BRPI0511954A - métodos de produção de um derivado de acetamidopirrolidina ou um sal do mesmo, de um derivado de ácido benzamidoacético ou sal do mesmo, e de um derivado de ácido 2-nitrobenzóico ou um sal do mesmo, e, composto ou um sal do mesmo - Google Patents

métodos de produção de um derivado de acetamidopirrolidina ou um sal do mesmo, de um derivado de ácido benzamidoacético ou sal do mesmo, e de um derivado de ácido 2-nitrobenzóico ou um sal do mesmo, e, composto ou um sal do mesmo

Info

Publication number
BRPI0511954A
BRPI0511954A BRPI0511954-5A BRPI0511954A BRPI0511954A BR PI0511954 A BRPI0511954 A BR PI0511954A BR PI0511954 A BRPI0511954 A BR PI0511954A BR PI0511954 A BRPI0511954 A BR PI0511954A
Authority
BR
Brazil
Prior art keywords
salt
derivative
acid derivative
producing
methods
Prior art date
Application number
BRPI0511954-5A
Other languages
English (en)
Inventor
Asahi Kawana
Takumi Takeyasu
Atsuo Hazato
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of BRPI0511954A publication Critical patent/BRPI0511954A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)

Abstract

MéTODOS DE PRODUçãO DE UM DERIVADO DE ACETAMIDOPIRROLIDINA OU UM SAL DO MESMO, DE UM DERIVADO DE áCIDO BENZAMIDOACéTICO OU UM SAL DO MESMO, E DE UM DERIVADO DE áCIDO 2-NITROBENZóICO OU UM SAL DO MESMO, E, COMPOSTO OU UM SAL DO MESMO. é apresentado um método para a produção de um derivado de acetamidopirrolodina ou um sal do mesmo que compreende um processo de reação expresso pelas fórmulas que seguem. Nas fórmulas R representa um átomo de hidrogênio ou um grupo alquila C~ 1~-C~ 6~; R¬ 13¬, R¬ 14¬, R¬ 15¬ e R¬ 16¬ independentemente representam um átomo de hidrogênio, um átomo de halogênio, um grupo alquila C~ 1~-C~ 6~, um grupo alcóxi C~ 1~-C~ 6~, um grupo hidróxi, um grupo alquila halogenado C~ 1~-C~ 6~ ou um grupo alcóxi halogenado C~ 1~-C~ 6~; e R¬ 21¬ representa um grupo de proteção de éster.
BRPI0511954-5A 2004-06-14 2005-06-13 métodos de produção de um derivado de acetamidopirrolidina ou um sal do mesmo, de um derivado de ácido benzamidoacético ou sal do mesmo, e de um derivado de ácido 2-nitrobenzóico ou um sal do mesmo, e, composto ou um sal do mesmo BRPI0511954A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2004175158 2004-06-14
JP2004175159 2004-06-14
PCT/JP2005/011187 WO2005121081A1 (ja) 2004-06-14 2005-06-13 アセトアミドピロリジン誘導体の製造方法およびその中間体化合物

Publications (1)

Publication Number Publication Date
BRPI0511954A true BRPI0511954A (pt) 2008-01-22

Family

ID=35502991

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0511954-5A BRPI0511954A (pt) 2004-06-14 2005-06-13 métodos de produção de um derivado de acetamidopirrolidina ou um sal do mesmo, de um derivado de ácido benzamidoacético ou sal do mesmo, e de um derivado de ácido 2-nitrobenzóico ou um sal do mesmo, e, composto ou um sal do mesmo

Country Status (12)

Country Link
US (1) US20070249847A1 (pt)
EP (1) EP1760075A4 (pt)
JP (1) JPWO2005121081A1 (pt)
KR (1) KR20070043770A (pt)
AU (1) AU2005252112A1 (pt)
BR (1) BRPI0511954A (pt)
CA (1) CA2570179A1 (pt)
IL (1) IL179724A0 (pt)
MX (1) MXPA06014262A (pt)
SG (1) SG136139A1 (pt)
TW (1) TW200604141A (pt)
WO (1) WO2005121081A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR053046A1 (es) * 2005-04-07 2007-04-18 Teijin Pharma Ltd Cristal de derivado de aminonopirrolidina y metodo de produccion del mismo

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK285729B6 (sk) * 1997-11-18 2007-07-06 Teijin Pharma Limited Zlúčenina derivátov cyklických amínov a jej použitie
CA2373942A1 (en) * 1999-05-18 2000-11-23 Teijin Limited Remedies or prophylactis for diseases in association with chemokines
CA2378499A1 (en) * 1999-08-04 2001-02-15 Teijin Limited Cyclic amine ccr3 antagonists
US6410566B1 (en) * 2000-05-16 2002-06-25 Teijin Limited Cyclic amine derivatives and their use as drugs

Also Published As

Publication number Publication date
SG136139A1 (en) 2007-10-29
CA2570179A1 (en) 2005-12-22
MXPA06014262A (es) 2007-03-12
WO2005121081A1 (ja) 2005-12-22
IL179724A0 (en) 2007-05-15
US20070249847A1 (en) 2007-10-25
AU2005252112A1 (en) 2005-12-22
EP1760075A1 (en) 2007-03-07
EP1760075A4 (en) 2009-10-28
JPWO2005121081A1 (ja) 2008-04-10
KR20070043770A (ko) 2007-04-25
TW200604141A (en) 2006-02-01

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.