BR0014145A - Compostos de benzimidazol substituìdo por alcóxi, preparações farmacêuticas contendo o mesmo, e métodos de uso do mesmo - Google Patents

Compostos de benzimidazol substituìdo por alcóxi, preparações farmacêuticas contendo o mesmo, e métodos de uso do mesmo

Info

Publication number
BR0014145A
BR0014145A BR0014145-3A BR0014145A BR0014145A BR 0014145 A BR0014145 A BR 0014145A BR 0014145 A BR0014145 A BR 0014145A BR 0014145 A BR0014145 A BR 0014145A
Authority
BR
Brazil
Prior art keywords
same
alkoxy
methods
pharmaceutical preparations
preparations containing
Prior art date
Application number
BR0014145-3A
Other languages
English (en)
Inventor
Robert R Whittle
Frederick D Sancilio
Grayson Walker Stowell
Douglas John Jenkins
Linda Whittall
Glen Alan Meyer
Steven A Fontana
Original Assignee
Aaipharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/519,976 external-priority patent/US6262085B1/en
Application filed by Aaipharma Inc filed Critical Aaipharma Inc
Publication of BR0014145A publication Critical patent/BR0014145A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: "COMPOSTOS DE BENZIMIDAZOL SUBSTITUìDO POR ALCóXI, PREPARAçõES FARMACêUTICAS CONTENDO O MESMO, E MéTODOS DE USO DO MESMO". Compostos representados pela fórmula (Ia) são descritos pela invenção, junto das composições e complexos destes, opcionalmente em combinação com compostos da fórmula (Ib). As formulações farmacêuticas e métodos de preparação e empregando tais compostos são também descritos.
BR0014145-3A 1999-08-26 2000-08-25 Compostos de benzimidazol substituìdo por alcóxi, preparações farmacêuticas contendo o mesmo, e métodos de uso do mesmo BR0014145A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15087899P 1999-08-26 1999-08-26
US09/519,976 US6262085B1 (en) 1999-08-26 2000-03-07 Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same
PCT/US2000/023363 WO2001014367A1 (en) 1999-08-26 2000-08-25 Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same

Publications (1)

Publication Number Publication Date
BR0014145A true BR0014145A (pt) 2002-05-14

Family

ID=26848119

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0014145-3A BR0014145A (pt) 1999-08-26 2000-08-25 Compostos de benzimidazol substituìdo por alcóxi, preparações farmacêuticas contendo o mesmo, e métodos de uso do mesmo

Country Status (16)

Country Link
EP (1) EP1206466B1 (pt)
JP (1) JP4312405B2 (pt)
KR (1) KR100712039B1 (pt)
CN (2) CN1636564A (pt)
AT (1) ATE306483T1 (pt)
AU (2) AU777667B2 (pt)
BR (1) BR0014145A (pt)
CA (1) CA2382867A1 (pt)
DE (1) DE60023154T2 (pt)
HR (1) HRP20020174A2 (pt)
MX (1) MXPA02002007A (pt)
NO (1) NO326849B1 (pt)
RO (1) RO122491B1 (pt)
RU (1) RU2263673C2 (pt)
SI (1) SI20974A (pt)
SK (1) SK286903B6 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2376231A (en) * 2001-06-06 2002-12-11 Cipla Ltd Benzimidazole-cyclodextrin inclusion complex
BRPI0512522A (pt) 2004-06-24 2008-03-11 Astrazeneca Ab processo para a preparação de sal de sódio de esomeprazol, composto, formulação farmacêutica, e, método de tratamento
ES2246149B1 (es) * 2004-07-02 2007-06-01 Esteve Quimica, S.A. Formas solidas de la sal magnesica de s-omeprazol y procedimientos para su preparacion.
CN103524491A (zh) * 2013-10-16 2014-01-22 江南大学 埃索美拉唑镁盐四水合物的三种晶型及其制备方法
CA3168170A1 (en) * 2020-03-09 2021-09-16 Pamela Ann Cacavas Method for removing interfering components of a liquid sample prior to dispensing same on a chemical reagent test slide
CN114558004B (zh) * 2022-03-29 2023-08-11 奎马特里克斯有限公司 Qtx125药物制剂
CN116082247B (zh) * 2023-01-19 2025-08-01 浙江工业大学 一种苯并咪唑类衍生物及其应用
CN118225938B (zh) * 2024-04-02 2024-08-30 江苏海洋大学 一种中药复方五神汤的质量检测方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US895292A (en) * 1904-07-22 1908-08-04 Marvin A Neeland Blowing-engine inlet-valve.
SE418966B (sv) * 1974-02-18 1981-07-06 Haessle Ab Analogiforfarande for framstellning av foreningar med magsyrasekretionsinhiberande verkan
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
SE8300736D0 (sv) * 1983-02-11 1983-02-11 Haessle Ab Novel pharmacologically active compounds
SE9301830D0 (sv) * 1993-05-28 1993-05-28 Ab Astra New compounds

Also Published As

Publication number Publication date
AU2005200203B2 (en) 2008-01-10
CN1636564A (zh) 2005-07-13
ATE306483T1 (de) 2005-10-15
SK286903B6 (sk) 2009-07-06
JP2003507475A (ja) 2003-02-25
NO326849B1 (no) 2009-03-02
MXPA02002007A (es) 2003-08-20
SK2812002A3 (en) 2002-07-02
SI20974A (sl) 2003-02-28
KR20020035861A (ko) 2002-05-15
RO122491B1 (ro) 2009-07-30
CA2382867A1 (en) 2001-03-01
DE60023154T2 (de) 2006-06-22
CN1183127C (zh) 2005-01-05
DE60023154D1 (de) 2006-02-23
KR100712039B1 (ko) 2007-04-27
RU2263673C2 (ru) 2005-11-10
AU7073700A (en) 2001-03-19
JP4312405B2 (ja) 2009-08-12
AU777667B2 (en) 2004-10-28
CN1384831A (zh) 2002-12-11
EP1206466A1 (en) 2002-05-22
EP1206466B1 (en) 2005-10-12
NO20020914D0 (no) 2002-02-25
HRP20020174A2 (en) 2005-12-31
AU2005200203A1 (en) 2005-02-10
NO20020914L (no) 2002-04-26

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 10(VIII), 11, 13, 24 E 25 DA LPI

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.