BRPI0611720A2 - "composto, composição, e, métodos de inibir a fertilidade,de evitar a concepção, e de bloquear o desenvolvimento folicular mediado por fsh em um mamífero" - Google Patents

"composto, composição, e, métodos de inibir a fertilidade,de evitar a concepção, e de bloquear o desenvolvimento folicular mediado por fsh em um mamífero"

Info

Publication number
BRPI0611720A2
BRPI0611720A2 BRPI0611720A BRPI0611720A BRPI0611720A2 BR PI0611720 A2 BRPI0611720 A2 BR PI0611720A2 BR PI0611720 A BRPI0611720 A BR PI0611720A BR PI0611720 A BRPI0611720 A BR PI0611720A BR PI0611720 A2 BRPI0611720 A2 BR PI0611720A2
Authority
BR
Brazil
Prior art keywords
mammal
compound
composition
methods
follicular development
Prior art date
Application number
BRPI0611720A
Other languages
English (en)
Inventor
Arthur A Santilli
Amedeo A Failli
Dominick A Quagliato
Emily S Chen
Eugene J Trybulski
Gavin Heffernan
Patrick M Andrae
Richard Coghlan
Susan C Croce
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of BRPI0611720A2 publication Critical patent/BRPI0611720A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Gynecology & Obstetrics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI0611720A 2005-06-09 2006-06-08 "composto, composição, e, métodos de inibir a fertilidade,de evitar a concepção, e de bloquear o desenvolvimento folicular mediado por fsh em um mamífero" BRPI0611720A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68898805P 2005-06-09 2005-06-09
PCT/US2006/022326 WO2006135687A1 (en) 2005-06-09 2006-06-08 Pyrrolobenzodiazepine pyridine carboxamides and derivatives as follicle-stimulating hormone receptor antagonists

Publications (1)

Publication Number Publication Date
BRPI0611720A2 true BRPI0611720A2 (pt) 2016-11-22

Family

ID=37102119

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0611720A BRPI0611720A2 (pt) 2005-06-09 2006-06-08 "composto, composição, e, métodos de inibir a fertilidade,de evitar a concepção, e de bloquear o desenvolvimento folicular mediado por fsh em um mamífero"

Country Status (9)

Country Link
US (1) US7678787B2 (pt)
EP (1) EP1893615A1 (pt)
JP (1) JP2008543765A (pt)
CN (1) CN101208342A (pt)
AU (1) AU2006258007A1 (pt)
BR (1) BRPI0611720A2 (pt)
CA (1) CA2609714A1 (pt)
MX (1) MX2007015643A (pt)
WO (1) WO2006135687A1 (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2660799C (en) * 2006-08-14 2013-03-19 Council Of Scientific & Industrial Research Pyrrolo[2,1-c][1,4]benzodiazepine hybrids and a process for the preparation thereof
MX2009013332A (es) 2007-06-08 2010-01-25 Mannkind Corp Inhibidores de ire-1 alfa.
US20100061976A1 (en) * 2008-07-24 2010-03-11 Searete Llc, A Limited Liability Corporation Of The State Of Delaware Method for treating or preventing osteoporosis by reducing follicle stimulating hormone to cyclic physiological levels in a mammalian subject
CA2891280C (en) 2012-11-24 2018-03-20 Hangzhou Dac Biotech Co., Ltd. Hydrophilic linkers and their uses for conjugation of drugs to cell binding molecules
US10464955B2 (en) 2014-02-28 2019-11-05 Hangzhou Dac Biotech Co., Ltd. Charged linkers and their uses for conjugation
CA2989269C (en) 2015-06-15 2020-09-22 Robert Yongxin Zhao Hydrophilic linkers for conjugation of a cytotoxic agent or chromophore molecule to a cell-binding molecule
NZ739830A (en) 2015-07-12 2021-12-24 Hangzhou Dac Biotech Co Ltd Bridge linkers for conjugation of cell-binding molecules
US9839687B2 (en) 2015-07-15 2017-12-12 Suzhou M-Conj Biotech Co., Ltd. Acetylenedicarboxyl linkers and their uses in specific conjugation of a cell-binding molecule
KR20220150408A (ko) 2016-11-14 2022-11-10 항저우 디에이씨 바이오테크 씨오, 엘티디 결합 링커, 그러한 결합 링커를 함유하는 세포 결합 분자-약물 결합체, 링커를 갖는 그러한 결합체의 제조 및 사용
CN113004284B (zh) * 2019-12-20 2022-08-12 成都康弘药业集团股份有限公司 作为血浆激肽释放酶抑制剂的四环类化合物及其用途
EP4426727A2 (en) 2021-11-03 2024-09-11 Hangzhou Dac Biotech Co., Ltd. Specific conjugation of an antibody
EP4548932A1 (en) 2022-06-30 2025-05-07 Toray Industries, Inc. Pharmaceutical composition for treating and/or preventing cancer
CN115710200B (zh) * 2022-11-21 2024-08-09 重庆医科大学 苯甲酰氟类化合物、苯甲酸类化合物及其制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6235755B1 (en) 1998-08-07 2001-05-22 Applied Research Systems Ars Holding N.A. FSH mimetics for the treatment of infertility
US6200963B1 (en) 1999-03-31 2001-03-13 American Home Products Corporation Aryl sulfonic acids as FSH antagonists
US6355633B1 (en) 1999-03-31 2002-03-12 American Home Products Corporation Aryl sulfonic acids and derivatives as FSH antagonists
WO2000058277A1 (en) 1999-03-31 2000-10-05 American Home Products Corporation Aryl sulfonic acids and derivatives as fsh antagonists
US6426357B1 (en) 1999-07-27 2002-07-30 Affymax, Inc. Antagonists of follicle stimulating hormone activity
WO2001047875A1 (en) 1999-12-27 2001-07-05 Ortho-Mcneil Pharmaceutical, Inc. Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
EP1307193A1 (en) 2000-07-27 2003-05-07 Affymax Research Institute Agonists of follicle stimulating hormone activity
ATE277913T1 (de) 2001-01-19 2004-10-15 Pharmacopeia Inc Bisarylderivate mit fsh rezeptor modulierender aktivität
US7064120B2 (en) 2001-04-12 2006-06-20 Wyeth Tricyclic pyridyl carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists
US7109193B2 (en) 2001-04-12 2006-09-19 Wyeth Tricyclic diazepines tocolytic oxytocin receptor antagonists
US6903087B2 (en) 2001-04-12 2005-06-07 Wyeth Pyrido cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists
US7202239B2 (en) * 2001-04-12 2007-04-10 Wyeth Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonists
US6900200B2 (en) 2001-04-12 2005-05-31 Wyeth Tricyclic hydroxy carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists
CZ20042A3 (en) 2001-07-02 2004-04-14 Akzo Nobel N. V. Tetrahydroquinoline derivatives
TWI322012B (en) 2002-12-20 2010-03-21 Organon Nv Tetrahydroquinoline derivatives
TWI306855B (en) * 2002-12-20 2009-03-01 Organon Nv Tetrahydroquinoline derivatives

Also Published As

Publication number Publication date
WO2006135687A1 (en) 2006-12-21
MX2007015643A (es) 2008-02-15
JP2008543765A (ja) 2008-12-04
CA2609714A1 (en) 2006-12-21
AU2006258007A1 (en) 2006-12-21
CN101208342A (zh) 2008-06-25
US20060287522A1 (en) 2006-12-21
US7678787B2 (en) 2010-03-16
EP1893615A1 (en) 2008-03-05

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Legal Events

Date Code Title Description
B06G Technical and formal requirements: other requirements [chapter 6.7 patent gazette]

Free format text: SOLICITA-SE A REGULARIZACAO DA PROCURACAO, UMA VEZ QUE BASEADO NO ARTIGO 216 1O DA LPI, O DOCUMENTO DE PROCURACAO DEVE SER APRESENTADO NO ORIGINAL, TRASLADO OU FOTOCOPIA AUTENTICADA.

B11Z Dismissal: petition dismissal - article 216, par 2 of industrial property law

Free format text: REFERENTE A PETICAO NO 20070174214/RJ DE 07/12/2007.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]