MA30886B1 - Modifications cristallines - Google Patents

Modifications cristallines

Info

Publication number
MA30886B1
MA30886B1 MA31867A MA31867A MA30886B1 MA 30886 B1 MA30886 B1 MA 30886B1 MA 31867 A MA31867 A MA 31867A MA 31867 A MA31867 A MA 31867A MA 30886 B1 MA30886 B1 MA 30886B1
Authority
MA
Morocco
Prior art keywords
crystalline modifications
quinazolin
piperazin
indol
dione
Prior art date
Application number
MA31867A
Other languages
English (en)
Inventor
Piotr Karpinski
Stephanie Monnier
Elias Ndzie
Dimitris Papoutsakis
Paul Allen Sutton
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38921707&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA30886(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MA30886B1 publication Critical patent/MA30886B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LA PRÉSENTE INVENTION CONCERNE UNE NOUVELLE FORME CRISTALLINE DU SEL D'ACÉTATE DE 3-(1H-INDOL-3-YL)-4-[2-(4-MÉTHYL-PIPÉRAZIN-1-YL)-QUINAZOLIN-4-YL]-PYRROLE-2,5-DIONE, QUI PEUT ÊTRE UTILISÉE PAR EXEMPLE POUR UNE TRANSPLANTATION.
MA31867A 2006-10-20 2009-05-13 Modifications cristallines MA30886B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85338406P 2006-10-20 2006-10-20

Publications (1)

Publication Number Publication Date
MA30886B1 true MA30886B1 (fr) 2009-11-02

Family

ID=38921707

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31867A MA30886B1 (fr) 2006-10-20 2009-05-13 Modifications cristallines

Country Status (23)

Country Link
US (1) US8865897B2 (fr)
EP (1) EP2102195A1 (fr)
JP (1) JP5302199B2 (fr)
KR (1) KR20090073231A (fr)
CN (2) CN103265533A (fr)
AR (1) AR063491A1 (fr)
AU (1) AU2007309558B2 (fr)
BR (1) BRPI0717461A2 (fr)
CA (1) CA2666965A1 (fr)
CL (1) CL2007003006A1 (fr)
EC (1) ECSP099344A (fr)
IL (1) IL197962A (fr)
MA (1) MA30886B1 (fr)
MX (1) MX2009004048A (fr)
MY (1) MY158026A (fr)
NO (1) NO20091970L (fr)
NZ (1) NZ576241A (fr)
PE (1) PE20081133A1 (fr)
RU (1) RU2481341C2 (fr)
TN (1) TN2009000147A1 (fr)
TW (1) TWI399374B (fr)
WO (1) WO2008051440A1 (fr)
ZA (1) ZA200902048B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0808354A2 (pt) * 2007-03-09 2014-07-29 Novartis Ag Sais de 3-(1h-indol-3-il)-4-[2-(4-metil-piperazin-1-il)-quinazolin-4 -il]-pirrola-2,5-diona
US9017528B2 (en) 2011-04-14 2015-04-28 Tel Nexx, Inc. Electro chemical deposition and replenishment apparatus
US9005409B2 (en) 2011-04-14 2015-04-14 Tel Nexx, Inc. Electro chemical deposition and replenishment apparatus
US9303329B2 (en) 2013-11-11 2016-04-05 Tel Nexx, Inc. Electrochemical deposition apparatus with remote catholyte fluid management

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2070921A1 (fr) * 2000-11-07 2009-06-17 Novartis Ag Dérivés d'indolylmaléimide comme inhibiteurs de la protéine kinase C
GB0504203D0 (en) * 2005-03-01 2005-04-06 Novartis Ag Organic compounds
AU2008266515B2 (en) 2007-06-18 2014-05-01 Sanofi Pyrrole derivatives as P2Y12 antagonists

Also Published As

Publication number Publication date
WO2008051440A1 (fr) 2008-05-02
US20100041884A1 (en) 2010-02-18
IL197962A0 (en) 2009-12-24
CN101522664A (zh) 2009-09-02
ECSP099344A (es) 2009-06-30
EP2102195A1 (fr) 2009-09-23
TWI399374B (zh) 2013-06-21
CN103265533A (zh) 2013-08-28
CA2666965A1 (fr) 2008-05-02
TW200829572A (en) 2008-07-16
MY158026A (en) 2016-08-30
BRPI0717461A2 (pt) 2013-10-08
RU2481341C2 (ru) 2013-05-10
NZ576241A (en) 2012-05-25
MX2009004048A (es) 2009-04-27
AU2007309558A1 (en) 2008-05-02
AU2007309558B2 (en) 2012-05-24
RU2009118816A (ru) 2010-11-27
KR20090073231A (ko) 2009-07-02
NO20091970L (no) 2009-05-20
ZA200902048B (en) 2010-01-27
CL2007003006A1 (es) 2008-05-23
AR063491A1 (es) 2009-01-28
US8865897B2 (en) 2014-10-21
CN101522664B (zh) 2013-06-12
PE20081133A1 (es) 2008-09-16
JP2010506927A (ja) 2010-03-04
JP5302199B2 (ja) 2013-10-02
IL197962A (en) 2013-08-29
TN2009000147A1 (en) 2010-10-18

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