BRPI0717461A2 - Modificações de cristais de -3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin- 4-il]-pirrol-2,5-diona - Google Patents

Modificações de cristais de -3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin- 4-il]-pirrol-2,5-diona

Info

Publication number
BRPI0717461A2
BRPI0717461A2 BRPI0717461-6A2A BRPI0717461A BRPI0717461A2 BR PI0717461 A2 BRPI0717461 A2 BR PI0717461A2 BR PI0717461 A BRPI0717461 A BR PI0717461A BR PI0717461 A2 BRPI0717461 A2 BR PI0717461A2
Authority
BR
Brazil
Prior art keywords
pirrol
diona
quinazolin
piperazin
indol
Prior art date
Application number
BRPI0717461-6A2A
Other languages
English (en)
Inventor
Piotr Karpinski
Stephanie Monnier
Elias Ndzie
Dimitris Papoutsakis
Paul Allen Sutton
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38921707&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0717461(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BRPI0717461A2 publication Critical patent/BRPI0717461A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0717461-6A2A 2006-10-20 2007-10-18 Modificações de cristais de -3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin- 4-il]-pirrol-2,5-diona BRPI0717461A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US85338406P 2006-10-20 2006-10-20
PCT/US2007/022241 WO2008051440A1 (en) 2006-10-20 2007-10-18 Crystal modifications -3- (1h-ind0l-3-yl) -4- [2- (4-methyl-piperazin-1-yl) -quinazolin-4-yl] -pyrrole-2, 5-d ione

Publications (1)

Publication Number Publication Date
BRPI0717461A2 true BRPI0717461A2 (pt) 2013-10-08

Family

ID=38921707

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0717461-6A2A BRPI0717461A2 (pt) 2006-10-20 2007-10-18 Modificações de cristais de -3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin- 4-il]-pirrol-2,5-diona

Country Status (23)

Country Link
US (1) US8865897B2 (pt)
EP (1) EP2102195A1 (pt)
JP (1) JP5302199B2 (pt)
KR (1) KR20090073231A (pt)
CN (2) CN103265533A (pt)
AR (1) AR063491A1 (pt)
AU (1) AU2007309558B2 (pt)
BR (1) BRPI0717461A2 (pt)
CA (1) CA2666965A1 (pt)
CL (1) CL2007003006A1 (pt)
EC (1) ECSP099344A (pt)
IL (1) IL197962A (pt)
MA (1) MA30886B1 (pt)
MX (1) MX2009004048A (pt)
MY (1) MY158026A (pt)
NO (1) NO20091970L (pt)
NZ (1) NZ576241A (pt)
PE (1) PE20081133A1 (pt)
RU (1) RU2481341C2 (pt)
TN (1) TN2009000147A1 (pt)
TW (1) TWI399374B (pt)
WO (1) WO2008051440A1 (pt)
ZA (1) ZA200902048B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0808354A2 (pt) * 2007-03-09 2014-07-29 Novartis Ag Sais de 3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin-4 -il]-pirrola-2,5-diona
US9017528B2 (en) 2011-04-14 2015-04-28 Tel Nexx, Inc. Electro chemical deposition and replenishment apparatus
US9005409B2 (en) 2011-04-14 2015-04-14 Tel Nexx, Inc. Electro chemical deposition and replenishment apparatus
US9303329B2 (en) 2013-11-11 2016-04-05 Tel Nexx, Inc. Electrochemical deposition apparatus with remote catholyte fluid management

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2070921A1 (en) * 2000-11-07 2009-06-17 Novartis Ag Indolylmaleimide derivatives as protein kinase c inhibitors
GB0504203D0 (en) * 2005-03-01 2005-04-06 Novartis Ag Organic compounds
AU2008266515B2 (en) 2007-06-18 2014-05-01 Sanofi Pyrrole derivatives as P2Y12 antagonists

Also Published As

Publication number Publication date
WO2008051440A1 (en) 2008-05-02
US20100041884A1 (en) 2010-02-18
MA30886B1 (fr) 2009-11-02
IL197962A0 (en) 2009-12-24
CN101522664A (zh) 2009-09-02
ECSP099344A (es) 2009-06-30
EP2102195A1 (en) 2009-09-23
TWI399374B (zh) 2013-06-21
CN103265533A (zh) 2013-08-28
CA2666965A1 (en) 2008-05-02
TW200829572A (en) 2008-07-16
MY158026A (en) 2016-08-30
RU2481341C2 (ru) 2013-05-10
NZ576241A (en) 2012-05-25
MX2009004048A (es) 2009-04-27
AU2007309558A1 (en) 2008-05-02
AU2007309558B2 (en) 2012-05-24
RU2009118816A (ru) 2010-11-27
KR20090073231A (ko) 2009-07-02
NO20091970L (no) 2009-05-20
ZA200902048B (en) 2010-01-27
CL2007003006A1 (es) 2008-05-23
AR063491A1 (es) 2009-01-28
US8865897B2 (en) 2014-10-21
CN101522664B (zh) 2013-06-12
PE20081133A1 (es) 2008-09-16
JP2010506927A (ja) 2010-03-04
JP5302199B2 (ja) 2013-10-02
IL197962A (en) 2013-08-29
TN2009000147A1 (en) 2010-10-18

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 9A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.