abstract 1
229960001760 dimethyl sulfoxide Drugs 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
BWHMMNNQKKPAPP-UHFFFAOYSA-L potassium carbonate Substances [K+].[K+].[O-]C([O-])=O BWHMMNNQKKPAPP-UHFFFAOYSA-L 0.000 abstract 1
229910000027 potassium carbonate Inorganic materials 0.000 abstract 1
239000011698 potassium fluoride Substances 0.000 abstract 1
235000003270 potassium fluoride Nutrition 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
239000011541 reaction mixture Substances 0.000 abstract 1
CDBYLPFSWZWCQE-UHFFFAOYSA-L sodium carbonate Substances [Na+].[Na+].[O-]C([O-])=O CDBYLPFSWZWCQE-UHFFFAOYSA-L 0.000 abstract 1
229910000029 sodium carbonate Inorganic materials 0.000 abstract 1
239000001488 sodium phosphate Substances 0.000 abstract 1
RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 abstract 1
229910000406 trisodium phosphate Inorganic materials 0.000 abstract 1
235000019801 trisodium phosphate Nutrition 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Indole Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

BG102484A 1995-11-30 1998-05-25 Method for the preparation of dioxoazabicyclohexanes BG102484A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB9524466.1A GB9524466D0 (en)	1995-11-30	1995-11-30	Process
PCT/EP1996/004782 WO1997019921A1 (fr)	1995-11-30	1996-10-31	Procede pour preparer de dioxoazabicyclohexanes

Publications (1)

Publication Number	Publication Date
BG102484A true BG102484A (en)	1999-03-31

Family

ID=10784676

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG102484A BG102484A (en)	1995-11-30	1998-05-25	Method for the preparation of dioxoazabicyclohexanes

Country Status (40)

Country	Link
EP (1)	EP0863874B1 (fr)
JP (1)	JP2000507919A (fr)
KR (1)	KR100286157B1 (fr)
CN (1)	CN1203588A (fr)
AP (1)	AP746A (fr)
AR (1)	AR004766A1 (fr)
AT (1)	ATE198325T1 (fr)
AU (1)	AU707221B2 (fr)
BG (1)	BG102484A (fr)
BR (1)	BR9611833A (fr)
CA (1)	CA2231590A1 (fr)
CO (1)	CO4480102A1 (fr)
CZ (1)	CZ162298A3 (fr)
DE (1)	DE69611380T2 (fr)
DK (1)	DK0863874T3 (fr)
ES (1)	ES2152571T3 (fr)
GB (1)	GB9524466D0 (fr)
GR (1)	GR3035341T3 (fr)
HR (1)	HRP960555A2 (fr)
HU (1)	HUP9903571A3 (fr)
IL (1)	IL123561A0 (fr)
IS (1)	IS4707A (fr)
MA (1)	MA24015A1 (fr)
MX (1)	MX9804311A (fr)
MY (1)	MY132595A (fr)
NO (1)	NO982503L (fr)
NZ (1)	NZ321968A (fr)
OA (1)	OA10692A (fr)
PE (1)	PE24898A1 (fr)
PL (1)	PL326978A1 (fr)
PT (1)	PT863874E (fr)
RU (1)	RU2156238C2 (fr)
SK (1)	SK70798A3 (fr)
TN (1)	TNSN96145A1 (fr)
TR (1)	TR199800957T2 (fr)
TW (1)	TW401397B (fr)
UY (1)	UY24379A1 (fr)
WO (1)	WO1997019921A1 (fr)
YU (1)	YU63196A (fr)
ZA (1)	ZA9610053B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH1087617A (ja) *	1996-07-09	1998-04-07	Pfizer Inc	キノリン系抗生物質の合成に有用な中間体の製法
HN1998000106A (es)	1997-08-01	1999-01-08	Pfizer Prod Inc	Composiciones parenterales de alatroflaxacino
US7019142B2 (en)	1998-01-16	2006-03-28	Pfizer Inc.	Process for preparing naphthyridones and intermediates
CN1320360C (zh) *	2002-03-25	2007-06-06	科学和工业研究委员会	超酸性植物的蛋白图谱
NL2000192C2 (nl) *	2006-08-23	2008-02-26	Veenvoort B V De	Stabiel bitumenschuim en de bereiding en het gebruik ervan.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5256791A (en) *	1992-03-02	1993-10-26	Pfizer Inc.	Preparation of intermediates in the synthesis of quinoline antibiotics
RU2147303C1 (ru) *	1994-01-18	2000-04-10	Пфайзер Инк.	Промежуточные продукты и способ получения солей нафтиридонкарбоновой кислоты

1995
- 1995-11-30 GB GBGB9524466.1A patent/GB9524466D0/en active Pending
1996
- 1996-10-21 TW TW085112856A patent/TW401397B/zh not_active IP Right Cessation
- 1996-10-31 DK DK96938058T patent/DK0863874T3/da active
- 1996-10-31 CZ CZ981622A patent/CZ162298A3/cs unknown
- 1996-10-31 JP JP9520100A patent/JP2000507919A/ja active Pending
- 1996-10-31 TR TR1998/00957T patent/TR199800957T2/xx unknown
- 1996-10-31 BR BR9611833A patent/BR9611833A/pt not_active Application Discontinuation
- 1996-10-31 AU AU75629/96A patent/AU707221B2/en not_active Ceased
- 1996-10-31 WO PCT/EP1996/004782 patent/WO1997019921A1/fr not_active Ceased
- 1996-10-31 HU HU9903571A patent/HUP9903571A3/hu unknown
- 1996-10-31 KR KR1019980703892A patent/KR100286157B1/ko not_active Expired - Fee Related
- 1996-10-31 PL PL96326978A patent/PL326978A1/xx unknown
- 1996-10-31 PT PT96938058T patent/PT863874E/pt unknown
- 1996-10-31 IL IL12356196A patent/IL123561A0/xx unknown
- 1996-10-31 ES ES96938058T patent/ES2152571T3/es not_active Expired - Lifetime
- 1996-10-31 NZ NZ321968A patent/NZ321968A/xx unknown
- 1996-10-31 SK SK707-98A patent/SK70798A3/sk unknown
- 1996-10-31 CN CN96198667A patent/CN1203588A/zh active Pending
- 1996-10-31 CA CA002231590A patent/CA2231590A1/fr not_active Abandoned
- 1996-10-31 EP EP96938058A patent/EP0863874B1/fr not_active Expired - Lifetime
- 1996-10-31 RU RU98112016/04A patent/RU2156238C2/ru active
- 1996-10-31 AT AT96938058T patent/ATE198325T1/de not_active IP Right Cessation
- 1996-10-31 DE DE69611380T patent/DE69611380T2/de not_active Expired - Fee Related
- 1996-11-21 HR HR9524466.1A patent/HRP960555A2/hr not_active Application Discontinuation
- 1996-11-27 PE PE1996000850A patent/PE24898A1/es not_active Application Discontinuation
- 1996-11-27 UY UY24379A patent/UY24379A1/es not_active IP Right Cessation
- 1996-11-27 AR ARP960105343A patent/AR004766A1/es unknown
- 1996-11-27 TN TNTNSN96145A patent/TNSN96145A1/fr unknown
- 1996-11-27 MA MA24403A patent/MA24015A1/fr unknown
- 1996-11-28 YU YU63196A patent/YU63196A/sh unknown
- 1996-11-28 AP APAP/P/1996/000885A patent/AP746A/en active
- 1996-11-28 CO CO96062767A patent/CO4480102A1/es unknown
- 1996-11-29 MY MYPI96005005A patent/MY132595A/en unknown
- 1996-11-29 ZA ZA9610053A patent/ZA9610053B/xx unknown
1998
- 1998-03-31 IS IS4707A patent/IS4707A/is unknown
- 1998-05-25 BG BG102484A patent/BG102484A/xx unknown
- 1998-05-29 OA OA9800068A patent/OA10692A/en unknown
- 1998-05-29 MX MX9804311A patent/MX9804311A/es unknown
- 1998-06-02 NO NO982503A patent/NO982503L/no not_active Application Discontinuation
2001
- 2001-02-01 GR GR20010400166T patent/GR3035341T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
MY132595A (en)	2007-10-31
TR199800957T2 (xx)	1998-09-21
IL123561A0 (en)	1998-10-30
HUP9903571A3 (en)	2001-01-29
YU63196A (sh)	1998-11-05
GB9524466D0 (en)	1996-01-31
AP746A (en)	1999-04-29
DE69611380D1 (de)	2001-02-01
AR004766A1 (es)	1999-03-10
NO982503D0 (no)	1998-06-02
PE24898A1 (es)	1998-06-02
EP0863874B1 (fr)	2000-12-27
BR9611833A (pt)	1999-03-09
CO4480102A1 (es)	1997-07-09
TW401397B (en)	2000-08-11
AU707221B2 (en)	1999-07-08
CN1203588A (zh)	1998-12-30
KR19990071616A (ko)	1999-09-27
PL326978A1 (en)	1998-11-09
GR3035341T3 (en)	2001-05-31
PT863874E (pt)	2001-04-30
HUP9903571A2 (hu)	2000-03-28
ZA9610053B (en)	1998-05-29
NZ321968A (en)	1999-05-28
JP2000507919A (ja)	2000-06-27
ES2152571T3 (es)	2001-02-01
HRP960555A2 (en)	1998-02-28
MA24015A1 (fr)	1997-07-01
AP9600885A0 (en)	1997-01-31
IS4707A (is)	1998-03-31
SK70798A3 (en)	1999-06-11
NO982503L (no)	1998-06-02
AU7562996A (en)	1997-06-19
CA2231590A1 (fr)	1997-06-05
WO1997019921A1 (fr)	1997-06-05
RU2156238C2 (ru)	2000-09-20
TNSN96145A1 (fr)	2005-03-15
OA10692A (en)	2000-11-06
UY24379A1 (es)	1997-05-20
EP0863874A1 (fr)	1998-09-16
KR100286157B1 (ko)	2001-04-16
MX9804311A (es)	1998-09-30
CZ162298A3 (cs)	1999-03-17
DE69611380T2 (de)	2001-04-26
DK0863874T3 (da)	2001-01-29
ATE198325T1 (de)	2001-01-15

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