BR0110643A - Benzoxazinas para uso no tratamento do mal de parkinson - Google Patents
Benzoxazinas para uso no tratamento do mal de parkinsonInfo
- Publication number
- BR0110643A BR0110643A BR0110643-0A BR0110643A BR0110643A BR 0110643 A BR0110643 A BR 0110643A BR 0110643 A BR0110643 A BR 0110643A BR 0110643 A BR0110643 A BR 0110643A
- Authority
- BR
- Brazil
- Prior art keywords
- parkinson
- disease
- alkyl
- benzoxazine
- hydrogen
- Prior art date
Links
- 208000018737 Parkinson disease Diseases 0.000 title abstract 2
- CMLFRMDBDNHMRA-UHFFFAOYSA-N 2h-1,2-benzoxazine Chemical compound C1=CC=C2C=CNOC2=C1 CMLFRMDBDNHMRA-UHFFFAOYSA-N 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 208000016285 Movement disease Diseases 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 150000005130 benzoxazines Chemical class 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000004356 hydroxy functional group Chemical group O* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
"BENZOXAZINAS PARA USO NO TRATAMENTO DO MAL DE PARKINSON". Benzoxazinas de fórmula (I) onde R^ 1^ é C~ 1~ - C~ 6~ alquila, C~ 2~-C~ 6~ alquenila ou (CH~ 2~)~ n~ fenila, R^ 2^ é C~ 3~ - C~ 6~ alquila, R^ 3^ é hidrogênio, halo, hidróxi, alcóxi ou alquiltio, R^ 4^ é hidrogênio ou alquila, ou um sal farmaceuticamente aceitável das mesmas, são úteis para tratar distúrbios do movimento tal como o mal de Parkinson.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20278700P | 2000-05-09 | 2000-05-09 | |
| PCT/US2001/012528 WO2001085734A1 (en) | 2000-05-09 | 2001-04-17 | Benzoxazines for use in the treatment of parkinson's disease |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0110643A true BR0110643A (pt) | 2003-03-18 |
Family
ID=22751255
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0110643-0A BR0110643A (pt) | 2000-05-09 | 2001-04-17 | Benzoxazinas para uso no tratamento do mal de parkinson |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6812228B2 (pt) |
| EP (1) | EP1282625B1 (pt) |
| JP (1) | JP2003532733A (pt) |
| AT (1) | ATE270295T1 (pt) |
| AU (1) | AU2001251662A1 (pt) |
| BR (1) | BR0110643A (pt) |
| CA (1) | CA2407789A1 (pt) |
| DE (1) | DE60104110T2 (pt) |
| DK (1) | DK1282625T3 (pt) |
| ES (1) | ES2223824T3 (pt) |
| MX (1) | MXPA02010270A (pt) |
| PT (1) | PT1282625E (pt) |
| WO (1) | WO2001085734A1 (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6087916B2 (ja) | 2011-07-05 | 2017-03-01 | エレクトロ サイエンティフィック インダストリーズ インコーポレーテッド | 使用中の音響光学ビーム偏向器および音響光学変調器の温度安定性を実現するためのシステムならびに方法 |
| US9463186B2 (en) | 2013-04-15 | 2016-10-11 | Northwestern University | Treatment for dopaminergic disorders |
| MX2021011588A (es) * | 2019-03-25 | 2021-12-15 | Cold Spring Harbor Laboratory | Antagonistas del receptor muscarinico de acetilcolina subtipo 4 en el tratamiento de la anemia. |
-
2001
- 2001-04-17 AU AU2001251662A patent/AU2001251662A1/en not_active Abandoned
- 2001-04-17 ES ES01925065T patent/ES2223824T3/es not_active Expired - Lifetime
- 2001-04-17 US US10/275,825 patent/US6812228B2/en not_active Expired - Fee Related
- 2001-04-17 CA CA002407789A patent/CA2407789A1/en not_active Abandoned
- 2001-04-17 MX MXPA02010270A patent/MXPA02010270A/es not_active Application Discontinuation
- 2001-04-17 JP JP2001582334A patent/JP2003532733A/ja active Pending
- 2001-04-17 AT AT01925065T patent/ATE270295T1/de not_active IP Right Cessation
- 2001-04-17 EP EP01925065A patent/EP1282625B1/en not_active Expired - Lifetime
- 2001-04-17 WO PCT/US2001/012528 patent/WO2001085734A1/en not_active Ceased
- 2001-04-17 PT PT01925065T patent/PT1282625E/pt unknown
- 2001-04-17 DE DE60104110T patent/DE60104110T2/de not_active Expired - Fee Related
- 2001-04-17 BR BR0110643-0A patent/BR0110643A/pt not_active IP Right Cessation
- 2001-04-17 DK DK01925065T patent/DK1282625T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| DE60104110T2 (de) | 2005-08-25 |
| US6812228B2 (en) | 2004-11-02 |
| US20030220335A1 (en) | 2003-11-27 |
| ES2223824T3 (es) | 2005-03-01 |
| WO2001085734A1 (en) | 2001-11-15 |
| MXPA02010270A (es) | 2003-04-25 |
| CA2407789A1 (en) | 2001-11-15 |
| JP2003532733A (ja) | 2003-11-05 |
| ATE270295T1 (de) | 2004-07-15 |
| DE60104110D1 (de) | 2004-08-05 |
| EP1282625B1 (en) | 2004-06-30 |
| PT1282625E (pt) | 2004-10-29 |
| EP1282625A1 (en) | 2003-02-12 |
| AU2001251662A1 (en) | 2001-11-20 |
| DK1282625T3 (da) | 2004-11-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A E 8A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO DA RPI 2016 DE 25/08/2009. |