BG105012A - N-свързани сулфонамиди на n-хетероциклични карбонови киселини или изостери на карбонови киселини - Google Patents

N-свързани сулфонамиди на n-хетероциклични карбонови киселини или изостери на карбонови киселини

Info

Publication number
BG105012A
BG105012A BG105012A BG10501200A BG105012A BG 105012 A BG105012 A BG 105012A BG 105012 A BG105012 A BG 105012A BG 10501200 A BG10501200 A BG 10501200A BG 105012 A BG105012 A BG 105012A
Authority
BG
Bulgaria
Prior art keywords
linked
carboxylic
isosteres
sulphonamides
heterocyclic
Prior art date
Application number
BG105012A
Other languages
English (en)
Inventor
Gregory Hamilton
Mark Norman
Yong-Qian Wu
Original Assignee
Gpi Nil Holdings, Inc
Amgen Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gpi Nil Holdings, Inc, Amgen Inc. filed Critical Gpi Nil Holdings, Inc
Publication of BG105012A publication Critical patent/BG105012A/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

Изобретението се отнася до N-свързани сулфонамидина N-хетероциклени карбоксилни киселини и изостери на карбоксилни киселини, до получаването и използването им за лечение на неврологични заболявания,включващи физически увредени нерви и невродегенеративни заболявания, за лечение на алопеция и за подпомагане растежа на косата.
BG105012A 1998-06-03 2000-12-01 N-свързани сулфонамиди на n-хетероциклични карбонови киселини или изостери на карбонови киселини BG105012A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8784298P 1998-06-03 1998-06-03
PCT/US1998/025572 WO1999062880A1 (en) 1998-06-03 1998-12-03 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres

Publications (1)

Publication Number Publication Date
BG105012A true BG105012A (bg) 2001-08-31

Family

ID=22207576

Family Applications (1)

Application Number Title Priority Date Filing Date
BG105012A BG105012A (bg) 1998-06-03 2000-12-01 N-свързани сулфонамиди на n-хетероциклични карбонови киселини или изостери на карбонови киселини

Country Status (17)

Country Link
US (3) US7459473B2 (bg)
EP (1) EP1084106A1 (bg)
JP (1) JP2002516904A (bg)
KR (1) KR20010052503A (bg)
CN (1) CN1295561A (bg)
AU (1) AU1708099A (bg)
BG (1) BG105012A (bg)
BR (1) BR9815882A (bg)
CA (1) CA2334002A1 (bg)
EA (1) EA200001247A1 (bg)
HU (1) HUP0102935A3 (bg)
IL (1) IL140040A0 (bg)
NO (1) NO20006078L (bg)
PL (1) PL348661A1 (bg)
SK (1) SK18302000A3 (bg)
WO (1) WO1999062880A1 (bg)
ZA (1) ZA9811060B (bg)

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SE0202539D0 (sv) 2002-08-27 2002-08-27 Astrazeneca Ab Compounds
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JP6541118B1 (ja) * 2018-04-27 2019-07-10 株式会社成和化成 化粧品基材および該化粧品基材を含有する毛髪用化粧品、美白剤
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CA2334002A1 (en) 1999-12-09
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SK18302000A3 (sk) 2001-06-11
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CN1295561A (zh) 2001-05-16
US7459473B2 (en) 2008-12-02
US20020052514A1 (en) 2002-05-02
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US7078424B2 (en) 2006-07-18
US20040082622A1 (en) 2004-04-29
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KR20010052503A (ko) 2001-06-25
BR9815882A (pt) 2002-09-17

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