BRPI0410906A - triazolopirimidinas - Google Patents

triazolopirimidinas

Info

Publication number
BRPI0410906A
BRPI0410906A BRPI0410906-6A BRPI0410906A BRPI0410906A BR PI0410906 A BRPI0410906 A BR PI0410906A BR PI0410906 A BRPI0410906 A BR PI0410906A BR PI0410906 A BRPI0410906 A BR PI0410906A
Authority
BR
Brazil
Prior art keywords
triazolopyrimidines
substances
preparing
relates
formulas
Prior art date
Application number
BRPI0410906-6A
Other languages
English (en)
Inventor
Olaf Gebauer
Ulrich Heinemann
Hans-Ludwig Elbe
Herbert Gayer
Stefan Herrmann
Joerg Nico Greul
Bernd-Wieland Krueger
Stefan Hillebrand
Ronald Ebbert
Ulrike Wachendorff-Neumann
Peter Dahmen
Karl-Heinz Kuck
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0410906A publication Critical patent/BRPI0410906A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

"TRIAZOLOPIRIMIDINAS". A invenção refere-se a triazolopirimidinas da fórmula (I) em que R¬ 1¬, R¬ 2¬, R¬ 3¬ e X possuem os significados mencionados na descrição, a um processo para preparação destas substâncias e ao seu uso para o combate de microorganismos indesejados. A invenção refere-se também a novos produtos intermediários das fórmulas (II), (IV), (V-a), (V-b), bem como a processos para preparação destas substâncias.
BRPI0410906-6A 2003-06-04 2004-06-01 triazolopirimidinas BRPI0410906A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10325133A DE10325133A1 (de) 2003-06-04 2003-06-04 Triazolopyrimidine
PCT/EP2004/005876 WO2004108727A1 (de) 2003-06-04 2004-06-01 Triazolopyrimidine

Publications (1)

Publication Number Publication Date
BRPI0410906A true BRPI0410906A (pt) 2006-06-27

Family

ID=33482458

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0410906-6A BRPI0410906A (pt) 2003-06-04 2004-06-01 triazolopirimidinas

Country Status (14)

Country Link
US (1) US20070275985A1 (pt)
EP (1) EP1641798A1 (pt)
JP (1) JP2006526587A (pt)
KR (1) KR20060015304A (pt)
CN (1) CN1802379A (pt)
BR (1) BRPI0410906A (pt)
CO (1) CO5721005A2 (pt)
CR (1) CR8074A (pt)
DE (1) DE10325133A1 (pt)
EC (1) ECSP056201A (pt)
IL (1) IL172098A0 (pt)
MX (1) MXPA05012951A (pt)
WO (1) WO2004108727A1 (pt)
ZA (1) ZA200509637B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1828190A1 (de) * 2004-12-17 2007-09-05 Basf Aktiengesellschaft 7-amino-6-heteroaryl-1,2,4-triazoloý1,5-a¨pyrimidine und ihre verwendung zur bek[mpfung von schadpilzen
US20080227796A1 (en) * 2004-12-17 2008-09-18 Basf Aktiengesellschaft 7-Amino-6-Hetaryl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds and the Use Thereof for Controlling Pathogenic Fungi
US20080139581A1 (en) * 2005-03-02 2008-06-12 Basf Aktiengesellschaft 2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
WO2006122740A2 (de) * 2005-05-17 2006-11-23 Basf Aktiengesellschaft 7-AMINO-6-HETARYLIMIDAZOLO[1,2-a]PYRIMIDIN-VERBINDUNGEN UND IHRE VERWENDUNG ZU BEKÄMPFUNG VON SCHADPILZEN
WO2007006723A1 (de) * 2005-07-13 2007-01-18 Basf Aktiengesellschaft 7-amino-6-tetrazolyl-1,2,4-triazolo[1,5-a]pyrimidin-verbindungen und ihre verwendung zur bekämpfung von schadpilzen
WO2007101870A1 (de) * 2006-03-08 2007-09-13 Basf Se Substituierte triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
CN101153041B (zh) * 2006-09-28 2010-05-12 中国科学院化学研究所 1,2,3-三唑并1,3-二氮杂环化合物及其制备方法与应用
EP2131658A2 (en) * 2007-01-30 2009-12-16 Basf Se Method for improving plant health
EP1952691A3 (en) * 2007-01-31 2008-09-17 Basf Se Method for improving plant health by application of a triazolopyrimidine derivative
US9101131B2 (en) 2007-12-03 2015-08-11 Valent U.S.A., Corporation Seed treatment formulations
CN101969765B (zh) * 2007-12-03 2014-03-19 瓦伦特美国有限公司 种子处理制剂及使用方法
EP2204366A1 (de) 2008-12-19 2010-07-07 Bayer CropScience AG Herbizid und insektizid wirksame phenylsubstituierte Pyridazinone
WO2011035878A1 (de) 2009-09-25 2011-03-31 Bayer Cropscience Ag Herbizid wirksame phenylsubstituierte pyridazinone
WO2011045271A1 (de) 2009-10-15 2011-04-21 Bayer Cropscience Ag Herbizid wirksame heterocyclylsubstituierte pyridazinone
WO2012028582A1 (de) 2010-09-01 2012-03-08 Bayer Cropscience Ag Herbizid wirksame ketosultame und diketopyridine
CN106810550A (zh) * 2017-01-10 2017-06-09 湖南华腾制药有限公司 一种萘啶衍生物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU407902A1 (ru) * 1971-11-16 1973-12-10 Институт органической химии Украинской ССР Способ получения диэтилового эфира 3,4,5,6-тетрахлорпиридил-2-малоновой кислоты
TW258648B (pt) * 1993-03-04 1995-10-01 Shell Internat Res Schappej Bv
IL108747A (en) * 1993-03-04 1999-03-12 Shell Int Research Mushroom-killing preparations containing a history of 6 metamorphoses of 5 - 7 Dihalo - 1, 2 - 4 Triazlo [A-1,5] Pyrimidine Certain such new compounds and their preparation
EE200000706A (et) * 1998-05-26 2002-06-17 Warner-Lambert Company Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
PT1204323E (pt) * 1999-08-18 2004-11-30 Aventis Cropscience Gmbh Fungicidas
CA2413802A1 (en) * 2000-06-30 2002-01-10 Mark R. Schmitt Substituted-triazolopyrimidines as anticancer agents
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
HUP0401746A3 (en) * 2001-07-18 2008-02-28 Basf Ag Substituted 6-(2-tolyl)-triazolopyrimidines as fungicides
WO2004011467A1 (ja) * 2002-07-29 2004-02-05 Hokko Chemical Industry Co., Ltd. トリアゾロピリミジン誘導体および農園芸用殺菌剤

Also Published As

Publication number Publication date
WO2004108727A1 (de) 2004-12-16
CR8074A (es) 2007-09-11
ECSP056201A (es) 2006-04-19
CN1802379A (zh) 2006-07-12
EP1641798A1 (de) 2006-04-05
MXPA05012951A (es) 2006-02-13
CO5721005A2 (es) 2007-01-31
DE10325133A1 (de) 2004-12-23
KR20060015304A (ko) 2006-02-16
IL172098A0 (en) 2009-02-11
US20070275985A1 (en) 2007-11-29
JP2006526587A (ja) 2006-11-24
ZA200509637B (en) 2007-02-28

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 6A. E 7A. ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 6A E 7A ANUIDADES.