BR112012000657A2 - novos azabicilohexanos - Google Patents
novos azabicilohexanosInfo
- Publication number
- BR112012000657A2 BR112012000657A2 BR112012000657A BR112012000657A BR112012000657A2 BR 112012000657 A2 BR112012000657 A2 BR 112012000657A2 BR 112012000657 A BR112012000657 A BR 112012000657A BR 112012000657 A BR112012000657 A BR 112012000657A BR 112012000657 A2 BR112012000657 A2 BR 112012000657A2
- Authority
- BR
- Brazil
- Prior art keywords
- azabicylhexanes
- new
- new azabicylhexanes
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Indole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1320DE2009 | 2009-06-26 | ||
| IN555DE2010 | 2010-03-10 | ||
| IN1297DE2010 | 2010-06-03 | ||
| PCT/IN2010/000428 WO2010150281A2 (en) | 2009-06-26 | 2010-06-22 | Novel azabicyclohexanes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012000657A2 true BR112012000657A2 (pt) | 2016-11-16 |
Family
ID=42790536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012000657A BR112012000657A2 (pt) | 2009-06-26 | 2010-06-22 | novos azabicilohexanos |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8906913B2 (pt) |
| EP (1) | EP2445887B1 (pt) |
| JP (1) | JP5696142B2 (pt) |
| KR (1) | KR20120106697A (pt) |
| CN (1) | CN102803224A (pt) |
| AR (1) | AR077251A1 (pt) |
| AU (1) | AU2010264027B9 (pt) |
| BR (1) | BR112012000657A2 (pt) |
| CA (1) | CA2765692A1 (pt) |
| MX (1) | MX2012000231A (pt) |
| RU (1) | RU2012102094A (pt) |
| WO (1) | WO2010150281A2 (pt) |
| ZA (1) | ZA201109437B (pt) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112013007566A2 (pt) | 2010-09-28 | 2016-08-02 | Panacea Biotec Ltd | novos compostos bicíclicos |
| US9724351B2 (en) | 2012-08-23 | 2017-08-08 | Alios Biopharma, Inc. | Compounds for the treatment of paramoxyvirus viral infections |
| PH12021550330A1 (en) * | 2013-08-21 | 2022-09-28 | Janssen Biopharma Inc | Antiviral compounds |
| CN104447501B (zh) * | 2014-11-02 | 2017-01-18 | 浙江医药高等专科学校 | 烷基取代的环己烷羧酸酰胺类衍生物及其用途 |
| CN104356047B (zh) * | 2014-11-02 | 2017-04-05 | 浙江医药高等专科学校 | 取代的环己烷羧酸酰胺类衍生物及其药物用途 |
| CN104447500B (zh) * | 2014-11-02 | 2017-01-18 | 浙江医药高等专科学校 | 卤素取代的环己烷羧酸酰胺类衍生物及其用途 |
| MA41614A (fr) | 2015-02-25 | 2018-01-02 | Alios Biopharma Inc | Composés antiviraux |
| WO2019021059A1 (en) | 2017-07-28 | 2019-01-31 | Novartis Ag | INDOLE DERIVATIVES AND USES THEREOF |
| CA3187566A1 (en) | 2020-06-22 | 2021-12-30 | Corcept Therapeutics Incorporated | Quaternary indazole glucocorticoid receptor antagonists |
| CN114079982B (zh) * | 2020-08-11 | 2023-07-25 | 维沃移动通信有限公司 | 网络转移方法、装置和设备 |
| EP4196118A1 (en) | 2020-08-13 | 2023-06-21 | Boehringer Ingelheim International GmbH | Treatment of cognitive impairement associated with schizophrenia |
| CN117567449A (zh) | 2020-10-13 | 2024-02-20 | 勃林格殷格翰国际有限公司 | 再加工方法 |
| US12115154B2 (en) | 2020-12-16 | 2024-10-15 | Srx Cardio, Llc | Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) |
| EP4357335A4 (en) * | 2021-06-15 | 2025-11-26 | Otsuka Pharma Co Ltd | AZABICYCLO[3.1.0]HEXANE COMPOUND |
| US12098144B2 (en) | 2021-12-21 | 2024-09-24 | Corcept Therapeutics Incorporated | Piperazine indazole glucocorticoid receptor antagonists |
| CA3243547A1 (en) | 2021-12-21 | 2023-06-29 | Corcept Therapeutics Incorporated | INDAZOLE GLUCOCORTICOID RECEPTOR BICYCLIC ANTAGONISTS |
| CN117209474B (zh) * | 2022-06-10 | 2026-03-10 | 康百达（四川）生物医药科技有限公司 | 吡咯烷衍生物、药物组合物及其在医药上的应用 |
| TW202348602A (zh) * | 2022-06-10 | 2023-12-16 | 大陸商成都百裕製藥股份有限公司 | 吡咯烷衍生物、藥物组合物及其製藥用途 |
| EP4624455A1 (en) * | 2022-11-23 | 2025-10-01 | Kangbaida (Sichuan) Biotechnology Co., Ltd. | Preparation method for chiral pyrrole derivative and intermediate thereof |
Family Cites Families (71)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4131611A (en) | 1975-07-31 | 1978-12-26 | American Cyanamid Company | Azabicyclohexanes |
| US4435419A (en) | 1981-07-01 | 1984-03-06 | American Cyanamid Company | Method of treating depression using azabicyclohexanes |
| AU667198B2 (en) | 1991-11-01 | 1996-03-14 | Pharmacia & Upjohn Company | Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents |
| US5646244A (en) | 1993-09-06 | 1997-07-08 | Fujisawa Pharmaceutical Co., Ltd. | Cyclodepsipeptide compound |
| AU702752B2 (en) | 1995-05-11 | 1999-03-04 | Pharmacia & Upjohn Company | Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
| AU1379900A (en) | 1998-11-17 | 2000-06-05 | Bayer Aktiengesellschaft | Novel substituted phenyloxazolidone derivatives |
| JP2003501351A (ja) | 1999-05-27 | 2003-01-14 | ファルマシア・アンド・アップジョン・カンパニー | 抗菌剤としての二環系オキサゾリジノン |
| US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| BR0111280A (pt) | 2000-06-05 | 2003-06-10 | Dong A Pharm Co Ltd | Novos derivados de oxazolidinona e um processo para a preparação dos mesmos |
| JP2004501965A (ja) | 2000-06-30 | 2004-01-22 | ファルマシア・アンド・アップジョン・カンパニー | 細菌感染を治療するための組成物および方法 |
| US6372919B1 (en) | 2001-01-11 | 2002-04-16 | Dov Pharmaceutical, Inc. | (+)-1-(3,4-dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as an anti-depressant agent |
| DOP2002000333A (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz |
| WO2002081470A1 (en) | 2001-04-07 | 2002-10-17 | Astrazeneca Ab | Oxazolidinones containing a sulfonimid group as antibiotics |
| GB0108793D0 (en) | 2001-04-07 | 2001-05-30 | Astrazeneca Ab | Chemical compounds |
| DE60206154T2 (de) | 2001-04-17 | 2006-06-29 | Merck & Co., Inc. | Bicyclo[3,1,0]hexan als strukturelement enthaltende oxazolidinon-antibiotika und deren derivate |
| EP1406889A2 (en) | 2001-07-09 | 2004-04-14 | Pharmacia Italia S.p.A. | Interaction inhibitors of tcf-4 with beta-catenin |
| EP1409464A4 (en) | 2001-07-16 | 2005-11-02 | Ranbaxy Lab Ltd | OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS |
| US6569887B2 (en) | 2001-08-24 | 2003-05-27 | Dov Pharmaceuticals Inc. | (−)-1-(3,4-Dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as a dopamine-reuptake |
| AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| BR0310074A (pt) | 2002-05-15 | 2005-03-08 | Ranbaxy Lab Ltd | Formas polimórficas de derivados de fenil oxazolidinona |
| WO2004009587A1 (en) | 2002-07-22 | 2004-01-29 | Orchid Chemicals & Pharmaceuticals Ltd | Oxazolidinone derivatives as antibacterial agents |
| CN1668308A (zh) | 2002-07-29 | 2005-09-14 | 兰贝克赛实验室有限公司 | 作为抗菌剂的噁唑烷酮衍生物 |
| EP1578734A1 (en) | 2002-08-22 | 2005-09-28 | Orchid Chemicals and Pharmaceuticals Ltd | Novel antibacterial agents |
| US6875784B2 (en) | 2002-10-09 | 2005-04-05 | Pharmacia & Upjohn Company | Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives |
| GB0229518D0 (en) | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| GB0229526D0 (en) | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| CA2521685A1 (en) | 2003-04-09 | 2004-10-21 | Pharmacia & Upjohn Company Llc | Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues |
| WO2005003087A2 (en) | 2003-07-01 | 2005-01-13 | Orchid Chemicals And Pharmaceuticals Ltd. | Oxazole derivatives as antibacterial agents |
| JP2007521284A (ja) * | 2003-07-02 | 2007-08-02 | メルク アンド カンパニー インコーポレーテッド | オキサゾリジノン系抗生物質及びその誘導体 |
| US20060247286A1 (en) * | 2003-07-02 | 2006-11-02 | Milton Hammond | Oxazolidinone antibiotics and derivatives thereof |
| EP1646629B1 (en) | 2003-07-02 | 2010-06-23 | Merck Sharp & Dohme Corp. | Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof |
| CN1816534A (zh) * | 2003-07-02 | 2006-08-09 | 默克制药公司 | 噁唑烷酮抗生素及其衍生物 |
| CN1816547A (zh) * | 2003-07-02 | 2006-08-09 | 默克制药公司 | 噁唑烷酮抗生素及其衍生物 |
| KR100854211B1 (ko) | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
| WO2005082897A1 (en) | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone antibacterial agents |
| WO2005082899A1 (en) * | 2004-01-28 | 2005-09-09 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| WO2005082900A2 (en) | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone amidoximes as antibacterial agents |
| ATE451364T1 (de) * | 2004-02-23 | 2009-12-15 | Glaxo Group Ltd | Als modulatoren des dopamin-d3-rezeptors geeignete azabicycloä3.1.0ühexanderivate |
| US20080064689A1 (en) | 2004-05-25 | 2008-03-13 | Astrazeneca Ab | 3-[4-(6-Pyridin-3-Yl)-3-Phenyl] -5-(1H-1,2,3-Triazol-1-Ylmethyl)-1,3-Oxazolidin-2-Ones as Antibacterial Agents |
| MXPA06013540A (es) | 2004-05-25 | 2007-01-26 | Astrazeneca Ab | Derivados de 3-(4-(2 -dihidroisoxasol -3-ilpiridin-5-il) fenil)-5- triazol-1- ilmetiloxazolidin -2-ona como inhibidores de mao para el tratamiento de infecciones bacterianas. |
| WO2006035283A1 (en) | 2004-09-27 | 2006-04-06 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| WO2006043121A1 (en) | 2004-10-20 | 2006-04-27 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| WO2006096810A2 (en) | 2005-03-08 | 2006-09-14 | Dov Pharmaceutical, Inc. | Methods and compositions for production, formulation and use of 1-aryl-3-azabicyclo[3.1.0] hexanes |
| KR101284573B1 (ko) | 2005-04-12 | 2013-07-11 | 바이코어 파마 아베 | 신규한 트리시클릭 안지오텐신 ⅱ 아고니스트 |
| GB0507602D0 (en) * | 2005-04-14 | 2005-05-18 | Glaxo Group Ltd | Compounds |
| GB0507601D0 (en) | 2005-04-14 | 2005-05-18 | Glaxo Group Ltd | Compounds |
| ATE484502T1 (de) | 2005-06-14 | 2010-10-15 | Glaxo Group Ltd | Neue verbindungen |
| EP1745784A1 (en) | 2005-06-27 | 2007-01-24 | Ferrer Internacional, S.A. | Oxazolidinone derivatives and use thereof as antibiotics |
| CA2614105A1 (en) | 2005-07-06 | 2007-01-11 | Pharmacia & Upjohn Company Llc | Oxazolidinone carboxamides containing azetidine and cyclobutane as antibacterial agents |
| AU2006275870B2 (en) | 2005-07-27 | 2013-01-10 | Otsuka America Pharmaceutical, Inc. | Novel 1-aryl-3-azabicyclo[3.1.0]hexanes: preparation and use to treat neuropsychiatric disorders |
| ATE487715T1 (de) | 2005-08-22 | 2010-11-15 | Glaxo Group Ltd | Triazolderivate als modulatoren von dopamin-d3- rezeptoren |
| GB0517193D0 (en) * | 2005-08-22 | 2005-09-28 | Glaxo Group Ltd | Novel use |
| GB0517191D0 (en) | 2005-08-22 | 2005-09-28 | Glaxo Group Ltd | Compounds |
| GB0517187D0 (en) * | 2005-08-22 | 2005-09-28 | Glaxo Group Ltd | Compounds |
| GB0517175D0 (en) | 2005-08-22 | 2005-09-28 | Glaxo Group Ltd | Compounds |
| KR20070038236A (ko) | 2005-10-05 | 2007-04-10 | 일동제약주식회사 | 신규 옥사졸리디논 포름 아미드 유도체 및 그 제조방법 |
| JP2009523764A (ja) | 2006-01-19 | 2009-06-25 | ラボラトリオス・サルバト・ソシエダッド・アノニマ | 抗菌活性を有するジカルボニル化合物 |
| DK1987025T3 (da) | 2006-02-14 | 2009-12-07 | Pfizer Prod Inc | Benzoxazinon og benzoxazepinonoxazolidinoner som antibakterielle midler |
| CN100406455C (zh) | 2006-02-20 | 2008-07-30 | 中国科学院上海药物研究所 | 含三氮唑基的噁唑烷酮类化合物及其制备方法和用途 |
| EP2181994B1 (en) | 2006-03-31 | 2014-05-28 | Research Foundation Itsuu Laboratory | Antimicrobial compounds |
| WO2007113258A1 (en) | 2006-04-03 | 2007-10-11 | Glaxo Group Limited | Azabicyclo [3. 1. o] hexane derivatives as modulators of dopamine d3 receptors |
| GB0607892D0 (en) * | 2006-04-03 | 2006-05-31 | Glaxo Group Ltd | Novel compounds |
| AU2007233715A1 (en) * | 2006-04-03 | 2007-10-11 | Glaxo Group Limited | Azabicyclo [3. 1. 0] hexyl derivatives as modulators of dopamine D3 receptors |
| AU2007252375A1 (en) | 2006-05-23 | 2007-11-29 | Joong-Hoon Nam | Golf swing training machine |
| US8138377B2 (en) | 2006-11-07 | 2012-03-20 | Dov Pharmaceutical, Inc. | Arylbicyclo[3.1.0]hexylamines and methods and compositions for their preparation and use |
| GB0625198D0 (en) | 2006-12-18 | 2007-01-24 | Glaxo Group Ltd | Chemical compounds |
| US20080176860A1 (en) | 2007-01-19 | 2008-07-24 | Lutz Weber | Pyridin-2-one compounds |
| WO2008136754A1 (en) | 2007-05-07 | 2008-11-13 | Astrazeneca Ab | Novel benzyl - 2 -oxo-piperazinyl/ 7-oxo/5-oxa- [1,4] diazepanyl/ 2 -oxo- tetrahydropyrimidinyl derivatives |
| EP2167083B1 (en) | 2007-06-06 | 2015-10-28 | Euthymics Bioscience, Inc. | 1- heteroaryl-3-azabicyclo[3.1.0]hexanes, methods for their preparation and their use as medicaments |
| GB0716632D0 (en) | 2007-08-24 | 2007-10-03 | Glaxo Group Ltd | Compounds |
| CN101434584A (zh) | 2007-11-15 | 2009-05-20 | 中山大学 | 具有抗菌活性的手性噁唑烷酮类化合物 |
-
2010
- 2010-06-22 MX MX2012000231A patent/MX2012000231A/es not_active Application Discontinuation
- 2010-06-22 CN CN2010800285561A patent/CN102803224A/zh active Pending
- 2010-06-22 CA CA2765692A patent/CA2765692A1/en not_active Abandoned
- 2010-06-22 BR BR112012000657A patent/BR112012000657A2/pt not_active IP Right Cessation
- 2010-06-22 JP JP2012516978A patent/JP5696142B2/ja not_active Expired - Fee Related
- 2010-06-22 WO PCT/IN2010/000428 patent/WO2010150281A2/en not_active Ceased
- 2010-06-22 US US13/380,744 patent/US8906913B2/en not_active Expired - Fee Related
- 2010-06-22 KR KR1020127000778A patent/KR20120106697A/ko not_active Withdrawn
- 2010-06-22 RU RU2012102094/04A patent/RU2012102094A/ru unknown
- 2010-06-22 EP EP10747300.1A patent/EP2445887B1/en not_active Not-in-force
- 2010-06-22 AU AU2010264027A patent/AU2010264027B9/en not_active Expired - Fee Related
- 2010-06-25 AR ARP100102281A patent/AR077251A1/es unknown
-
2011
- 2011-12-21 ZA ZA2011/09437A patent/ZA201109437B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2765692A1 (en) | 2010-12-29 |
| US20120165320A1 (en) | 2012-06-28 |
| JP5696142B2 (ja) | 2015-04-08 |
| KR20120106697A (ko) | 2012-09-26 |
| EP2445887B1 (en) | 2014-11-05 |
| RU2012102094A (ru) | 2013-08-10 |
| AR077251A1 (es) | 2011-08-10 |
| CN102803224A (zh) | 2012-11-28 |
| ZA201109437B (en) | 2013-03-27 |
| AU2010264027B2 (en) | 2013-05-30 |
| AU2010264027B9 (en) | 2013-06-13 |
| WO2010150281A3 (en) | 2011-04-21 |
| MX2012000231A (es) | 2012-03-07 |
| US8906913B2 (en) | 2014-12-09 |
| AU2010264027A1 (en) | 2012-01-19 |
| EP2445887A2 (en) | 2012-05-02 |
| WO2010150281A2 (en) | 2010-12-29 |
| JP2012531403A (ja) | 2012-12-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FIC20230010I1 (fi) | Sasitutsumabigovitekaani | |
| FIC20210039I1 (fi) | Duvelisibi | |
| NL301265I1 (nl) | Quizartinib | |
| NL300873I2 (nl) | Venetoclax | |
| HUE045331T2 (hu) | Szikkasztótest | |
| DK2430035T3 (da) | Uracylspipooxetannukleosider | |
| BRPI1008827A2 (pt) | deisobutenizador | |
| DE112010004249A5 (de) | Spindelaktor | |
| DE112009005323A5 (de) | Hebelarmprüfmaschine | |
| BR112012004964A2 (pt) | girocóptero | |
| BRPI1008070A2 (pt) | tricianoboratos | |
| EP2409976A4 (en) | GLYCINE TRANSPORTER INHIBITOR | |
| FI20095891A0 (fi) | Polttomoottorisovitelma | |
| DK2483126T3 (da) | Skinnekøretøj | |
| DK2506968T3 (da) | Faujasit-zeolit | |
| DE112010003255A5 (de) | Fördergutverteiler | |
| EP2518828A4 (en) | Rfid tag | |
| FI20090100A0 (fi) | Biotinidaasimääritys | |
| BR112012003616A2 (pt) | metilpirroloprimidinacarboxamidas | |
| DE112010003843T8 (de) | Lastansteuervorrichtung | |
| FI8660U1 (fi) | Pilaripehmuste | |
| FI20090173A0 (fi) | Pystypuun karsintalaite | |
| AT506924A3 (de) | Bauprojektor | |
| AT508508A3 (de) | Heuballenbohrer | |
| NO20091744L (no) | Babylogger |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application fees: application dismissed [chapter 8.6 patent gazette] | ||
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |