BG107538A - Дозирана лекарствена форма с хидрогелен механизъм - Google Patents

Дозирана лекарствена форма с хидрогелен механизъм Download PDF

Info

Publication number: BG107538A
Authority: BG; Bulgaria
Prior art keywords: drug; weight; water; dosage form; composition
Prior art date: 2000-08-09

Application number

BG107538A

Other languages

Bulgarian (bg)

English (en)

Inventor

Leah APPEL

Walter Babcock

Ronald BEYERINCK

Mark CHIDLAW

William Curatolo

Dwayne Friesen

Scott HERBIG

Avinash THOMBRE

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-08-09

Filing date

2003-02-06

Publication date

2003-11-28

2003-02-06 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

2003-11-28 Publication of BG107538A publication Critical patent/BG107538A/bg

Links

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238000007920 subcutaneous administration Methods 0.000 description 1
125000001424 substituent group Chemical group 0.000 description 1
KDYFGRWQOYBRFD-UHFFFAOYSA-L succinate(2-) Chemical compound [O-]C(=O)CCC([O-])=O KDYFGRWQOYBRFD-UHFFFAOYSA-L 0.000 description 1
150000003444 succinic acids Chemical class 0.000 description 1
229940035023 sucrose monostearate Drugs 0.000 description 1
150000003460 sulfonic acids Chemical class 0.000 description 1
229960004940 sulpiride Drugs 0.000 description 1
239000000829 suppository Substances 0.000 description 1
230000002522 swelling effect Effects 0.000 description 1
239000000454 talc Substances 0.000 description 1
229910052623 talc Inorganic materials 0.000 description 1
229960000580 terconazole Drugs 0.000 description 1
IWVCMVBTMGNXQD-UHFFFAOYSA-N terramycin dehydrate Natural products C1=CC=C2C(O)(C)C3C(O)C4C(N(C)C)C(O)=C(C(N)=O)C(=O)C4(O)C(O)=C3C(=O)C2=C1O IWVCMVBTMGNXQD-UHFFFAOYSA-N 0.000 description 1
RBTVSNLYYIMMKS-UHFFFAOYSA-N tert-butyl 3-aminoazetidine-1-carboxylate;hydrochloride Chemical compound Cl.CC(C)(C)OC(=O)N1CC(N)C1 RBTVSNLYYIMMKS-UHFFFAOYSA-N 0.000 description 1
239000012085 test solution Substances 0.000 description 1
229960003604 testosterone Drugs 0.000 description 1
229940072172 tetracycline antibiotic Drugs 0.000 description 1
YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
235000010296 thiabendazole Nutrition 0.000 description 1
239000004308 thiabendazole Substances 0.000 description 1
229960004546 thiabendazole Drugs 0.000 description 1
WJCNZQLZVWNLKY-UHFFFAOYSA-N thiabendazole Chemical compound S1C=NC(C=2NC3=CC=CC=C3N=2)=C1 WJCNZQLZVWNLKY-UHFFFAOYSA-N 0.000 description 1
229960000882 thiothixene hydrochloride Drugs 0.000 description 1
229960004605 timolol Drugs 0.000 description 1
230000007704 transition Effects 0.000 description 1
150000003626 triacylglycerols Chemical class 0.000 description 1
JOFWLTCLBGQGBO-UHFFFAOYSA-N triazolam Chemical compound C12=CC(Cl)=CC=C2N2C(C)=NN=C2CN=C1C1=CC=CC=C1Cl JOFWLTCLBGQGBO-UHFFFAOYSA-N 0.000 description 1
229960003386 triazolam Drugs 0.000 description 1
229960002906 trimazosin Drugs 0.000 description 1
YNZXWQJZEDLQEG-UHFFFAOYSA-N trimazosin Chemical compound N1=C2C(OC)=C(OC)C(OC)=CC2=C(N)N=C1N1CCN(C(=O)OCC(C)(C)O)CC1 YNZXWQJZEDLQEG-UHFFFAOYSA-N 0.000 description 1
229960005041 troleandomycin Drugs 0.000 description 1
LQCLVBQBTUVCEQ-QTFUVMRISA-N troleandomycin Chemical compound O1[C@@H](C)[C@H](OC(C)=O)[C@@H](OC)C[C@@H]1O[C@@H]1[C@@H](C)C(=O)O[C@H](C)[C@H](C)[C@H](OC(C)=O)[C@@H](C)C(=O)[C@@]2(OC2)C[C@H](C)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)OC(C)=O)[C@H]1C LQCLVBQBTUVCEQ-QTFUVMRISA-N 0.000 description 1
210000002438 upper gastrointestinal tract Anatomy 0.000 description 1
239000006200 vaporizer Substances 0.000 description 1
229940124549 vasodilator Drugs 0.000 description 1
239000003071 vasodilator agent Substances 0.000 description 1
PNVNVHUZROJLTJ-UHFFFAOYSA-N venlafaxine Chemical compound C1=CC(OC)=CC=C1C(CN(C)C)C1(O)CCCCC1 PNVNVHUZROJLTJ-UHFFFAOYSA-N 0.000 description 1
229960004688 venlafaxine Drugs 0.000 description 1
229920006163 vinyl copolymer Polymers 0.000 description 1
229920002554 vinyl polymer Polymers 0.000 description 1
229940100050 virazole Drugs 0.000 description 1
235000013343 vitamin Nutrition 0.000 description 1
229930003231 vitamin Natural products 0.000 description 1
239000011782 vitamin Substances 0.000 description 1
229940088594 vitamin Drugs 0.000 description 1
BCEHBSKCWLPMDN-MGPLVRAMSA-N voriconazole Chemical compound C1([C@H](C)[C@](O)(CN2N=CN=C2)C=2C(=CC(F)=CC=2)F)=NC=NC=C1F BCEHBSKCWLPMDN-MGPLVRAMSA-N 0.000 description 1
229960004740 voriconazole Drugs 0.000 description 1
239000003643 water by type Substances 0.000 description 1
230000004584 weight gain Effects 0.000 description 1
235000019786 weight gain Nutrition 0.000 description 1
238000005550 wet granulation Methods 0.000 description 1
XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical compound [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
229960000607 ziprasidone Drugs 0.000 description 1
MVWVFYHBGMAFLY-UHFFFAOYSA-N ziprasidone Chemical compound C1=CC=C2C(N3CCN(CC3)CCC3=CC=4CC(=O)NC=4C=C3Cl)=NSC2=C1 MVWVFYHBGMAFLY-UHFFFAOYSA-N 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer

Landscapes

Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

BG107538A 2000-08-09 2003-02-06 Дозирана лекарствена форма с хидрогелен механизъм BG107538A (bg)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US22419900P	2000-08-09	2000-08-09
PCT/IB2001/001390 WO2002011702A2 (fr)	2000-08-09	2001-08-03	Forme posologique de medicament entraine par un hydrogel

Publications (1)

Publication Number	Publication Date
BG107538A true BG107538A (bg)	2003-11-28

Family

ID=22839665

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG107538A BG107538A (bg)	2000-08-09	2003-02-06	Дозирана лекарствена форма с хидрогелен механизъм

Country Status (30)

Country	Link
US (2)	US20030086972A1 (fr)
EP (1)	EP1326587A2 (fr)
JP (1)	JP2004505907A (fr)
KR (1)	KR20030024844A (fr)
CN (1)	CN1461212A (fr)
AP (1)	AP2001002237A0 (fr)
AU (1)	AU2002229141A1 (fr)
BG (1)	BG107538A (fr)
BR (1)	BR0113067A (fr)
CA (1)	CA2418907A1 (fr)
DO (1)	DOP2001000229A (fr)
EA (1)	EA200300081A1 (fr)
EC (1)	ECSP034455A (fr)
EE (1)	EE200300055A (fr)
GT (1)	GT200100161A (fr)
HR (1)	HRP20030082A2 (fr)
HU (1)	HUP0300722A2 (fr)
IL (1)	IL154012A0 (fr)
IS (1)	IS6686A (fr)
MA (1)	MA26939A1 (fr)
MX (1)	MXPA03001209A (fr)
NO (1)	NO20030627L (fr)
OA (1)	OA12365A (fr)
PA (1)	PA8524901A1 (fr)
PE (1)	PE20020307A1 (fr)
PL (1)	PL360658A1 (fr)
SV (1)	SV2002000586A (fr)
TN (1)	TNSN01123A1 (fr)
UY (1)	UY26876A1 (fr)
WO (1)	WO2002011702A2 (fr)

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2001
- 2001-08-01 US US09/920,056 patent/US20030086972A1/en not_active Abandoned
- 2001-08-03 OA OA1200300043A patent/OA12365A/en unknown
- 2001-08-03 WO PCT/IB2001/001390 patent/WO2002011702A2/fr not_active Ceased
- 2001-08-03 CA CA002418907A patent/CA2418907A1/fr not_active Abandoned
- 2001-08-03 HU HU0300722A patent/HUP0300722A2/hu unknown
- 2001-08-03 BR BR0113067-6A patent/BR0113067A/pt not_active IP Right Cessation
- 2001-08-03 CN CN01816024A patent/CN1461212A/zh active Pending
- 2001-08-03 MX MXPA03001209A patent/MXPA03001209A/es not_active Application Discontinuation
- 2001-08-03 AU AU2002229141A patent/AU2002229141A1/en not_active Abandoned
- 2001-08-03 AP APAP/P/2001/002237A patent/AP2001002237A0/en unknown
- 2001-08-03 EE EEP200300055A patent/EE200300055A/xx unknown
- 2001-08-03 HR HR20030082A patent/HRP20030082A2/hr not_active Application Discontinuation
- 2001-08-03 EA EA200300081A patent/EA200300081A1/ru unknown
- 2001-08-03 PL PL36065801A patent/PL360658A1/xx not_active Application Discontinuation
- 2001-08-03 EP EP01984471A patent/EP1326587A2/fr not_active Withdrawn
- 2001-08-03 US US10/344,171 patent/US20040052845A1/en not_active Abandoned
- 2001-08-03 IL IL15401201A patent/IL154012A0/xx unknown
- 2001-08-03 KR KR10-2003-7001861A patent/KR20030024844A/ko not_active Ceased
- 2001-08-03 JP JP2002517039A patent/JP2004505907A/ja active Pending
- 2001-08-08 PE PE2001000791A patent/PE20020307A1/es not_active Application Discontinuation
- 2001-08-08 TN TNTNSN01123A patent/TNSN01123A1/fr unknown
- 2001-08-08 GT GT200100161A patent/GT200100161A/es unknown
- 2001-08-08 UY UY26876A patent/UY26876A1/es not_active Application Discontinuation
- 2001-08-08 DO DO2001000229A patent/DOP2001000229A/es unknown
- 2001-08-08 SV SV2001000586A patent/SV2002000586A/es not_active Application Discontinuation
- 2001-08-09 PA PA20018524901A patent/PA8524901A1/es unknown
2003
- 2003-01-16 IS IS6686A patent/IS6686A/is unknown
- 2003-01-28 EC EC2003004455A patent/ECSP034455A/es unknown
- 2003-01-29 MA MA27017A patent/MA26939A1/fr unknown
- 2003-02-06 BG BG107538A patent/BG107538A/bg unknown
- 2003-02-07 NO NO20030627A patent/NO20030627L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
MA26939A1 (fr)	2004-12-20
CA2418907A1 (fr)	2002-02-14
PL360658A1 (en)	2004-09-20
TNSN01123A1 (fr)	2005-11-10
PE20020307A1 (es)	2002-04-23
US20040052845A1 (en)	2004-03-18
ECSP034455A (es)	2003-03-10
CN1461212A (zh)	2003-12-10
AP2001002237A0 (en)	2001-09-30
EE200300055A (et)	2004-12-15
GT200100161A (es)	2002-03-22
WO2002011702A2 (fr)	2002-02-14
NO20030627L (no)	2003-04-08
DOP2001000229A (es)	2002-09-30
JP2004505907A (ja)	2004-02-26
OA12365A (en)	2006-05-16
EA200300081A1 (ru)	2003-08-28
AU2002229141A1 (en)	2002-02-18
IL154012A0 (en)	2003-07-31
WO2002011702A3 (fr)	2002-11-28
MXPA03001209A (es)	2003-06-30
HRP20030082A2 (en)	2003-04-30
SV2002000586A (es)	2002-10-24
UY26876A1 (es)	2002-03-22
HUP0300722A2 (hu)	2003-11-28
US20030086972A1 (en)	2003-05-08
NO20030627D0 (no)	2003-02-07
KR20030024844A (ko)	2003-03-26
EP1326587A2 (fr)	2003-07-16
IS6686A (is)	2003-01-16
PA8524901A1 (es)	2002-04-25
BR0113067A (pt)	2003-07-01

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TWI257302B (en)	2006-07-01	Controlled-release of an active substance into a high fat environment
US20040052844A1 (en)	2004-03-18	Time-controlled, sustained release, pharmaceutical composition containing water-soluble resins
CN100563637C (zh)	2009-12-02	一种控释给药的药芯组合物和控释制剂及其制备方法
WO2007057762A2 (fr)	2007-05-24	Forme posologique a liberation controlee