BRPI0513453A - processo para a preparação de compostos, e composto - Google Patents
processo para a preparação de compostos, e compostoInfo
- Publication number
- BRPI0513453A BRPI0513453A BRPI0513453-6A BRPI0513453A BRPI0513453A BR PI0513453 A BRPI0513453 A BR PI0513453A BR PI0513453 A BRPI0513453 A BR PI0513453A BR PI0513453 A BRPI0513453 A BR PI0513453A
- Authority
- BR
- Brazil
- Prior art keywords
- variables
- compounds
- compound
- preparation
- formula
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 abstract 2
- 230000000269 nucleophilic effect Effects 0.000 abstract 2
- 150000004657 carbamic acid derivatives Chemical class 0.000 abstract 1
- 150000002081 enamines Chemical class 0.000 abstract 1
- 239000013067 intermediate product Substances 0.000 abstract 1
- 125000000446 sulfanediyl group Chemical group *S* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCESSO PARA A PREPARAçãO DE COMPOSTOS, E COMPOSTO A invenção refere-se a um processo para a produção de 3-fenil (tio) uracilas e -ditiuracilas de fórmula I, em que as variáveis têm os significados citados no relatório descritivo, caracterizado pelo fato de que carbamatos de fórmula II, em que as variáveis X¬ 1¬, X¬ 3¬, Ar e A têm os significados mencionados acima e L representa um nucleófugo que pode ser deslocado nucleofilicamente, pode ser reagido com enaminas de fórmula III, em que as variáveis X¬ 2¬, R¬ 1¬, R¬ 2¬ e R¬ 3¬ têm os significados mencionados acima e L representa um nucleófugo que pode ser deslocado nucleofilicamente. A invenção também se refere a produtos intermediários para a produção das mesmas.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004035656.4 | 2004-07-22 | ||
| DE102004035656 | 2004-07-22 | ||
| PCT/EP2005/007577 WO2006010474A1 (de) | 2004-07-22 | 2005-07-13 | Verfahren zur herstellung von 3-phenyl(thio)uracilen und - dithiouracilen |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0513453A true BRPI0513453A (pt) | 2008-05-06 |
| BRPI0513453B1 BRPI0513453B1 (pt) | 2014-12-30 |
Family
ID=34972926
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0513453-6A BRPI0513453B1 (pt) | 2004-07-22 | 2005-07-13 | Processo para a preparação de compostos, e composto |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US8252925B2 (pt) |
| EP (1) | EP1773787B1 (pt) |
| JP (2) | JP4860613B2 (pt) |
| KR (1) | KR101238470B1 (pt) |
| CN (1) | CN1989111B (pt) |
| AR (1) | AR050005A1 (pt) |
| AU (1) | AU2005266622B8 (pt) |
| BR (1) | BRPI0513453B1 (pt) |
| CA (1) | CA2574406C (pt) |
| DK (1) | DK1773787T3 (pt) |
| EA (1) | EA012035B1 (pt) |
| ES (1) | ES2465499T3 (pt) |
| IL (1) | IL180180A (pt) |
| MX (1) | MX2007000067A (pt) |
| PL (1) | PL1773787T3 (pt) |
| SI (1) | SI1773787T1 (pt) |
| UA (1) | UA83764C2 (pt) |
| WO (1) | WO2006010474A1 (pt) |
| ZA (1) | ZA200701464B (pt) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8252925B2 (en) * | 2004-07-22 | 2012-08-28 | Basf Aktiengesellschaft | Method for the production of 3-phenyl(thio)uracils and dithiouracils |
| EA200801432A1 (ru) * | 2005-12-01 | 2008-12-30 | Басф Се | Способ получения сульфонамидов |
| AR063306A1 (es) * | 2006-10-13 | 2009-01-21 | Basf Ag | Forma cristalina de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluorometil)-1-(2h)-pirimidinil]-4-fluoro-n-[[metil(1-metiletil)amino]sulfonil]benzamida |
| MY149140A (en) * | 2006-10-13 | 2013-07-15 | Basf Se | Hydrates of 2-chloro 5-y3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoro-methyl)-1-(2h)-pyrimidinyl"-4-fluoro-n- yymethyl-(1-methylethyl)-amino"sulphonyl"benzamide |
| CN101821233B (zh) * | 2007-10-12 | 2016-06-29 | 巴斯夫欧洲公司 | 生产磺酸二酰胺的方法 |
| CN103130727B (zh) * | 2013-02-27 | 2015-07-08 | 江苏省农用激素工程技术研究中心有限公司 | 苯嘧磺草胺中间体的制备方法 |
| CA3210637A1 (en) | 2021-03-04 | 2022-09-09 | Michael Grabarnick | Solid forms of saflufenacil-sodium and saflufenacil-potassium, process of preparation and use thereof |
| BR112023019613A2 (pt) | 2021-03-26 | 2023-11-14 | Adama Agan Ltd | Preparação de ácido 2-cloro-4-fluoro-5-nitrobenzoico |
| CN115246791B (zh) * | 2021-04-26 | 2024-11-05 | 内蒙古世杰化工有限公司 | 一种合成6-三氟甲基尿嘧啶的方法及其中间体 |
| WO2023017518A1 (en) | 2021-08-09 | 2023-02-16 | Adama Agan Ltd. | A new process of saflufenacil production using novel intermediates |
| CN114478326B (zh) * | 2022-01-21 | 2023-10-03 | 安徽宁亿泰科技有限公司 | 一种苯嘧磺草胺关键中间体的合成方法 |
| WO2023198484A1 (en) | 2022-04-12 | 2023-10-19 | BASF Agro B.V. | Improved process for recovering n,n-dimethylformamide (dmf) from an aqueous process stream |
| EP4306508A1 (en) | 2022-07-14 | 2024-01-17 | BASF Agro B.V. | Improved process for recovering n,n-dimethylformamide (dmf) from an aqueous process stream |
| AR130348A1 (es) | 2022-08-31 | 2024-11-27 | Adama Agan Ltd | Preparación de ácido 2-cloro-4-fluoro-5-nitrobenzoico |
| WO2025124942A1 (en) | 2023-12-12 | 2025-06-19 | BASF Agro B.V. | Process for preparing a saflufenacil intermediate |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1989002891A1 (fr) | 1987-09-23 | 1989-04-06 | F. Hoffmann-La Roche & Co. Aktiengesellschaft | Composes heterocycliques |
| DE19632005A1 (de) | 1996-08-08 | 1998-02-12 | Bayer Ag | Substituierte p-Trifluormethylphenyluracile |
| DE19755926A1 (de) | 1997-12-17 | 1999-06-24 | Basf Ag | Herbizide 3-(Benzazol-4-yl)pyrimidindion-Derivate |
| HU229494B1 (en) * | 2000-05-04 | 2014-01-28 | Basf Ag | Uracil substituted phenyl sulfamoyl carboxamides |
| AU2003240656A1 (en) * | 2002-05-16 | 2003-12-02 | Basf Aktiengesellschaft | Method for the production of sulphamic acid halogenides |
| KR101055954B1 (ko) * | 2002-10-30 | 2011-08-09 | 바스프 에스이 | 이관능성 페닐이소(티오)시아네이트, 그의 제조 방법 및그의 제조를 위한 중간체 생성물 |
| ITMI20022758A1 (it) | 2002-12-23 | 2004-06-24 | Isagro Ricerca Srl | Nuovi uracili ad attivita' erbicida. |
| US8252925B2 (en) * | 2004-07-22 | 2012-08-28 | Basf Aktiengesellschaft | Method for the production of 3-phenyl(thio)uracils and dithiouracils |
-
2005
- 2005-07-13 US US11/631,972 patent/US8252925B2/en active Active
- 2005-07-13 PL PL05763570T patent/PL1773787T3/pl unknown
- 2005-07-13 KR KR1020077004099A patent/KR101238470B1/ko not_active Expired - Lifetime
- 2005-07-13 WO PCT/EP2005/007577 patent/WO2006010474A1/de not_active Ceased
- 2005-07-13 AU AU2005266622A patent/AU2005266622B8/en not_active Expired
- 2005-07-13 MX MX2007000067A patent/MX2007000067A/es active IP Right Grant
- 2005-07-13 CN CN200580024680XA patent/CN1989111B/zh not_active Expired - Lifetime
- 2005-07-13 SI SI200531847T patent/SI1773787T1/sl unknown
- 2005-07-13 BR BRPI0513453-6A patent/BRPI0513453B1/pt active IP Right Grant
- 2005-07-13 JP JP2007521854A patent/JP4860613B2/ja not_active Expired - Lifetime
- 2005-07-13 EP EP05763570.8A patent/EP1773787B1/de not_active Expired - Lifetime
- 2005-07-13 UA UAA200701779A patent/UA83764C2/ru unknown
- 2005-07-13 EA EA200700289A patent/EA012035B1/ru not_active IP Right Cessation
- 2005-07-13 DK DK05763570.8T patent/DK1773787T3/da active
- 2005-07-13 CA CA2574406A patent/CA2574406C/en not_active Expired - Lifetime
- 2005-07-13 ES ES05763570.8T patent/ES2465499T3/es not_active Expired - Lifetime
- 2005-07-21 AR ARP050103026A patent/AR050005A1/es active IP Right Grant
-
2006
- 2006-12-19 IL IL180180A patent/IL180180A/en active IP Right Grant
-
2007
- 2007-02-20 ZA ZA200701464A patent/ZA200701464B/xx unknown
-
2011
- 2011-03-04 US US13/040,292 patent/US8124818B2/en not_active Expired - Lifetime
- 2011-07-22 JP JP2011160861A patent/JP2012006936A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AR050005A1 (es) | 2006-09-20 |
| EA012035B1 (ru) | 2009-06-30 |
| MX2007000067A (es) | 2007-03-28 |
| SI1773787T1 (sl) | 2014-05-30 |
| IL180180A0 (en) | 2007-06-03 |
| KR101238470B1 (ko) | 2013-03-04 |
| PL1773787T3 (pl) | 2014-09-30 |
| JP2012006936A (ja) | 2012-01-12 |
| EP1773787B1 (de) | 2014-04-02 |
| US20080033174A1 (en) | 2008-02-07 |
| CA2574406C (en) | 2013-02-19 |
| DK1773787T3 (da) | 2014-06-23 |
| ZA200701464B (en) | 2009-03-25 |
| CN1989111A (zh) | 2007-06-27 |
| JP4860613B2 (ja) | 2012-01-25 |
| EA200700289A1 (ru) | 2007-08-31 |
| CN1989111B (zh) | 2012-12-05 |
| US8124818B2 (en) | 2012-02-28 |
| AU2005266622A1 (en) | 2006-02-02 |
| US8252925B2 (en) | 2012-08-28 |
| UA83764C2 (ru) | 2008-08-11 |
| JP2008506733A (ja) | 2008-03-06 |
| AU2005266622B8 (en) | 2011-05-19 |
| KR20070034127A (ko) | 2007-03-27 |
| WO2006010474A1 (de) | 2006-02-02 |
| ES2465499T3 (es) | 2014-06-05 |
| EP1773787A1 (de) | 2007-04-18 |
| BRPI0513453B1 (pt) | 2014-12-30 |
| US20110152522A1 (en) | 2011-06-23 |
| AU2005266622B2 (en) | 2011-03-31 |
| IL180180A (en) | 2011-09-27 |
| CA2574406A1 (en) | 2006-02-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B25D | Requested change of name of applicant approved |
Owner name: BASF SE (DE) |
|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 13/07/2005, OBSERVADAS AS CONDICOES LEGAIS. |