BR0012864A - Forma aperfeiçoada de forma i do hidrocloreto de celiprolol - Google Patents
Forma aperfeiçoada de forma i do hidrocloreto de celiprololInfo
- Publication number
- BR0012864A BR0012864A BR0012864-3A BR0012864A BR0012864A BR 0012864 A BR0012864 A BR 0012864A BR 0012864 A BR0012864 A BR 0012864A BR 0012864 A BR0012864 A BR 0012864A
- Authority
- BR
- Brazil
- Prior art keywords
- celiprolol hydrochloride
- optimized
- hydrochloride
- celiprolol
- propoxy
- Prior art date
Links
- VKJHTUVLJYWAEY-UHFFFAOYSA-N Celiprolol hydrochloride Chemical compound Cl.CCN(CC)C(=O)NC1=CC=C(OCC(O)CNC(C)(C)C)C(C(C)=O)=C1 VKJHTUVLJYWAEY-UHFFFAOYSA-N 0.000 title abstract 3
- 229960000384 celiprolol hydrochloride Drugs 0.000 title abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
- C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1035DE1999 | 1999-07-30 | ||
| PCT/IB2000/001023 WO2001008633A2 (en) | 1999-07-30 | 2000-07-24 | An improved form of form i celiprolol hydrochloride |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0012864A true BR0012864A (pt) | 2002-06-04 |
Family
ID=11092063
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0012864-3A BR0012864A (pt) | 1999-07-30 | 2000-07-24 | Forma aperfeiçoada de forma i do hidrocloreto de celiprolol |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1204408A2 (de) |
| JP (1) | JP2003505485A (de) |
| AU (1) | AU5839000A (de) |
| BR (1) | BR0012864A (de) |
| PL (1) | PL353243A1 (de) |
| WO (1) | WO2001008633A2 (de) |
| ZA (1) | ZA200200693B (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030135041A1 (en) | 2002-01-04 | 2003-07-17 | Orchid Chemicals & Pharmaceuticals Limited, India | Synthesis of ceftiofur intermediate |
| JP4547245B2 (ja) * | 2004-12-16 | 2010-09-22 | 株式会社パーマケム・アジア | ペリンドプリルエルブミンのｉ型結晶、及びその製造方法 |
| WO2007029155A2 (en) * | 2005-09-05 | 2007-03-15 | Ranbaxy Laboratories Limited | An improved process for preparation of pure celiprolol base |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3544172A1 (de) * | 1985-12-13 | 1987-06-19 | Lentia Gmbh | Neue kristalline salze von aryloxy-propanolaminen, verfahren zu ihrer herstellung und ihre verwendung |
| US5980882A (en) * | 1997-04-16 | 1999-11-09 | Medeva Pharmaceuticals Manufacturing | Drug-resin complexes stabilized by chelating agents |
-
2000
- 2000-07-24 EP EP00944158A patent/EP1204408A2/de not_active Withdrawn
- 2000-07-24 BR BR0012864-3A patent/BR0012864A/pt not_active Application Discontinuation
- 2000-07-24 AU AU58390/00A patent/AU5839000A/en not_active Abandoned
- 2000-07-24 PL PL00353243A patent/PL353243A1/xx not_active Application Discontinuation
- 2000-07-24 WO PCT/IB2000/001023 patent/WO2001008633A2/en not_active Ceased
- 2000-07-24 JP JP2001513366A patent/JP2003505485A/ja active Pending
-
2002
- 2002-01-25 ZA ZA200200693A patent/ZA200200693B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1204408A2 (de) | 2002-05-15 |
| WO2001008633A3 (en) | 2001-08-23 |
| AU5839000A (en) | 2001-02-19 |
| ZA200200693B (en) | 2002-10-30 |
| WO2001008633A2 (en) | 2001-02-08 |
| PL353243A1 (en) | 2003-11-03 |
| JP2003505485A (ja) | 2003-02-12 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR9903984B1 (pt) | processo para a produção de uma composição aquosa que contém um peptìdeo farmaceuticamente efetivo. | |
| WO2002004404A3 (en) | 7,8 and 9-substituted tetracycline compounds | |
| BR0016882A (pt) | ésteres derivados de (rr,ss)-3-(2-dimetilaminometil-1-hidroxicicloexil)fenil 2-hidroxibenzoato | |
| BR9401959A (pt) | Processo para a fabricação de uma mousse de carboneto de silício,processo para a fabricação de um catalisador, carboneto de silício bem como sua aplicação | |
| BR9812837A (pt) | Processo para fazer um composto, e, composto | |
| BR9503619A (pt) | Processo para a síntese de trans-1,4-polibutadieno | |
| CA2262566A1 (en) | Benzamidine derivatives and the use thereof as medicaments with ltb4-antagonistic effect | |
| BRPI9814894A (pt) | processo para a preparação de ácidos 8-metóxi-quinolonocarboxílicos. | |
| BR0002073A (pt) | Processo para a preparação de um composto quiral | |
| BR0212772A (pt) | Processo para a preparação de repaglinida | |
| BR9809650A (pt) | Composição oral para remineralização dos dentes, e, processo para remineralizar porções desmineralizadas das estruturas de dentes | |
| CA2256514A1 (en) | Veterinary use of a pleuromutilin derivative | |
| BR9814495A (pt) | Composto, processo para prepará-lo, uso do mesmo, composição farmacêutica, e, processo | |
| BR9807988B1 (pt) | processo para a preparaÇço de um composto, e, composto. | |
| BR9808642A (pt) | Processo para preparar eprosartan | |
| ATE554071T1 (de) | Herstellung chinolin-substituierter carbonat- und carbamat-derivate | |
| AU4300497A (en) | Process for the manufacture of aliphatic alpha, omega amino nitriles | |
| BR9808664A (pt) | Processo para preparar eprosartan | |
| ES2185196T3 (es) | Un procedimiento para la preparacion de tetraazamacrociclos. | |
| BR0205804A (pt) | Suporte radial para um eixo de acionamento | |
| BR9807785A (pt) | Processo para a preparação do composto, e, composto | |
| HUT77239A (hu) | Oldószer nélküli eljárás 2,6-difluor-benzonitril előállítására | |
| BR9712773A (pt) | Processo para a sìntese de benzotiofenos | |
| BR9703299A (pt) | Processo para a preparação de um composto de 3-amino-4,4,4-tri-halocrotonato | |
| ES2173586T3 (es) | Derivados de ciclohexandiol. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA10 | Dismissal: dismissal - article 33 of industrial property law | ||
| B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |