BRPI0409791A - ligandos de receptores de canabinóides e sua utilização - Google Patents

ligandos de receptores de canabinóides e sua utilização

Info

Publication number
BRPI0409791A
BRPI0409791A BRPI0409791-2A BRPI0409791A BRPI0409791A BR PI0409791 A BRPI0409791 A BR PI0409791A BR PI0409791 A BRPI0409791 A BR PI0409791A BR PI0409791 A BRPI0409791 A BR PI0409791A
Authority
BR
Brazil
Prior art keywords
cannabinoid receptor
receptor ligands
cannabinide
animals
act
Prior art date
Application number
BRPI0409791-2A
Other languages
English (en)
Inventor
Philip Albert Carpino
Robert Lee Dow
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BRPI0409791A publication Critical patent/BRPI0409791A/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Reproductive Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Rheumatology (AREA)
  • Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"LIGANDOS DE RECEPTORES DE CANABINóIDES E SUA UTILIZAçãO". Estão aqui descritos compostos de Fórmula (I) e (I) que atuam como ligandos de receptores de canabinóides e a sua utilização no tratamento de doenças ligadas à mediação dos receptores de canabinóides em animais.
BRPI0409791-2A 2003-04-23 2004-04-13 ligandos de receptores de canabinóides e sua utilização BRPI0409791A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46490803P 2003-04-23 2003-04-23
PCT/IB2004/001357 WO2004094421A1 (en) 2003-04-23 2004-04-13 Cannabinoid receptor ligands and uses thereof

Publications (1)

Publication Number Publication Date
BRPI0409791A true BRPI0409791A (pt) 2006-05-30

Family

ID=33310977

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0409791-2A BRPI0409791A (pt) 2003-04-23 2004-04-13 ligandos de receptores de canabinóides e sua utilização

Country Status (31)

Country Link
US (1) US20040214856A1 (pt)
EP (1) EP1622903B1 (pt)
JP (1) JP2006524225A (pt)
KR (1) KR20060006048A (pt)
CN (1) CN1809566A (pt)
AP (1) AP2005003427A0 (pt)
AR (1) AR044037A1 (pt)
AT (1) ATE409700T1 (pt)
AU (1) AU2004232552A1 (pt)
BR (1) BRPI0409791A (pt)
CA (1) CA2521538A1 (pt)
CL (1) CL2004000827A1 (pt)
CO (1) CO5640084A2 (pt)
DE (1) DE602004016839D1 (pt)
EA (1) EA200501504A1 (pt)
EC (1) ECSP056117A (pt)
ES (1) ES2309517T3 (pt)
GT (1) GT200400076A (pt)
IS (1) IS8054A (pt)
MA (1) MA27766A1 (pt)
MX (1) MXPA05011454A (pt)
NL (1) NL1026027C2 (pt)
NO (1) NO20055516L (pt)
OA (1) OA13047A (pt)
PA (1) PA8600601A1 (pt)
PE (1) PE20050419A1 (pt)
TN (1) TNSN05272A1 (pt)
TW (1) TW200510419A (pt)
UY (1) UY28276A1 (pt)
WO (1) WO2004094421A1 (pt)
ZA (1) ZA200508568B (pt)

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TW200510419A (en) 2005-03-16
NL1026027C2 (nl) 2005-07-05
IS8054A (is) 2005-09-29
ECSP056117A (es) 2006-03-01
MXPA05011454A (es) 2005-12-12
CO5640084A2 (es) 2006-05-31
OA13047A (en) 2006-11-10
AR044037A1 (es) 2005-08-24
EP1622903A1 (en) 2006-02-08
EA200501504A1 (ru) 2006-04-28
KR20060006048A (ko) 2006-01-18
CA2521538A1 (en) 2004-11-04
ATE409700T1 (de) 2008-10-15
CL2004000827A1 (es) 2005-03-04
TNSN05272A1 (fr) 2007-07-10
WO2004094421A1 (en) 2004-11-04
MA27766A1 (fr) 2006-02-01
DE602004016839D1 (de) 2008-11-13
GT200400076A (es) 2004-12-16
NO20055516L (no) 2005-11-22
AU2004232552A1 (en) 2004-11-04
PE20050419A1 (es) 2005-06-18
CN1809566A (zh) 2006-07-26
UY28276A1 (es) 2004-11-30
US20040214856A1 (en) 2004-10-28
ZA200508568B (en) 2007-04-25
JP2006524225A (ja) 2006-10-26
NL1026027A1 (nl) 2004-10-27
ES2309517T3 (es) 2008-12-16
EP1622903B1 (en) 2008-10-01
AP2005003427A0 (en) 2005-12-31
PA8600601A1 (es) 2005-05-24

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