BG103180A - Метод за лечение на сърдечна недостатъчност - Google Patents

Метод за лечение на сърдечна недостатъчност Download PDF

Info

Publication number: BG103180A
Authority: BG; Bulgaria
Prior art keywords: dimethyl; phenoxy; trimethyl; ethyl; propoxy
Prior art date: 1998-02-17

Application number

BG103180A

Other languages

Bulgarian (bg)

English (en)

Inventor

Yuhpyng Chen

Anthony FOSSA

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-02-17

Filing date

1999-02-16

Publication date

1999-09-30

1999-02-16 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

1999-09-30 Publication of BG103180A publication Critical patent/BG103180A/bg

Links

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QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
229960000281 trometamol Drugs 0.000 description 1
231100000397 ulcer Toxicity 0.000 description 1
230000002861 ventricular Effects 0.000 description 1
238000010792 warming Methods 0.000 description 1
238000005303 weighing Methods 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

BG103180A 1998-02-17 1999-02-16 Метод за лечение на сърдечна недостатъчност BG103180A (bg)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US7493498P	1998-02-17	1998-02-17

Publications (1)

Publication Number	Publication Date
BG103180A true BG103180A (bg)	1999-09-30

Family

ID=22122537

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG103180A BG103180A (bg)	1998-02-17	1999-02-16	Метод за лечение на сърдечна недостатъчност

Country Status (28)

Country	Link
US (1)	US6043260A (fr)
EP (1)	EP0951906A1 (fr)
JP (1)	JPH11292766A (fr)
KR (1)	KR19990072616A (fr)
CN (1)	CN1231176A (fr)
AP (1)	AP9901464A0 (fr)
AR (1)	AR017723A1 (fr)
AU (1)	AU1732999A (fr)
BG (1)	BG103180A (fr)
BR (1)	BR9900653A (fr)
CA (1)	CA2262252C (fr)
EA (1)	EA199900124A3 (fr)
GT (1)	GT199900015A (fr)
HR (1)	HRP990054A2 (fr)
HU (1)	HUP9900386A3 (fr)
ID (1)	ID23218A (fr)
IL (1)	IL128531A0 (fr)
IS (1)	IS4975A (fr)
MA (1)	MA26608A1 (fr)
NO (1)	NO990722L (fr)
OA (1)	OA10976A (fr)
PA (1)	PA8467401A1 (fr)
PE (1)	PE20000266A1 (fr)
PL (1)	PL331507A1 (fr)
SG (1)	SG81261A1 (fr)
TN (1)	TNSN99024A1 (fr)
TR (1)	TR199900328A2 (fr)
ZA (1)	ZA991220B (fr)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
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US7125880B1 (en)	1995-06-06	2006-10-24	Pfizer Inc.	Corticotropin releasing factor antagonists
US6956047B1 (en)	1995-06-06	2005-10-18	Pfizer Inc.	Corticotropin releasing factor antagonists
US6403599B1 (en)	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
US6387894B1 (en) *	1999-06-11	2002-05-14	Pfizer Inc.	Use of CRF antagonists and renin-angiotensin system inhibitors
AU7604400A (en)	1999-09-21	2001-04-24	Emory University	Methods and compositions for treating platelet-related disorders using mpl pathway inhibitory agents
KR20020063934A (ko) *	2000-01-18	2002-08-07	화이자 프로덕츠 인코포레이티드	코르티코트로핀 방출 인자 길항제
US6737430B2 (en)	2000-11-09	2004-05-18	Pfizer, Inc.	Mutual prodrug of amlodipine and atorvastatin
GB0027410D0 (en) *	2000-11-09	2000-12-27	Pfizer Ltd	Mutual prodrug of amlodipine and atorvastatin
US6992087B2 (en)	2001-11-21	2006-01-31	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
US7015229B2 (en)	2002-02-22	2006-03-21	Pfizer Inc	Substituted pyrimidinones and pyrimidinthiones
AU2003220190A1 (en) *	2002-03-13	2003-09-29	Pharmacia & Upjohn Company Llc	Pyrazolo(1,5-a)pyridine derivatives as neurotransmitter modulators
JP2005533014A (ja) *	2002-04-26	2005-11-04	ファルマシア・アンド・アップジョン・カンパニー・エルエルシー	置換ピラジン誘導体
JP2006506350A (ja) *	2002-09-12	2006-02-23	ファルマシア・アンド・アップジョン・カンパニー・エルエルシー	置換１，４−ピラジン誘導体
AR041470A1 (es) *	2002-10-17	2005-05-18	Upjohn Co	Compuestos de pirrolo (1,2 - b) piridazina y sus usos
EP1565454A1 (fr) *	2002-11-21	2005-08-24	Pharmacia & Upjohn Company LLC	Composes de pyrazine en tant que modulateurs de crf
BRPI0409649A (pt) *	2003-04-23	2006-04-25	Pharmacia & Upjohn Co Llc	pirimidinonas e pirimidinotionas substituìdas como antagonistas de crf
MXPA05011993A (es) *	2003-05-07	2006-02-02	Pharmacia & Upjohn Co Llc	Compuestos de pirrolo[1,2-b]piridazina.
EP1625125A1 (fr) *	2003-05-09	2006-02-15	Pharmacia & Upjohn Company LLC	Composes utilises comme antagonistes du recepteur de type 1 de la corticoliberine (crf)
MXPA05012081A (es) *	2003-05-09	2006-02-22	Pharmacia & Upjohn Co Llc	Derivados de pirimidina sustituidos.
EP1626965A1 (fr) *	2003-05-09	2006-02-22	Pharmacia & Upjohn Company LLC	Pyrazinones a titre d'antagonistes du recepteur de crf1 dans le traitement des troubles du systeme nerveux central
WO2005089639A2 (fr) *	2004-03-16	2005-09-29	Talarico M D Matthew T	Procede de deregulation vasculaire
US20060211710A1 (en) *	2005-03-17	2006-09-21	Pfizer Inc	Substituted aryl 1,4-pyrazine derivatives
US8338441B2 (en) *	2009-05-15	2012-12-25	Gilead Sciences, Inc.	Inhibitors of human immunodeficiency virus replication

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW574214B (en) *	1994-06-08	2004-02-01	Pfizer	Corticotropin releasing factor antagonists
US6403599B1 (en) *	1995-11-08	2002-06-11	Pfizer Inc	Corticotropin releasing factor antagonists
EP0795327A1 (fr) *	1996-03-13	1997-09-17	Pfizer Inc.	Utilisation de l'amlodipine pour le traitement et la prophylaxie de l'insuffisance cardiaque congestive d'origine non-ischémique

1999
- 1999-01-18 PA PA19998467401A patent/PA8467401A1/es unknown
- 1999-02-02 GT GT199900015A patent/GT199900015A/es unknown
- 1999-02-10 US US09/248,073 patent/US6043260A/en not_active Expired - Fee Related
- 1999-02-10 SG SG9900526A patent/SG81261A1/en unknown
- 1999-02-11 EP EP99301006A patent/EP0951906A1/fr not_active Withdrawn
- 1999-02-11 CN CN99102122A patent/CN1231176A/zh active Pending
- 1999-02-11 IS IS4975A patent/IS4975A/is unknown
- 1999-02-11 AP APAP/P/1999/001464A patent/AP9901464A0/en unknown
- 1999-02-12 KR KR1019990004934A patent/KR19990072616A/ko not_active Ceased
- 1999-02-12 PE PE1999000127A patent/PE20000266A1/es not_active Application Discontinuation
- 1999-02-12 BR BR9900653-7A patent/BR9900653A/pt not_active Application Discontinuation
- 1999-02-15 CA CA002262252A patent/CA2262252C/fr not_active Expired - Fee Related
- 1999-02-15 ID IDP990113D patent/ID23218A/id unknown
- 1999-02-15 IL IL12853199A patent/IL128531A0/xx unknown
- 1999-02-16 NO NO990722A patent/NO990722L/no unknown
- 1999-02-16 BG BG103180A patent/BG103180A/bg unknown
- 1999-02-16 AR ARP990100619A patent/AR017723A1/es unknown
- 1999-02-16 JP JP11037464A patent/JPH11292766A/ja active Pending
- 1999-02-16 TR TR1999/00328A patent/TR199900328A2/xx unknown
- 1999-02-16 ZA ZA9901220A patent/ZA991220B/xx unknown
- 1999-02-16 HU HU9900386A patent/HUP9900386A3/hu unknown
- 1999-02-16 TN TNTNSN99024A patent/TNSN99024A1/fr unknown
- 1999-02-16 EA EA199900124A patent/EA199900124A3/ru unknown
- 1999-02-16 MA MA25465A patent/MA26608A1/fr unknown
- 1999-02-16 OA OA9900034A patent/OA10976A/en unknown
- 1999-02-16 AU AU17329/99A patent/AU1732999A/en not_active Abandoned
- 1999-02-17 HR HR60/074,934A patent/HRP990054A2/hr not_active Application Discontinuation
- 1999-02-17 PL PL99331507A patent/PL331507A1/xx unknown

Also Published As

Publication number	Publication date
PL331507A1 (en)	1999-08-30
IL128531A0 (en)	2000-01-31
ID23218A (id)	2000-03-30
AR017723A1 (es)	2001-09-12
IS4975A (is)	1999-08-18
AU1732999A (en)	1999-09-02
PA8467401A1 (es)	2000-09-29
SG81261A1 (en)	2001-06-19
PE20000266A1 (es)	2000-04-07
TR199900328A2 (xx)	1999-10-21
BR9900653A (pt)	2000-10-17
CA2262252C (fr)	2006-01-10
TNSN99024A1 (fr)	2005-11-10
HRP990054A2 (en)	2000-02-29
JPH11292766A (ja)	1999-10-26
HUP9900386A2 (hu)	1999-11-29
AP9901464A0 (en)	1999-03-31
NO990722L (no)	1999-08-18
ZA991220B (en)	2000-08-16
NO990722D0 (no)	1999-02-16
CA2262252A1 (fr)	1999-08-17
HU9900386D0 (en)	1999-04-28
KR19990072616A (ko)	1999-09-27
EA199900124A2 (ru)	1999-08-26
EA199900124A3 (ru)	1999-12-29
US6043260A (en)	2000-03-28
EP0951906A1 (fr)	1999-10-27
MA26608A1 (fr)	2004-12-20
HUP9900386A3 (en)	1999-12-28
CN1231176A (zh)	1999-10-13
GT199900015A (es)	2000-07-26
OA10976A (en)	2001-11-05

Publication	Publication Date	Title
BG103180A (bg)	1999-09-30	Метод за лечение на сърдечна недостатъчност
DE60027729T2 (de)	2006-11-16	Benzophenone als reverse transcriptase inhibitore
KR900004693B1 (ko)	1990-07-02	4,5,6-치환-n-(치환페닐)-2-피리미딘아민, 그 제조방법 및 그 화합물이 들어있는 조성물
DE60021370T2 (de)	2006-04-27	Piperazinderivate verwendbar als ccr5 antagonisten
JP4323803B2 (ja)	2009-09-02	置換２−アニリノーベンゾイミダゾール及びｎｈｅ阻害剤としてのその使用
PL175788B1 (pl)	1999-02-26	Amidowe pochodne indolu i zawierające je kompozycje farmaceutyczne
US5693674A (en)	1997-12-02	Method of using triaryl-ethylene derivatives in the treatment and prevention of osteoporosis
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JP3962110B2 (ja)	2007-08-22	置換されたベンジルオキシカルボニルグアニジン、それらの製造法、医薬または診断剤としてのそれらの使用およびそれらを含有する医薬
EP1176144B1 (fr)	2003-07-09	Dérivés de N-triazolylméthyl-piperazine, en tant qu' antagonistes récepteurs de la neuroquinine
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CN117143039A (zh)	2023-12-01	一种苯并五元氮环类化合物、其制备方法及医药用途
JPH07502273A (ja)	1995-03-09	ベンゾピラン　クラス３抗不整脈薬
EP3921308B1 (fr)	2022-08-03	Composés inhibiteurs de l'échangeur sodium-hydrogène 3
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JPH11100382A (ja)	1999-04-13	スルホンアミド置換化合物、その製法、医薬または診断薬としての使用およびそれを含有する医薬
US20100222365A1 (en)	2010-09-02	Substituted triazole deriviatives as oxytocin antagonists
CN104788423A (zh)	2015-07-22	一种新的囊性纤维化跨膜传导调节因子抑制剂
EP0266563B1 (fr)	1992-01-29	Utilisation de 1-benzyl-amino-alkyl-pyrrolidinones comme antidépresseurs