BRPI0418166A - compostos de bicicloeteroarilamina como ligandos de canal de ìon e usos destes - Google Patents

compostos de bicicloeteroarilamina como ligandos de canal de ìon e usos destes

Info

Publication number
BRPI0418166A
BRPI0418166A BRPI0418166-2A BRPI0418166A BRPI0418166A BR PI0418166 A BRPI0418166 A BR PI0418166A BR PI0418166 A BRPI0418166 A BR PI0418166A BR PI0418166 A BRPI0418166 A BR PI0418166A
Authority
BR
Brazil
Prior art keywords
compounds
ion channel
bicycloetheroylamine
channel ligands
ligands
Prior art date
Application number
BRPI0418166-2A
Other languages
English (en)
Inventor
Michael G Kelly
Satyanarayana Janagani
Guoxian Wu
John Kincaid
David Lonergan
Yunfeng Fang
Zhi-Liang Wei
Original Assignee
Renovis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Renovis Inc filed Critical Renovis Inc
Publication of BRPI0418166A publication Critical patent/BRPI0418166A/pt

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Abstract

COMPOSTOS DE BICICLOETEROARILAMINA COMO LIGANDOS DE CANAL DE ìON E USOS DESTES. A presente invenção refere-se a compostos de amina que têm uma fórmula representada pela seguinte: Os compostos podem ser preparados como composições farmacêuticas e podem ser empregados para a prevenção e tratamento de uma veriedade de condições em mamíferos incluindo seres humanos, incluindo por meio de exemplos não limitantes,dor, inflamação, lesão traumática e outros.
BRPI0418166-2A 2003-12-24 2004-12-23 compostos de bicicloeteroarilamina como ligandos de canal de ìon e usos destes BRPI0418166A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53237103P 2003-12-24 2003-12-24
PCT/US2004/043456 WO2005066171A1 (en) 2003-12-24 2004-12-23 Bicycloheteroarylamine compounds as ion channel ligands and uses thereof

Publications (1)

Publication Number Publication Date
BRPI0418166A true BRPI0418166A (pt) 2007-06-19

Family

ID=34748796

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0418166-2A BRPI0418166A (pt) 2003-12-24 2004-12-23 compostos de bicicloeteroarilamina como ligandos de canal de ìon e usos destes

Country Status (8)

Country Link
US (1) US7414131B2 (pt)
EP (1) EP1697361A1 (pt)
JP (1) JP2007517045A (pt)
AR (1) AR051156A1 (pt)
BR (1) BRPI0418166A (pt)
CA (1) CA2550717A1 (pt)
TW (1) TW200530235A (pt)
WO (1) WO2005066171A1 (pt)

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EP1697361A1 (en) 2006-09-06
TW200530235A (en) 2005-09-16
US7414131B2 (en) 2008-08-19
WO2005066171A1 (en) 2005-07-21
AR051156A1 (es) 2006-12-27

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