BG102484A - Method for the preparation of dioxoazabicyclohexanes - Google Patents

Method for the preparation of dioxoazabicyclohexanes

Info

Publication number: BG102484A
Authority: BG; Bulgaria
Prior art keywords: formulawhere; alkyl; potassium; benzyl; dioxoazabicyclohexanes
Prior art date: 1995-11-30

Application number

BG102484A

Other languages

Bulgarian (bg)

English (en)

Inventor

Stephen Ray

John RUMPUS

Original Assignee

Pfizer Research And Development Company, N.V./S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-11-30

Filing date

1998-05-25

Publication date

1999-03-31

1998-05-25 Application filed by Pfizer Research And Development Company, N.V./S.A. filed Critical Pfizer Research And Development Company, N.V./S.A.

1999-03-31 Publication of BG102484A publication Critical patent/BG102484A/xx

Links

HGCBTXNRSHFSOF-UHFFFAOYSA-N 1-cyclohexylpiperidine-2,3-dione Chemical class O=C1C(=O)CCCN1C1CCCCC1 HGCBTXNRSHFSOF-UHFFFAOYSA-N 0.000 title 1
WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 abstract 3
ZMXDDKWLCZADIW-UHFFFAOYSA-N N,N-Dimethylformamide Chemical compound CN(C)C=O ZMXDDKWLCZADIW-UHFFFAOYSA-N 0.000 abstract 3
CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 abstract 2
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
FJDQFPXHSGXQBY-UHFFFAOYSA-L caesium carbonate Chemical compound [Cs+].[Cs+].[O-]C([O-])=O FJDQFPXHSGXQBY-UHFFFAOYSA-L 0.000 abstract 2
239000003960 organic solvent Substances 0.000 abstract 2
NROKBHXJSPEDAR-UHFFFAOYSA-M potassium fluoride Chemical compound [F-].[K+] NROKBHXJSPEDAR-UHFFFAOYSA-M 0.000 abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
XTHFKEDIFFGKHM-UHFFFAOYSA-N Dimethoxyethane Chemical compound COCCOC XTHFKEDIFFGKHM-UHFFFAOYSA-N 0.000 abstract 1
IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 abstract 1
DGAQECJNVWCQMB-PUAWFVPOSA-M Ilexoside XXIX Chemical compound C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)OS(=O)(=O)[O-])C)C)[C@@H]2[C@]1(C)O)C)C(=O)O[C@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O.[Na+] DGAQECJNVWCQMB-PUAWFVPOSA-M 0.000 abstract 1
ZLMJMSJWJFRBEC-UHFFFAOYSA-N Potassium Chemical compound [K] ZLMJMSJWJFRBEC-UHFFFAOYSA-N 0.000 abstract 1
229910000024 caesium carbonate Inorganic materials 0.000 abstract 1
229960001760 dimethyl sulfoxide Drugs 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
BWHMMNNQKKPAPP-UHFFFAOYSA-L potassium carbonate Substances [K+].[K+].[O-]C([O-])=O BWHMMNNQKKPAPP-UHFFFAOYSA-L 0.000 abstract 1
229910000027 potassium carbonate Inorganic materials 0.000 abstract 1
239000011698 potassium fluoride Substances 0.000 abstract 1
235000003270 potassium fluoride Nutrition 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
239000011541 reaction mixture Substances 0.000 abstract 1
CDBYLPFSWZWCQE-UHFFFAOYSA-L sodium carbonate Substances [Na+].[Na+].[O-]C([O-])=O CDBYLPFSWZWCQE-UHFFFAOYSA-L 0.000 abstract 1
229910000029 sodium carbonate Inorganic materials 0.000 abstract 1
239000001488 sodium phosphate Substances 0.000 abstract 1
RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 abstract 1
229910000406 trisodium phosphate Inorganic materials 0.000 abstract 1
235000019801 trisodium phosphate Nutrition 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Indole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

BG102484A 1995-11-30 1998-05-25 Method for the preparation of dioxoazabicyclohexanes BG102484A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB9524466.1A GB9524466D0 (en)	1995-11-30	1995-11-30	Process
PCT/EP1996/004782 WO1997019921A1 (fr)	1995-11-30	1996-10-31	Procede pour preparer de dioxoazabicyclohexanes

Publications (1)

Publication Number	Publication Date
BG102484A true BG102484A (en)	1999-03-31

Family

ID=10784676

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG102484A BG102484A (en)	1995-11-30	1998-05-25	Method for the preparation of dioxoazabicyclohexanes

Country Status (40)

Country	Link
EP (1)	EP0863874B1 (fr)
JP (1)	JP2000507919A (fr)
KR (1)	KR100286157B1 (fr)
CN (1)	CN1203588A (fr)
AP (1)	AP746A (fr)
AR (1)	AR004766A1 (fr)
AT (1)	ATE198325T1 (fr)
AU (1)	AU707221B2 (fr)
BG (1)	BG102484A (fr)
BR (1)	BR9611833A (fr)
CA (1)	CA2231590A1 (fr)
CO (1)	CO4480102A1 (fr)
CZ (1)	CZ162298A3 (fr)
DE (1)	DE69611380T2 (fr)
DK (1)	DK0863874T3 (fr)
ES (1)	ES2152571T3 (fr)
GB (1)	GB9524466D0 (fr)
GR (1)	GR3035341T3 (fr)
HR (1)	HRP960555A2 (fr)
HU (1)	HUP9903571A3 (fr)
IL (1)	IL123561A0 (fr)
IS (1)	IS4707A (fr)
MA (1)	MA24015A1 (fr)
MX (1)	MX9804311A (fr)
MY (1)	MY132595A (fr)
NO (1)	NO982503L (fr)
NZ (1)	NZ321968A (fr)
OA (1)	OA10692A (fr)
PE (1)	PE24898A1 (fr)
PL (1)	PL326978A1 (fr)
PT (1)	PT863874E (fr)
RU (1)	RU2156238C2 (fr)
SK (1)	SK70798A3 (fr)
TN (1)	TNSN96145A1 (fr)
TR (1)	TR199800957T2 (fr)
TW (1)	TW401397B (fr)
UY (1)	UY24379A1 (fr)
WO (1)	WO1997019921A1 (fr)
YU (1)	YU63196A (fr)
ZA (1)	ZA9610053B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH1087617A (ja) *	1996-07-09	1998-04-07	Pfizer Inc	キノリン系抗生物質の合成に有用な中間体の製法
HN1998000106A (es)	1997-08-01	1999-01-08	Pfizer Prod Inc	Composiciones parenterales de alatroflaxacino
US7019142B2 (en)	1998-01-16	2006-03-28	Pfizer Inc.	Process for preparing naphthyridones and intermediates
BR0215659A (pt) *	2002-03-25	2005-01-25	Council Scient Ind Res	Perfilamento de proteìnas de plantas hiper acìdicas
NL2000192C2 (nl) *	2006-08-23	2008-02-26	Veenvoort B V De	Stabiel bitumenschuim en de bereiding en het gebruik ervan.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5256791A (en) *	1992-03-02	1993-10-26	Pfizer Inc.	Preparation of intermediates in the synthesis of quinoline antibiotics
CZ286896B6 (en) *	1994-01-18	2000-07-12	Pfizer	Process for preparing pharmaceutically acceptable salts of naphthyridone carboxylic acid and intermediates for this preparation

1995
- 1995-11-30 GB GBGB9524466.1A patent/GB9524466D0/en active Pending
1996
- 1996-10-21 TW TW085112856A patent/TW401397B/zh not_active IP Right Cessation
- 1996-10-31 SK SK707-98A patent/SK70798A3/sk unknown
- 1996-10-31 PL PL96326978A patent/PL326978A1/xx unknown
- 1996-10-31 EP EP96938058A patent/EP0863874B1/fr not_active Expired - Lifetime
- 1996-10-31 DK DK96938058T patent/DK0863874T3/da active
- 1996-10-31 HU HU9903571A patent/HUP9903571A3/hu unknown
- 1996-10-31 KR KR1019980703892A patent/KR100286157B1/ko not_active Expired - Fee Related
- 1996-10-31 CZ CZ981622A patent/CZ162298A3/cs unknown
- 1996-10-31 RU RU98112016/04A patent/RU2156238C2/ru active
- 1996-10-31 CA CA002231590A patent/CA2231590A1/fr not_active Abandoned
- 1996-10-31 TR TR1998/00957T patent/TR199800957T2/xx unknown
- 1996-10-31 WO PCT/EP1996/004782 patent/WO1997019921A1/fr not_active Ceased
- 1996-10-31 AU AU75629/96A patent/AU707221B2/en not_active Ceased
- 1996-10-31 ES ES96938058T patent/ES2152571T3/es not_active Expired - Lifetime
- 1996-10-31 JP JP9520100A patent/JP2000507919A/ja active Pending
- 1996-10-31 BR BR9611833A patent/BR9611833A/pt not_active Application Discontinuation
- 1996-10-31 CN CN96198667A patent/CN1203588A/zh active Pending
- 1996-10-31 DE DE69611380T patent/DE69611380T2/de not_active Expired - Fee Related
- 1996-10-31 NZ NZ321968A patent/NZ321968A/xx unknown
- 1996-10-31 AT AT96938058T patent/ATE198325T1/de not_active IP Right Cessation
- 1996-10-31 PT PT96938058T patent/PT863874E/pt unknown
- 1996-10-31 IL IL12356196A patent/IL123561A0/xx unknown
- 1996-11-21 HR HR9524466.1A patent/HRP960555A2/hr not_active Application Discontinuation
- 1996-11-27 TN TNTNSN96145A patent/TNSN96145A1/fr unknown
- 1996-11-27 AR ARP960105343A patent/AR004766A1/es unknown
- 1996-11-27 MA MA24403A patent/MA24015A1/fr unknown
- 1996-11-27 UY UY24379A patent/UY24379A1/es not_active IP Right Cessation
- 1996-11-27 PE PE1996000850A patent/PE24898A1/es not_active Application Discontinuation
- 1996-11-28 CO CO96062767A patent/CO4480102A1/es unknown
- 1996-11-28 AP APAP/P/1996/000885A patent/AP746A/en active
- 1996-11-28 YU YU63196A patent/YU63196A/sh unknown
- 1996-11-29 MY MYPI96005005A patent/MY132595A/en unknown
- 1996-11-29 ZA ZA9610053A patent/ZA9610053B/xx unknown
1998
- 1998-03-31 IS IS4707A patent/IS4707A/is unknown
- 1998-05-25 BG BG102484A patent/BG102484A/xx unknown
- 1998-05-29 OA OA9800068A patent/OA10692A/en unknown
- 1998-05-29 MX MX9804311A patent/MX9804311A/es unknown
- 1998-06-02 NO NO982503A patent/NO982503L/no not_active Application Discontinuation
2001
- 2001-02-01 GR GR20010400166T patent/GR3035341T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
PT863874E (pt)	2001-04-30
TR199800957T2 (xx)	1998-09-21
EP0863874A1 (fr)	1998-09-16
AR004766A1 (es)	1999-03-10
MA24015A1 (fr)	1997-07-01
EP0863874B1 (fr)	2000-12-27
WO1997019921A1 (fr)	1997-06-05
NZ321968A (en)	1999-05-28
IL123561A0 (en)	1998-10-30
DE69611380T2 (de)	2001-04-26
ATE198325T1 (de)	2001-01-15
CA2231590A1 (fr)	1997-06-05
HUP9903571A3 (en)	2001-01-29
TNSN96145A1 (fr)	2005-03-15
CO4480102A1 (es)	1997-07-09
CZ162298A3 (cs)	1999-03-17
SK70798A3 (en)	1999-06-11
CN1203588A (zh)	1998-12-30
GB9524466D0 (en)	1996-01-31
DE69611380D1 (de)	2001-02-01
AU707221B2 (en)	1999-07-08
OA10692A (en)	2000-11-06
MX9804311A (es)	1998-09-30
AP746A (en)	1999-04-29
YU63196A (sh)	1998-11-05
PE24898A1 (es)	1998-06-02
PL326978A1 (en)	1998-11-09
ZA9610053B (en)	1998-05-29
IS4707A (is)	1998-03-31
HRP960555A2 (en)	1998-02-28
NO982503D0 (no)	1998-06-02
TW401397B (en)	2000-08-11
MY132595A (en)	2007-10-31
KR100286157B1 (ko)	2001-04-16
BR9611833A (pt)	1999-03-09
RU2156238C2 (ru)	2000-09-20
GR3035341T3 (en)	2001-05-31
HUP9903571A2 (hu)	2000-03-28
UY24379A1 (es)	1997-05-20
AU7562996A (en)	1997-06-19
AP9600885A0 (en)	1997-01-31
DK0863874T3 (da)	2001-01-29
ES2152571T3 (es)	2001-02-01
KR19990071616A (ko)	1999-09-27
NO982503L (no)	1998-06-02
JP2000507919A (ja)	2000-06-27

Publication	Publication Date	Title
DK0981525T3 (da)	2004-05-10	(2-(2-Thienyl)-ethylamino)-(2-halophenyl)-acetonitriler som mellemprodukter og fremgangsmåde til deres fremstilling
BG102484A (en)	1999-03-31	Method for the preparation of dioxoazabicyclohexanes
CA2270386A1 (fr)	1998-05-22	Procede de preparation de pyridines substituees
AU2923384A (en)	1984-12-13	Nitro-substituted benzotrifluorides
SE8601646D0 (sv)	1986-04-11	Intermediates for the production of epipodophyllotoxin and related compounds and processes for the preparation and use thereof
ZA9410023B (en)	1995-09-29	Herbicides
JPS6416791A (en)	1989-01-20	Guanidine related compound containing substituted tetraphenylborate ion and its production
TR199900321T2 (xx)	1999-04-21	N-(1-nbutil - 4 - piperidil)metil) -3,4-dihidro -2H- (1,3) oksazino (3.2A) indol-10- Karboksamit haz�rlama prosesi ve prosesteki tuzlar ve ara �r�nler.
ES8307751A1 (es)	1983-07-01	"un procedimiento para la preparacion de derivados de piridinona".
GR851657B (fr)	1985-11-26
AU2646897A (en)	1997-11-19	Process for the preparation of fluoro compounds from the corresponding amines
ES2151077T3 (es)	2000-12-16	Procedimiento para la obtencion de imidazolidinonas 1,3-disubstituidas.
EP0169051A3 (fr)	1986-12-10	Composés de pyridazinylurées
DK0727423T3 (da)	2001-09-24	Fremgangsmåde til fremstilling af sulfonylurinstofderivater og mellemprodukter til denne fremgangsmåde
IL128186A0 (en)	1999-11-30	Intermediates for the preparation of 2-imidazoline-5-ones
EA199800242A1 (ru)	1998-08-27	Амиды карбамоилкарбоновой кислоты
BG103651A (en)	2000-02-29	Compounds and methods for the preparation of substituted 4-phenyl-4-cyanocyclohexanoic acids
CA2194119A1 (fr)	1997-07-06	Methode pour preparer des derives de substitution en 2 de 5-chloro-imidazole-4-c_arbaldehydes
AU8055887A (en)	1988-02-18	Compounds useful as intermediates for the production of substituted 1-pyridlyoxy-3-indolyalkylamino-2-propanols
GB9713292D0 (en)	1997-08-27	Novel cation receptor
IL86722A (en)	1993-01-31	Guanidine-related compounds comprising a tetraphenylborate ion and their preparation
AU546890B2 (en)	1985-09-26	4-aminomethyl-5-acyl-1,3 dihydro-2h-imidazol-2-ones
GEP19981332B (en)	1998-07-06	Derivatives of acrylic acid
AU547243B2 (en)	1985-10-10	5-aminomethyl-2,3-dihydro-2-oxo-1h-imidazole-4-carboxylic acid derivatives
HUP0000144A2 (hu)	2000-06-28	Eljárás hidroxi-heteroaromás vegyületek aril-aminokká való átalakítására