BRPI0407012A - Processo para a produção de um composto e uso do composto - Google Patents
Processo para a produção de um composto e uso do compostoInfo
- Publication number
- BRPI0407012A BRPI0407012A BR0407012-7A BRPI0407012A BRPI0407012A BR PI0407012 A BRPI0407012 A BR PI0407012A BR PI0407012 A BRPI0407012 A BR PI0407012A BR PI0407012 A BRPI0407012 A BR PI0407012A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- iii
- producing
- pyrrolidone
- salt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Addiction (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
Abstract
"PROCESSO PARA A PRODUçãO DE UM COMPOSTO E USO DO COMPOSTO". A presente invenção refere-se a processos para a produção de um composto tendo a seguinte fórmula (I) pela conversão de um composto tendo a fórmula (II) com 2-pirrolidona, o referido 2-pirrolidona sendo usado em excesso, com relação ao composto (II); assim como a processos para a produção de um composto tendo a seguinte fórmula (III) compreendendo as seguintes etapas: (A) a preparação do composto (I); (B) a reação de redução, a qual produz o composto (III) na forma de um sal; e (C) a liberação do composto (III) a partir do sal.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10304141A DE10304141B4 (de) | 2003-02-03 | 2003-02-03 | Verfahren zur Herstellung von Chinazolin-Alkaloiden |
| PCT/EP2004/000485 WO2004069836A1 (de) | 2003-02-03 | 2004-01-22 | Verfahren zur herstellung von chinazolin-alkaloiden |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0407012A true BRPI0407012A (pt) | 2006-01-10 |
Family
ID=32747532
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0407012-7A BRPI0407012A (pt) | 2003-02-03 | 2004-01-22 | Processo para a produção de um composto e uso do composto |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US7495096B2 (pt) |
| EP (1) | EP1590351B1 (pt) |
| JP (1) | JP2006516578A (pt) |
| KR (1) | KR20050096165A (pt) |
| CN (1) | CN100558727C (pt) |
| AR (1) | AR042946A1 (pt) |
| AT (1) | ATE407135T1 (pt) |
| AU (1) | AU2004208873B2 (pt) |
| BR (1) | BRPI0407012A (pt) |
| CA (1) | CA2514945A1 (pt) |
| DE (2) | DE10304141B4 (pt) |
| DK (1) | DK1590351T3 (pt) |
| EA (1) | EA009047B1 (pt) |
| ES (1) | ES2314366T3 (pt) |
| MX (1) | MXPA05008179A (pt) |
| MY (1) | MY141734A (pt) |
| NO (1) | NO20053689L (pt) |
| NZ (1) | NZ541101A (pt) |
| PL (1) | PL378406A1 (pt) |
| PT (1) | PT1590351E (pt) |
| SI (1) | SI1590351T1 (pt) |
| TW (1) | TW200418811A (pt) |
| UA (1) | UA81287C2 (pt) |
| WO (1) | WO2004069836A1 (pt) |
| ZA (1) | ZA200505160B (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102004048927A1 (de) * | 2004-10-06 | 2006-04-20 | Lts Lohmann Therapie-Systeme Ag | Pharmazeutische Kombination enthaltend Desoxypeganin und Cyp2D6 Inhibitoren |
| BR112020001698A2 (pt) | 2017-08-03 | 2020-07-21 | Galectin Sciences, Llc | compostos para prevenção e tratamento de distúrbios médicos e usos dos mesmos |
| KR102728780B1 (ko) * | 2021-11-30 | 2024-11-08 | 이화여자대학교 산학협력단 | 데옥시바시시논을 유효성분으로 포함하는 미백용 조성물 및 상기 데옥시바시시논 제조방법 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU605614A1 (ru) * | 1971-10-20 | 1978-05-05 | Ордена Трудового Красного Знамени Институт Химии Растительных Веществ Ан Узбекской Сср | Антихолинэстеразное средство |
| JP3180464B2 (ja) * | 1991-08-30 | 2001-06-25 | 新日本理化株式会社 | ジアセタール化合物の製造方法 |
| DE19530606A1 (de) * | 1995-08-21 | 1997-02-27 | Basf Ag | 1-(Pyridyl)-pyrazole |
| JP3958452B2 (ja) * | 1997-10-31 | 2007-08-15 | 大日精化工業株式会社 | 新規化学発光試薬及びその製造方法 |
| DE19906979B4 (de) | 1999-02-19 | 2004-07-08 | Lts Lohmann Therapie-Systeme Ag | Verwendung von Desoxypeganin zur Behandlung der Nikotinabhängigkeit |
| DE19906978B4 (de) | 1999-02-19 | 2004-07-08 | Lts Lohmann Therapie-Systeme Ag | Pharmazeutische Zusammensetzung enthaltend Desoxypeganin zur Behandlung der Drogenabhängigkeit |
| DE19906975B4 (de) | 1999-02-19 | 2004-04-15 | Lts Lohmann Therapie-Systeme Ag | Arzneiform zur Behandlung von Alzheimer'scher Demenz |
-
2003
- 2003-02-03 DE DE10304141A patent/DE10304141B4/de not_active Expired - Fee Related
-
2004
- 2004-01-22 JP JP2006501573A patent/JP2006516578A/ja active Pending
- 2004-01-22 MX MXPA05008179A patent/MXPA05008179A/es active IP Right Grant
- 2004-01-22 EA EA200501135A patent/EA009047B1/ru not_active IP Right Cessation
- 2004-01-22 CA CA002514945A patent/CA2514945A1/en not_active Abandoned
- 2004-01-22 DK DK04704202T patent/DK1590351T3/da active
- 2004-01-22 AT AT04704202T patent/ATE407135T1/de active
- 2004-01-22 BR BR0407012-7A patent/BRPI0407012A/pt not_active Application Discontinuation
- 2004-01-22 AU AU2004208873A patent/AU2004208873B2/en not_active Ceased
- 2004-01-22 KR KR1020057013954A patent/KR20050096165A/ko not_active Ceased
- 2004-01-22 SI SI200430943T patent/SI1590351T1/sl unknown
- 2004-01-22 WO PCT/EP2004/000485 patent/WO2004069836A1/de not_active Ceased
- 2004-01-22 ES ES04704202T patent/ES2314366T3/es not_active Expired - Lifetime
- 2004-01-22 PL PL378406A patent/PL378406A1/pl not_active Application Discontinuation
- 2004-01-22 EP EP04704202A patent/EP1590351B1/de not_active Expired - Lifetime
- 2004-01-22 US US10/544,265 patent/US7495096B2/en not_active Expired - Fee Related
- 2004-01-22 DE DE502004007980T patent/DE502004007980D1/de not_active Expired - Lifetime
- 2004-01-22 NZ NZ541101A patent/NZ541101A/en not_active IP Right Cessation
- 2004-01-22 UA UAA200507716A patent/UA81287C2/uk unknown
- 2004-01-22 PT PT04704202T patent/PT1590351E/pt unknown
- 2004-01-22 CN CNB2004800034182A patent/CN100558727C/zh not_active Expired - Fee Related
- 2004-01-28 AR ARP040100246A patent/AR042946A1/es unknown
- 2004-01-30 MY MYPI20040294A patent/MY141734A/en unknown
- 2004-02-02 TW TW093102290A patent/TW200418811A/zh unknown
-
2005
- 2005-06-24 ZA ZA200505160A patent/ZA200505160B/en unknown
- 2005-07-29 NO NO20053689A patent/NO20053689L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MY141734A (en) | 2010-06-15 |
| EA009047B1 (ru) | 2007-10-26 |
| AR042946A1 (es) | 2005-07-06 |
| JP2006516578A (ja) | 2006-07-06 |
| PL378406A1 (pl) | 2006-04-03 |
| TW200418811A (en) | 2004-10-01 |
| ZA200505160B (en) | 2007-01-31 |
| US20060084669A1 (en) | 2006-04-20 |
| KR20050096165A (ko) | 2005-10-05 |
| CA2514945A1 (en) | 2004-08-19 |
| ES2314366T3 (es) | 2009-03-16 |
| DE10304141B4 (de) | 2006-03-09 |
| UA81287C2 (en) | 2007-12-25 |
| PT1590351E (pt) | 2008-11-21 |
| CN1745084A (zh) | 2006-03-08 |
| AU2004208873A1 (en) | 2004-08-19 |
| EP1590351A1 (de) | 2005-11-02 |
| WO2004069836A1 (de) | 2004-08-19 |
| NZ541101A (en) | 2009-03-31 |
| SI1590351T1 (sl) | 2009-02-28 |
| MXPA05008179A (es) | 2006-02-17 |
| DE502004007980D1 (de) | 2008-10-16 |
| NO20053689L (no) | 2005-07-29 |
| US7495096B2 (en) | 2009-02-24 |
| ATE407135T1 (de) | 2008-09-15 |
| CN100558727C (zh) | 2009-11-11 |
| EA200501135A1 (ru) | 2006-02-24 |
| DK1590351T3 (da) | 2008-12-15 |
| DE10304141A1 (de) | 2004-08-26 |
| HK1075898A1 (zh) | 2005-12-30 |
| EP1590351B1 (de) | 2008-09-03 |
| AU2004208873B2 (en) | 2009-12-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B11E | Dismissal acc. art. 34 of ipl - requirements for examination incomplete | ||
| B11T | Dismissal of application maintained [chapter 11.20 patent gazette] |