BRPI0607894A2 - utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais - Google Patents
utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renaisInfo
- Publication number
- BRPI0607894A2 BRPI0607894A2 BRPI0607894-0A BRPI0607894A BRPI0607894A2 BR PI0607894 A2 BRPI0607894 A2 BR PI0607894A2 BR PI0607894 A BRPI0607894 A BR PI0607894A BR PI0607894 A2 BRPI0607894 A2 BR PI0607894A2
- Authority
- BR
- Brazil
- Prior art keywords
- prevention
- preparation
- treatment
- kidney disease
- medicinal products
- Prior art date
Links
- 230000002265 prevention Effects 0.000 title abstract 3
- 208000017169 kidney disease Diseases 0.000 title abstract 2
- 229940126601 medicinal product Drugs 0.000 title abstract 2
- 150000003217 pyrazoles Chemical class 0.000 title 1
- 229940123158 Cannabinoid CB1 receptor antagonist Drugs 0.000 abstract 1
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000003555 cannabinoid 1 receptor antagonist Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
UTILIZAçãO DE UM DERIVADO DE PIRAZOL PARA A PREPARAçãO DE MEDICAMENTOS úTEIS NA PREVENçãO E NO TRATAMENTO DAS DOENçAS RENAIS. A presente invenção refere-se a utilização de um composto antagonista dos receptores CB1 aos canabinóides, sozinho ou associado a um outro princípio ativo, derivado do pirazol, para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0501919A FR2882262B1 (fr) | 2005-02-23 | 2005-02-23 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales |
| FR0504798A FR2882263B1 (fr) | 2005-02-23 | 2005-05-12 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales |
| PCT/FR2006/000369 WO2006090047A1 (fr) | 2005-02-23 | 2006-02-17 | Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0607894A2 true BRPI0607894A2 (pt) | 2009-10-20 |
Family
ID=36603585
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0607894-0A BRPI0607894A2 (pt) | 2005-02-23 | 2006-02-17 | utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7622488B2 (pt) |
| EP (1) | EP1855675A1 (pt) |
| JP (1) | JP2008531526A (pt) |
| KR (1) | KR20070104916A (pt) |
| AR (1) | AR054003A1 (pt) |
| AU (1) | AU2006217794A1 (pt) |
| BR (1) | BRPI0607894A2 (pt) |
| CA (1) | CA2597802A1 (pt) |
| CR (1) | CR9270A (pt) |
| EA (1) | EA011655B1 (pt) |
| FR (1) | FR2882263B1 (pt) |
| IL (1) | IL185165A0 (pt) |
| MA (1) | MA29263B1 (pt) |
| MX (1) | MX2007009995A (pt) |
| NO (1) | NO20074768L (pt) |
| TN (1) | TNSN07291A1 (pt) |
| TW (1) | TW200640458A (pt) |
| WO (1) | WO2006090047A1 (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010079241A1 (es) | 2009-01-12 | 2010-07-15 | Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion | Uso de antagonistas y/o agonistas inversos de los receptores cb1 para la preparación de medicamentos que incrementen la excitabilidad de las motoneuronas |
| FR2958850B1 (fr) * | 2010-04-14 | 2012-07-06 | Centre Nat Rech Scient | Medicaments pour la prevention ou le traitement des addictions aux drogues |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2692575B1 (fr) * | 1992-06-23 | 1995-06-30 | Sanofi Elf | Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant. |
| FR2713225B1 (fr) * | 1993-12-02 | 1996-03-01 | Sanofi Sa | N-pipéridino-3-pyrazolecarboxamide substitué. |
| FR2789079B3 (fr) | 1999-02-01 | 2001-03-02 | Sanofi Synthelabo | Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant |
| US20040122033A1 (en) * | 2002-12-10 | 2004-06-24 | Nargund Ravi P. | Combination therapy for the treatment of obesity |
| US20040214804A1 (en) * | 2003-04-25 | 2004-10-28 | Pharmacia Corporation | Combination of an aldosterone receptor antagonist and an anti-obesity agent |
| AR051446A1 (es) * | 2004-09-23 | 2007-01-17 | Bristol Myers Squibb Co | Glucosidos de c-arilo como inhibidores selectivos de transportadores de glucosa (sglt2) |
-
2005
- 2005-05-12 FR FR0504798A patent/FR2882263B1/fr not_active Expired - Fee Related
-
2006
- 2006-02-17 KR KR1020077019170A patent/KR20070104916A/ko not_active Withdrawn
- 2006-02-17 CA CA002597802A patent/CA2597802A1/fr not_active Abandoned
- 2006-02-17 EP EP06709339A patent/EP1855675A1/fr not_active Withdrawn
- 2006-02-17 AU AU2006217794A patent/AU2006217794A1/en not_active Abandoned
- 2006-02-17 JP JP2007556630A patent/JP2008531526A/ja not_active Withdrawn
- 2006-02-17 BR BRPI0607894-0A patent/BRPI0607894A2/pt not_active IP Right Cessation
- 2006-02-17 EA EA200701800A patent/EA011655B1/ru not_active IP Right Cessation
- 2006-02-17 MX MX2007009995A patent/MX2007009995A/es active IP Right Grant
- 2006-02-17 WO PCT/FR2006/000369 patent/WO2006090047A1/fr not_active Ceased
- 2006-02-21 AR ARP060100612A patent/AR054003A1/es unknown
- 2006-02-22 TW TW095105981A patent/TW200640458A/zh unknown
-
2007
- 2007-07-20 CR CR9270A patent/CR9270A/es not_active Application Discontinuation
- 2007-07-24 TN TNP2007000291A patent/TNSN07291A1/en unknown
- 2007-08-02 US US11/832,861 patent/US7622488B2/en not_active Expired - Fee Related
- 2007-08-09 IL IL185165A patent/IL185165A0/en unknown
- 2007-08-23 MA MA30159A patent/MA29263B1/fr unknown
- 2007-09-18 NO NO20074768A patent/NO20074768L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2882263A1 (fr) | 2006-08-25 |
| MA29263B1 (fr) | 2008-02-01 |
| US7622488B2 (en) | 2009-11-24 |
| AR054003A1 (es) | 2007-05-30 |
| CR9270A (es) | 2007-10-01 |
| EP1855675A1 (fr) | 2007-11-21 |
| CA2597802A1 (fr) | 2006-08-31 |
| TNSN07291A1 (en) | 2008-12-31 |
| TW200640458A (en) | 2006-12-01 |
| AU2006217794A1 (en) | 2006-08-31 |
| MX2007009995A (es) | 2007-10-10 |
| JP2008531526A (ja) | 2008-08-14 |
| NO20074768L (no) | 2007-11-23 |
| EA200701800A1 (ru) | 2008-02-28 |
| EA011655B1 (ru) | 2009-04-28 |
| WO2006090047A1 (fr) | 2006-08-31 |
| KR20070104916A (ko) | 2007-10-29 |
| US20080015228A1 (en) | 2008-01-17 |
| IL185165A0 (en) | 2008-06-05 |
| FR2882263B1 (fr) | 2007-04-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A E 6A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012. |