BRPI0607894A2 - utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais - Google Patents

utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais

Info

Publication number
BRPI0607894A2
BRPI0607894A2 BRPI0607894-0A BRPI0607894A BRPI0607894A2 BR PI0607894 A2 BRPI0607894 A2 BR PI0607894A2 BR PI0607894 A BRPI0607894 A BR PI0607894A BR PI0607894 A2 BRPI0607894 A2 BR PI0607894A2
Authority
BR
Brazil
Prior art keywords
prevention
preparation
treatment
kidney disease
medicinal products
Prior art date
Application number
BRPI0607894-0A
Other languages
English (en)
Inventor
Mohammed Bensaid
Jean-Marc Herbert
Philip Janiak
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR0501919A external-priority patent/FR2882262B1/fr
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of BRPI0607894A2 publication Critical patent/BRPI0607894A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

UTILIZAçãO DE UM DERIVADO DE PIRAZOL PARA A PREPARAçãO DE MEDICAMENTOS úTEIS NA PREVENçãO E NO TRATAMENTO DAS DOENçAS RENAIS. A presente invenção refere-se a utilização de um composto antagonista dos receptores CB1 aos canabinóides, sozinho ou associado a um outro princípio ativo, derivado do pirazol, para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais.
BRPI0607894-0A 2005-02-23 2006-02-17 utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais BRPI0607894A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0501919A FR2882262B1 (fr) 2005-02-23 2005-02-23 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
FR0504798A FR2882263B1 (fr) 2005-02-23 2005-05-12 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
PCT/FR2006/000369 WO2006090047A1 (fr) 2005-02-23 2006-02-17 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales

Publications (1)

Publication Number Publication Date
BRPI0607894A2 true BRPI0607894A2 (pt) 2009-10-20

Family

ID=36603585

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607894-0A BRPI0607894A2 (pt) 2005-02-23 2006-02-17 utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais

Country Status (18)

Country Link
US (1) US7622488B2 (pt)
EP (1) EP1855675A1 (pt)
JP (1) JP2008531526A (pt)
KR (1) KR20070104916A (pt)
AR (1) AR054003A1 (pt)
AU (1) AU2006217794A1 (pt)
BR (1) BRPI0607894A2 (pt)
CA (1) CA2597802A1 (pt)
CR (1) CR9270A (pt)
EA (1) EA011655B1 (pt)
FR (1) FR2882263B1 (pt)
IL (1) IL185165A0 (pt)
MA (1) MA29263B1 (pt)
MX (1) MX2007009995A (pt)
NO (1) NO20074768L (pt)
TN (1) TNSN07291A1 (pt)
TW (1) TW200640458A (pt)
WO (1) WO2006090047A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010079241A1 (es) 2009-01-12 2010-07-15 Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion Uso de antagonistas y/o agonistas inversos de los receptores cb1 para la preparación de medicamentos que incrementen la excitabilidad de las motoneuronas
FR2958850B1 (fr) * 2010-04-14 2012-07-06 Centre Nat Rech Scient Medicaments pour la prevention ou le traitement des addictions aux drogues

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2789079B3 (fr) 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
US20040122033A1 (en) * 2002-12-10 2004-06-24 Nargund Ravi P. Combination therapy for the treatment of obesity
US20040214804A1 (en) * 2003-04-25 2004-10-28 Pharmacia Corporation Combination of an aldosterone receptor antagonist and an anti-obesity agent
AR051446A1 (es) * 2004-09-23 2007-01-17 Bristol Myers Squibb Co Glucosidos de c-arilo como inhibidores selectivos de transportadores de glucosa (sglt2)

Also Published As

Publication number Publication date
FR2882263A1 (fr) 2006-08-25
MA29263B1 (fr) 2008-02-01
US7622488B2 (en) 2009-11-24
AR054003A1 (es) 2007-05-30
CR9270A (es) 2007-10-01
EP1855675A1 (fr) 2007-11-21
CA2597802A1 (fr) 2006-08-31
TNSN07291A1 (en) 2008-12-31
TW200640458A (en) 2006-12-01
AU2006217794A1 (en) 2006-08-31
MX2007009995A (es) 2007-10-10
JP2008531526A (ja) 2008-08-14
NO20074768L (no) 2007-11-23
EA200701800A1 (ru) 2008-02-28
EA011655B1 (ru) 2009-04-28
WO2006090047A1 (fr) 2006-08-31
KR20070104916A (ko) 2007-10-29
US20080015228A1 (en) 2008-01-17
IL185165A0 (en) 2008-06-05
FR2882263B1 (fr) 2007-04-06

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012.