BRPI0406913A - Dispersão de cristais de sabor mascarado ou de grânulos de substâncias ativas, cápsulas macias mascáveis preenchidas com a referida dispersão, e processo para a preparação da mesma - Google Patents

Dispersão de cristais de sabor mascarado ou de grânulos de substâncias ativas, cápsulas macias mascáveis preenchidas com a referida dispersão, e processo para a preparação da mesma

Info

Publication number
BRPI0406913A
BRPI0406913A BR0406913-7A BRPI0406913A BRPI0406913A BR PI0406913 A BRPI0406913 A BR PI0406913A BR PI0406913 A BRPI0406913 A BR PI0406913A BR PI0406913 A BRPI0406913 A BR PI0406913A
Authority
BR
Brazil
Prior art keywords
dispersion
granules
preparing
capsules filled
crystals
Prior art date
Application number
BR0406913-7A
Other languages
English (en)
Inventor
Julien Meissonnier
Fabrice Rose
Marie Madeleine Bohn
Original Assignee
Scherer Technologies Inc R P
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scherer Technologies Inc R P filed Critical Scherer Technologies Inc R P
Publication of BRPI0406913A publication Critical patent/BRPI0406913A/pt
Publication of BRPI0406913B1 publication Critical patent/BRPI0406913B1/pt
Publication of BRPI0406913B8 publication Critical patent/BRPI0406913B8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4816—Wall or shell material
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Physiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nutrition Science (AREA)
  • Organic Chemistry (AREA)
  • Rheumatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cosmetics (AREA)

Abstract

"DISPERSãO DE CRISTAIS DE SABOR MASCARADO OU DE GRâNULOS DE SUBSTâNCIAS ATIVAS, CáPSULAS MACIAS MASCáVEIS PREENCHIDAS COM A REFERIDA DISPERSãO, E PROCESSO PARA A PREPARAçãO DA MESMA". A presente invenção se refere a uma dispersão de cristais ou de grânulos de substância ativa em um veículo lipófilo, os referidos cristais e grânulos sendo revestidos por um revestimento com o objetivo de mascaramento de sabor. A presente invenção também se refere a formas de dosagem unitárias e de forma preferida a cápsulas de gelatina macia mascáveis ou de rápida dissolução, preenchidas com a referida dispersão assim como a processo para a fabricação da mesma.
BRPI0406913A 2003-01-24 2004-01-21 dispersão de cristais de sabor mascarado ou de grânulos de substâncias ativas, cápsulas macias mascáveis preenchidas com a referida dispersão, e processo para a preparação da mesma BRPI0406913B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0300824A FR2850275B1 (fr) 2003-01-24 2003-01-24 Capsules molles a macher contenant une substance active a gout masque
PCT/US2004/001463 WO2004066925A2 (en) 2003-01-24 2004-01-21 Dispersion of taste masked crystals or granules of active substances, chewable soft capsules filled with said dispersion, and process for preparing same

Publications (3)

Publication Number Publication Date
BRPI0406913A true BRPI0406913A (pt) 2006-01-03
BRPI0406913B1 BRPI0406913B1 (pt) 2016-03-01
BRPI0406913B8 BRPI0406913B8 (pt) 2021-05-25

Family

ID=32669215

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0406913A BRPI0406913B8 (pt) 2003-01-24 2004-01-21 dispersão de cristais de sabor mascarado ou de grânulos de substâncias ativas, cápsulas macias mascáveis preenchidas com a referida dispersão, e processo para a preparação da mesma

Country Status (18)

Country Link
EP (1) EP1592402B1 (pt)
JP (1) JP5371187B2 (pt)
CN (2) CN103169655A (pt)
AR (1) AR042902A1 (pt)
AU (1) AU2004207498B2 (pt)
BR (1) BRPI0406913B8 (pt)
CA (1) CA2512988C (pt)
DK (1) DK1592402T3 (pt)
ES (1) ES2415660T3 (pt)
FR (1) FR2850275B1 (pt)
MX (1) MXPA05007683A (pt)
NO (1) NO339528B1 (pt)
NZ (1) NZ541753A (pt)
PT (1) PT1592402E (pt)
RU (1) RU2362546C2 (pt)
SI (1) SI1592402T1 (pt)
UA (1) UA84140C2 (pt)
WO (1) WO2004066925A2 (pt)

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US8124072B2 (en) 2003-09-29 2012-02-28 Soft Gel Technologies, Inc. Solubilized CoQ-10
US7169385B2 (en) 2003-09-29 2007-01-30 Ronald G. Udell Solubilized CoQ-10 and carnitine
US20070292501A1 (en) * 2006-06-05 2007-12-20 Udell Ronald G Chewable soft gelatin capsules
US20080020022A1 (en) * 2006-06-05 2008-01-24 Udell Ronald G Chewable co-enzyme q-10 capsule
US8343541B2 (en) 2007-03-15 2013-01-01 Soft Gel Technologies, Inc. Ubiquinol and alpha lipoic acid compositions
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FR2935084B1 (fr) * 2008-08-19 2011-05-06 Pancosma Sa Pour L Ind Des Produits Biochimiques Additif pour l'alimentation animale et son procede de preparation
GB201006218D0 (en) 2010-04-14 2010-06-02 Ayanda As Composition
CA2706270C (en) * 2010-06-03 2020-01-07 Accucaps Industries Limited Pharmaceutical formulations of statins and omega-3 fatty acids for encapsulation
CA3065589C (en) * 2010-06-03 2022-04-26 Catalent Ontario Limited Multi phase soft gel capsules, apparatus and method thereof
BR112013020237A2 (pt) * 2011-02-11 2021-03-16 Ctc Bio, Inc. Processo para preparar um filme contendo base livre de sildenafila e filme contendo base livre de sildenafila
EP2696846B1 (en) * 2011-04-11 2018-01-17 Vitux Group AS Oral pharmaceutical dispersion compositions
WO2012144943A1 (en) * 2011-04-18 2012-10-26 Lipidor Ab Liquid carrier for oral delivery of a pharmacologically active agent
CN102241782B (zh) * 2011-05-18 2013-01-30 清华大学 一种淀粉乙酸酯的制备方法及其在去除水中硝酸盐的应用
CN102813275B (zh) * 2011-06-10 2015-09-30 杭州养生堂保健品有限公司 一种咀嚼型软胶囊皮和咀嚼型软胶囊
DE102012014848A1 (de) * 2012-07-27 2012-10-31 Heilerde-Gesellschaft Luvos Just GmbH & Co. KG Heilerde-Zubereitung
US20150209360A1 (en) * 2014-01-30 2015-07-30 Orbz, Llc Oral caffeine delivery composition
FR3027802B1 (fr) * 2014-10-31 2018-03-02 Ethypharm Granules de principe actif a double masquage de gout, leur procede de preparation et comprimes orodispersibles les contenant
US9867779B2 (en) 2015-03-26 2018-01-16 Patheon Softgels Inc. Liquisoft capsules
US20170266115A1 (en) 2016-03-15 2017-09-21 Acer Therapeutics Inc. Palatable compositions including sodium phenylbutyrate and uses thereof
JP6942342B2 (ja) * 2016-11-02 2021-09-29 富士カプセル株式会社 ソフトカプセル皮膜
JP2018121699A (ja) * 2017-01-30 2018-08-09 株式会社アクレス クリルオイルを充填したカプセル剤
CN107373744B (zh) * 2017-07-13 2018-11-09 云南中烟工业有限责任公司 一种维生素c微胶囊的制备方法及其在卷烟中的应用
CN108524464A (zh) * 2018-05-17 2018-09-14 安士制药（中山）有限公司 一种西甲硅油软胶囊的制备方法
AU2020225818B2 (en) 2019-02-22 2025-09-18 Catalent U.K. Swindon Zydis Limited Preserving functionally-coated API particles produced by solventless mixing processes in aqueous suspension
KR20210129649A (ko) 2019-02-22 2021-10-28 카탈렌트 유.케이. 스윈던 지디스 리미티드 이부프로펜을 포함하는 약학적 조성물의 응집, 에어레이션 최소화 및 코팅 보존
JP7543291B2 (ja) 2019-02-22 2024-09-02 キャタレント・ユーケー・スウィンドン・ザイディス・リミテッド 医薬品の崩壊時間を安定させるための、保管中の薬物粒子コーティング材料の凝集を最小限に抑える
ES2961850T3 (es) 2019-02-22 2024-03-14 Catalent Uk Swindon Zydis Ltd Minimización de la aireación de suspensiones durante la mezcla en línea
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WO2022106923A1 (en) 2020-11-18 2022-05-27 BioPharma Synergies, S. L. Orodispersible powder composition comprising an antihistamine compound

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Also Published As

Publication number Publication date
BRPI0406913B8 (pt) 2021-05-25
PT1592402E (pt) 2013-06-25
AU2004207498A1 (en) 2004-08-12
NZ541753A (en) 2008-12-24
CA2512988C (en) 2015-11-10
AU2004207498B2 (en) 2008-10-30
CA2512988A1 (en) 2004-08-12
MXPA05007683A (es) 2005-09-30
NO20053681L (no) 2005-08-23
NO339528B1 (no) 2016-12-27
SI1592402T1 (sl) 2013-08-30
RU2362546C2 (ru) 2009-07-27
EP1592402B1 (en) 2013-03-20
EP1592402A4 (en) 2009-01-14
AR042902A1 (es) 2005-07-06
WO2004066925B1 (en) 2004-12-09
HK1082659A1 (en) 2006-06-16
CN103169655A (zh) 2013-06-26
DK1592402T3 (da) 2013-06-24
JP2007525413A (ja) 2007-09-06
WO2004066925A3 (en) 2004-10-28
EP1592402A2 (en) 2005-11-09
ES2415660T3 (es) 2013-07-26
JP5371187B2 (ja) 2013-12-18
BRPI0406913B1 (pt) 2016-03-01
RU2005126729A (ru) 2006-03-10
UA84140C2 (ru) 2008-09-25
FR2850275B1 (fr) 2005-04-08
WO2004066925A2 (en) 2004-08-12
CN1741787A (zh) 2006-03-01
FR2850275A1 (fr) 2004-07-30

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B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
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Ipc: A61K 47/06 (2011.01), A61K 9/00 (2011.01), A61K 9/

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