BRPI0507894A - pirazolopirimidinas - Google Patents

pirazolopirimidinas

Info

Publication number
BRPI0507894A
BRPI0507894A BRPI0507894-6A BRPI0507894A BRPI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A
Authority
BR
Brazil
Prior art keywords
pyrazolopyrimidines
pirazolopyrimidines
substances
formula
production
Prior art date
Application number
BRPI0507894-6A
Other languages
English (en)
Inventor
Olaf Gebauer
Herbert Gayer
Ulrich Heinemann
Stefan Herrmann
Stefan Hillebrand
Hans-Ludwid Elbe
Ronald Ebbert
Ulrike Wachendorff-Neumann
Peter Dahmen
Karl-Heinz Kuck
Mamorau Hatazawa
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0507894A publication Critical patent/BRPI0507894A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

PIRAZOLOPIRIMIDINAS. Pirazolopirimidinas da fórmula na qual R¬ 1¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, R¬ 5¬ e X têm os significados indicados na descrição, um processo para a produção dessas substâncias e seu uso para o combater de microorganismos indesejáveis.
BRPI0507894-6A 2004-02-20 2005-02-18 pirazolopirimidinas BRPI0507894A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004008807A DE102004008807A1 (de) 2004-02-20 2004-02-20 Pyrazolopyrimidine
PCT/EP2005/001694 WO2005082907A2 (de) 2004-02-20 2005-02-18 Pyrazolopyrimidine zur bekämpfung unerwünschter mikroorganismen

Publications (1)

Publication Number Publication Date
BRPI0507894A true BRPI0507894A (pt) 2007-07-24

Family

ID=34832976

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507894-6A BRPI0507894A (pt) 2004-02-20 2005-02-18 pirazolopirimidinas

Country Status (15)

Country Link
US (1) US7629294B2 (pt)
EP (1) EP1718652A2 (pt)
JP (1) JP2007524691A (pt)
KR (1) KR20070015386A (pt)
CN (1) CN1946293A (pt)
AR (1) AR048857A1 (pt)
BR (1) BRPI0507894A (pt)
CA (1) CA2556798A1 (pt)
CR (1) CR8559A (pt)
DE (1) DE102004008807A1 (pt)
EA (1) EA200601515A1 (pt)
IL (1) IL177510A0 (pt)
MX (1) MXPA06009311A (pt)
TW (1) TW200538044A (pt)
WO (1) WO2005082907A2 (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4926720B2 (ja) * 2003-12-22 2012-05-09 スミスクライン ビーチャム （コーク） リミテッド Ｃｒｆ受容体アンタゴニストおよびそれらに関連する方法
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
US8188097B2 (en) 2005-10-21 2012-05-29 Mitsubishi Tanabe Pharma Corporation Pyrazolo[1,5-A]pyrimidine compounds
JP4847275B2 (ja) * 2005-10-21 2011-12-28 田辺三菱製薬株式会社 ピラゾロ［１，５−ａ］ピリミジン化合物
AR061793A1 (es) 2006-07-05 2008-09-24 Mitsubishi Tanabe Pharma Corp Compuesto de pirazolo[1,5-a] pirimidina y composicion farmaceutica
TW201345908A (zh) * 2006-07-05 2013-11-16 Mitsubishi Tanabe Pharma Corp 吡唑并〔１，５-ａ〕嘧啶化合物
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
JP4837701B2 (ja) * 2007-04-20 2011-12-14 田辺三菱製薬株式会社 医薬組成物
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
US8507673B2 (en) * 2008-12-11 2013-08-13 Emory University Process for preparing 5,7 diaminopyrazolo [1,5-A] pyrimidine compounds
WO2014153172A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
EP2970135B1 (en) 2013-03-14 2018-07-18 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
CA2903394C (en) 2013-03-14 2021-08-31 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
US9120757B2 (en) 2013-03-14 2015-09-01 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
US9133189B2 (en) 2013-03-14 2015-09-15 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
US20160039767A1 (en) 2013-03-14 2016-02-11 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
US9394258B2 (en) 2013-03-14 2016-07-19 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
EP2970181B1 (en) 2013-03-14 2017-06-07 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
EP3363434A1 (en) 2013-03-14 2018-08-22 Epizyme Inc Arginine methyltransferase inhibitors and uses thereof
JP2016514164A (ja) 2013-03-14 2016-05-19 エピザイム，インコーポレイティド アルギニンメチルトランスフェラーゼ阻害剤としてのピラゾール誘導体およびその使用
IL317854A (en) * 2017-07-28 2025-02-01 Takeda Pharmaceuticals Co TYK2 inhibitors and their uses
JP7619951B2 (ja) * 2018-10-15 2025-01-22 武田薬品工業株式会社 Ｔｙｋ２阻害剤およびその使用

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS423174Y1 (pt) * 1964-01-17 1967-02-24
JPS423173Y1 (pt) * 1964-01-24 1967-02-24
US3515715A (en) 1967-01-23 1970-06-02 Eastman Kodak Co Quaternized pyrazolylazo dyes
US3634391A (en) 1969-07-25 1972-01-11 Eastman Kodak Co Pyrazolyl-azo-indole dyestuffs
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
FR2537137B1 (fr) 1982-12-03 1985-07-19 Roussel Uclaf Procede de preparation de derives de l'acide 2-thiophene acetique et produits intermediaires necessaires pour leur preparation
DE3338292A1 (de) * 1983-10-21 1985-05-02 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)-pyrimidine und diese enthaltende fungizide
DE3533050A1 (de) 1985-09-17 1987-03-26 Basf Ag 7-amino-azolo(1,5-a)pyrimidine, verfahren zu ihrer herstellung und diese enthaltende fungizide, bzw. deren verwendung als fungizide
GB9510459D0 (en) 1995-05-24 1995-07-19 Zeneca Ltd Bicyclic amines
FR2750048B1 (fr) * 1996-06-21 1998-08-14 Oreal Compositions de teinture des fibres keratiniques contenant des derives pyrazolo-(1, 5-a)-pyrimidine, procede de teinture, nouveaux derives pyrazolo-(1, 5-a)-pyrimidine et leur procede de preparation
GB9624611D0 (en) 1996-11-26 1997-01-15 Zeneca Ltd Bicyclic amine compounds
TW370451B (en) 1996-11-26 1999-09-21 Zeneca Ltd Bicyclic amine derivatives
US6156925A (en) 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6552026B2 (en) * 1999-06-14 2003-04-22 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
JP2001019693A (ja) * 1999-06-14 2001-01-23 American Cyanamid Co 殺菌・殺カビ性６−フェニル−ピラゾロピリミジン
AU2001223641A1 (en) * 2000-12-11 2002-06-24 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
UA76486C2 (en) 2001-07-26 2006-08-15 Basf Ag 7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi
DE10223917A1 (de) 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine
JP4564485B2 (ja) * 2003-02-28 2010-10-20 帝人ファーマ株式会社 ピラゾロ［１，５−ａ］ピリミジン誘導体
AU2004242850A1 (en) 2003-06-03 2004-12-09 Basf Aktiengesellschaft Substituted pyrazolopyrimidines, methods for the production thereof, use of the same for controlling pathogenic fungi, and agents containing said compounds
ATE388138T1 (de) * 2003-06-27 2008-03-15 Bayer Cropscience Ag Pyrazolopyrimidine

Also Published As

Publication number Publication date
TW200538044A (en) 2005-12-01
CN1946293A (zh) 2007-04-11
US7629294B2 (en) 2009-12-08
EP1718652A2 (de) 2006-11-08
AR048857A1 (es) 2006-06-07
DE102004008807A1 (de) 2005-09-08
KR20070015386A (ko) 2007-02-02
MXPA06009311A (es) 2007-03-01
JP2007524691A (ja) 2007-08-30
EA200601515A1 (ru) 2006-12-29
WO2005082907A2 (de) 2005-09-09
IL177510A0 (en) 2006-12-10
CA2556798A1 (en) 2005-09-09
US20050187224A1 (en) 2005-08-25
CR8559A (es) 2006-11-23
WO2005082907A3 (de) 2006-06-29

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.