BRPI0507894A - pirazolopirimidinas - Google Patents

pirazolopirimidinas

Info

Publication number
BRPI0507894A
BRPI0507894A BRPI0507894-6A BRPI0507894A BRPI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A BR PI0507894 A BRPI0507894 A BR PI0507894A
Authority
BR
Brazil
Prior art keywords
pyrazolopyrimidines
pirazolopyrimidines
substances
formula
production
Prior art date
Application number
BRPI0507894-6A
Other languages
English (en)
Inventor
Olaf Gebauer
Herbert Gayer
Ulrich Heinemann
Stefan Herrmann
Stefan Hillebrand
Hans-Ludwid Elbe
Ronald Ebbert
Ulrike Wachendorff-Neumann
Peter Dahmen
Karl-Heinz Kuck
Mamorau Hatazawa
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BRPI0507894A publication Critical patent/BRPI0507894A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

PIRAZOLOPIRIMIDINAS. Pirazolopirimidinas da fórmula na qual R¬ 1¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, R¬ 5¬ e X têm os significados indicados na descrição, um processo para a produção dessas substâncias e seu uso para o combater de microorganismos indesejáveis.
BRPI0507894-6A 2004-02-20 2005-02-18 pirazolopirimidinas BRPI0507894A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004008807A DE102004008807A1 (de) 2004-02-20 2004-02-20 Pyrazolopyrimidine
PCT/EP2005/001694 WO2005082907A2 (de) 2004-02-20 2005-02-18 Pyrazolopyrimidine zur bekämpfung unerwünschter mikroorganismen

Publications (1)

Publication Number Publication Date
BRPI0507894A true BRPI0507894A (pt) 2007-07-24

Family

ID=34832976

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507894-6A BRPI0507894A (pt) 2004-02-20 2005-02-18 pirazolopirimidinas

Country Status (15)

Country Link
US (1) US7629294B2 (pt)
EP (1) EP1718652A2 (pt)
JP (1) JP2007524691A (pt)
KR (1) KR20070015386A (pt)
CN (1) CN1946293A (pt)
AR (1) AR048857A1 (pt)
BR (1) BRPI0507894A (pt)
CA (1) CA2556798A1 (pt)
CR (1) CR8559A (pt)
DE (1) DE102004008807A1 (pt)
EA (1) EA200601515A1 (pt)
IL (1) IL177510A0 (pt)
MX (1) MXPA06009311A (pt)
TW (1) TW200538044A (pt)
WO (1) WO2005082907A2 (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY143499A (en) * 2003-12-22 2011-05-31 Sb Pharmco Inc Crf receptor antagonist and methods relating thereto
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
DE102005007534A1 (de) * 2005-02-17 2006-08-31 Bayer Cropscience Ag Pyrazolopyrimidine
JP4847275B2 (ja) * 2005-10-21 2011-12-28 田辺三菱製薬株式会社 ピラゾロ［１，５−ａ］ピリミジン化合物
AR056876A1 (es) 2005-10-21 2007-10-31 Tanabe Seiyaku Co Compuestos de pirazolo[1-5-a]pirimidina, antagonistas de receptores canabinoides cb1, composiciones farmaceuticas que los contienen y usos en el tratamiento de enfermedades del sistema nervioso central, tales como trastornos psicoticos, neurologicos y similares
AR061793A1 (es) 2006-07-05 2008-09-24 Mitsubishi Tanabe Pharma Corp Compuesto de pirazolo[1,5-a] pirimidina y composicion farmaceutica
TWI419889B (zh) * 2006-07-05 2013-12-21 Mitsubishi Tanabe Pharma Corp 吡唑并〔１，５-ａ〕嘧啶化合物
DE102006039255A1 (de) * 2006-08-17 2008-02-21 Bayer Cropscience Ag Insektizide heterocyclische Carbonsäurederivate
WO2008046856A2 (de) * 2006-10-18 2008-04-24 Basf Se Fungizide zusammensetzungen
JP4837701B2 (ja) * 2007-04-20 2011-12-14 田辺三菱製薬株式会社 医薬組成物
EP2014661A1 (de) * 2007-06-13 2009-01-14 Bayer CropScience AG Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate
US8507673B2 (en) * 2008-12-11 2013-08-13 Emory University Process for preparing 5,7 diaminopyrazolo [1,5-A] pyrimidine compounds
WO2014153208A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
JP2016518336A (ja) 2013-03-14 2016-06-23 エピザイム，インコーポレイティド Ｐｒｍｔ１阻害剤としてのピラゾール誘導体およびその使用
US9120757B2 (en) 2013-03-14 2015-09-01 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
EP2970135B1 (en) 2013-03-14 2018-07-18 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
US9765035B2 (en) 2013-03-14 2017-09-19 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
KR102028793B1 (ko) 2013-03-14 2019-10-07 에피자임, 인코포레이티드 아르기닌 메틸기 전이효소 억제제 및 이의 용도
WO2014153214A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyl transferase inhibtors and uses thereof
EP2970137A1 (en) 2013-03-14 2016-01-20 Epizyme, Inc. Pyrazole derivatives as arginine methyltransferase inhibitors and uses thereof
WO2014153100A2 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Arginine methyltransferase inhibitors and uses thereof
WO2014153172A1 (en) 2013-03-14 2014-09-25 Epizyme, Inc. Pyrazole derivatives as prmt1 inhibitors and uses thereof
SI3658557T1 (sl) * 2017-07-28 2024-10-30 Takeda Pharmaceutical Company Limited Zaviralci TYK2 in njihova uporaba
CN113271940A (zh) * 2018-10-15 2021-08-17 林伯士拉克许米公司 Tyk2抑制剂和其用途

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS423174Y1 (pt) * 1964-01-17 1967-02-24
JPS423173Y1 (pt) * 1964-01-24 1967-02-24
US3515715A (en) 1967-01-23 1970-06-02 Eastman Kodak Co Quaternized pyrazolylazo dyes
US3634391A (en) 1969-07-25 1972-01-11 Eastman Kodak Co Pyrazolyl-azo-indole dyestuffs
DE3130633A1 (de) 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
FR2537137B1 (fr) 1982-12-03 1985-07-19 Roussel Uclaf Procede de preparation de derives de l'acide 2-thiophene acetique et produits intermediaires necessaires pour leur preparation
DE3338292A1 (de) 1983-10-21 1985-05-02 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)-pyrimidine und diese enthaltende fungizide
DE3533050A1 (de) 1985-09-17 1987-03-26 Basf Ag 7-amino-azolo(1,5-a)pyrimidine, verfahren zu ihrer herstellung und diese enthaltende fungizide, bzw. deren verwendung als fungizide
GB9510459D0 (en) 1995-05-24 1995-07-19 Zeneca Ltd Bicyclic amines
FR2750048B1 (fr) * 1996-06-21 1998-08-14 Oreal Compositions de teinture des fibres keratiniques contenant des derives pyrazolo-(1, 5-a)-pyrimidine, procede de teinture, nouveaux derives pyrazolo-(1, 5-a)-pyrimidine et leur procede de preparation
CA2271749A1 (en) 1996-11-26 1998-06-18 Christopher Richard Ayles Godfrey 8-azabicyclo¬3.2.1|octane-, 8-azabicyclo¬3.2.1|oct-6-ene-, 9-azabicyclo¬3.3.1|nonane-, 9-aza-3-oxabicyclo¬3.3.1|nonane- and 9-aza-3-thiabicyclo¬3.3.1|nonane derivatives, their preparation and their use as insecticides
GB9624611D0 (en) 1996-11-26 1997-01-15 Zeneca Ltd Bicyclic amine compounds
US6156925A (en) 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
JP2001019693A (ja) * 1999-06-14 2001-01-23 American Cyanamid Co 殺菌・殺カビ性６−フェニル−ピラゾロピリミジン
US6552026B2 (en) * 1999-06-14 2003-04-22 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
WO2002048151A1 (en) * 2000-12-11 2002-06-20 Basf Aktiengesellschaft 6-phenyl-pyrazolopyrimidines
DK1414302T3 (da) 2001-07-26 2007-06-18 Basf Ag 7-aminotriazolopyrimidiner til bekæmpelse af skadelige svampe
DE10223917A1 (de) * 2002-05-29 2003-12-11 Bayer Cropscience Ag Pyrazolopyrimidine
US7557110B2 (en) * 2003-02-28 2009-07-07 Teijin Pharma Limited Pyrazolo[1,5-A] pyrimidine derivatives
BRPI0410610A (pt) 2003-06-03 2006-07-04 Basf Ag compostos, processos para a produção dos mesmos e para o combate de fungos nocivos fitopatogênicos, produtos intermediários, e, agente adequado para o combate de fungos nocivos
ATE388138T1 (de) * 2003-06-27 2008-03-15 Bayer Cropscience Ag Pyrazolopyrimidine

Also Published As

Publication number Publication date
DE102004008807A1 (de) 2005-09-08
US7629294B2 (en) 2009-12-08
IL177510A0 (en) 2006-12-10
CA2556798A1 (en) 2005-09-09
JP2007524691A (ja) 2007-08-30
AR048857A1 (es) 2006-06-07
TW200538044A (en) 2005-12-01
EP1718652A2 (de) 2006-11-08
EA200601515A1 (ru) 2006-12-29
US20050187224A1 (en) 2005-08-25
CR8559A (es) 2006-11-23
KR20070015386A (ko) 2007-02-02
WO2005082907A2 (de) 2005-09-09
WO2005082907A3 (de) 2006-06-29
MXPA06009311A (es) 2007-03-01
CN1946293A (zh) 2007-04-11

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.