BRPI0719486A2 - "forma farmacêutica sólida oral desitegrante, não-efervescente, métodos para tratar uma mulher que necessite de um contraceptivo de emergência, pacote terapêutico para tratar uma mulher que necessite de contracepção de emergência e processo para a preparação de uma forma sólida de dosagem farmacêutica oral desintegrante, não-efervescente" - Google Patents
"forma farmacêutica sólida oral desitegrante, não-efervescente, métodos para tratar uma mulher que necessite de um contraceptivo de emergência, pacote terapêutico para tratar uma mulher que necessite de contracepção de emergência e processo para a preparação de uma forma sólida de dosagem farmacêutica oral desintegrante, não-efervescente"Info
- Publication number
- BRPI0719486A2 BRPI0719486A2 BRPI0719486-2A2A BRPI0719486A BRPI0719486A2 BR PI0719486 A2 BRPI0719486 A2 BR PI0719486A2 BR PI0719486 A BRPI0719486 A BR PI0719486A BR PI0719486 A2 BRPI0719486 A2 BR PI0719486A2
- Authority
- BR
- Brazil
- Prior art keywords
- treat
- woman
- preemphere
- desidgrant
- proparation
- Prior art date
Links
- 239000003433 contraceptive agent Substances 0.000 title 1
- 230000002254 contraceptive effect Effects 0.000 title 1
- 239000007787 solid Substances 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Zoology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87582706P | 2006-12-20 | 2006-12-20 | |
| PCT/US2007/025974 WO2008079245A2 (en) | 2006-12-20 | 2007-12-20 | Orally disintegrating solid dosage forms comprising progestin and methods of making and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0719486A2 true BRPI0719486A2 (pt) | 2014-02-18 |
Family
ID=39563076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0719486-2A2A BRPI0719486A2 (pt) | 2006-12-20 | 2007-12-20 | "forma farmacêutica sólida oral desitegrante, não-efervescente, métodos para tratar uma mulher que necessite de um contraceptivo de emergência, pacote terapêutico para tratar uma mulher que necessite de contracepção de emergência e processo para a preparação de uma forma sólida de dosagem farmacêutica oral desintegrante, não-efervescente" |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US7867515B2 (pt) |
| EP (1) | EP2124900B1 (pt) |
| JP (1) | JP5649305B2 (pt) |
| AU (1) | AU2007338843B2 (pt) |
| BR (1) | BRPI0719486A2 (pt) |
| CA (1) | CA2674776A1 (pt) |
| ES (1) | ES2531929T3 (pt) |
| IL (1) | IL199472A0 (pt) |
| MX (1) | MX2009006823A (pt) |
| RU (1) | RU2465907C2 (pt) |
| WO (1) | WO2008079245A2 (pt) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1984443B1 (en) * | 2006-02-14 | 2014-04-02 | The Procter and Gamble Company | Personal care compositions comprising responsive particles |
| ES2531929T3 (es) * | 2006-12-20 | 2015-03-20 | Teva Women's Health, Inc. | Formas de dosificación solidas que se disgregan en la boca que comprenden progestina y métodos para hacer y usar las mismas |
| EA201070715A1 (ru) * | 2007-12-20 | 2011-02-28 | Тева Вимен'С Хелс, Инк. | Режимы дозирования, фармацевтические композиции и упаковки для экстренной контрацепции |
| FR2937862B1 (fr) * | 2008-11-03 | 2010-11-19 | Mohammed Ridha Chakroun | Kit contraceptif |
| US8512745B2 (en) | 2008-12-08 | 2013-08-20 | Laboratoire Hra Pharma | Ulipristal acetate tablets |
| HRP20161437T1 (hr) * | 2009-04-14 | 2017-02-10 | Laboratoire Hra Pharma | Postupak hitne kontracepcije |
| WO2012164096A1 (en) | 2011-06-01 | 2012-12-06 | Estetra S.A. | Process for the production of estetrol intermediates |
| BR112013030833B1 (pt) | 2011-06-01 | 2019-09-03 | Estetra S A | processo para a preparação de um composto de fórmula (i) e processo para a preparação de estetrol |
| EP2383279A1 (en) | 2011-07-19 | 2011-11-02 | Pantarhei Bioscience B.V. | Process for the preparation of estetrol |
| JP5928159B2 (ja) * | 2012-05-28 | 2016-06-01 | ニプロ株式会社 | 医薬組成物 |
| FR2997627B1 (fr) | 2012-11-08 | 2015-01-16 | Hra Pharma Lab | Produit de co-micronisation comprenant de l'ulipristal acetate |
| HUE035848T2 (en) * | 2013-12-12 | 2018-05-28 | Donesta Bioscience B V | Solid dispensing unit containing an estetrol compound in the mouth |
| CN103877048A (zh) * | 2014-03-26 | 2014-06-25 | 邵娜 | 一种黄体酮口腔崩解片及其制备方法 |
| WO2015160595A1 (en) * | 2014-04-14 | 2015-10-22 | Abbott Molecular, Inc. | Medium used for blood sample collection and transport |
| RS57328B1 (sr) | 2015-06-18 | 2018-08-31 | Mithra Pharmaceuticals S A | Orodisperzibilna dozna jedinica koja sadrži estetrolsku komponentu |
| WO2016203044A1 (en) | 2015-06-18 | 2016-12-22 | Mithra Pharmaceuticals S.A. | Orodispersible tablet containing estetrol |
| LT3310345T (lt) | 2015-06-18 | 2021-06-25 | Estetra Sprl | Burnoje disperguojama tabletė, turinti estetrolio |
| NZ737945A (en) | 2015-06-18 | 2023-06-30 | Estetra Sprl | Orodispersible dosage unit containing an estetrol component |
| CN107595788B (zh) * | 2016-07-11 | 2020-08-21 | 武汉朗来科技发展有限公司 | 一种用于口服固体制剂的复合崩解剂体系及含有该复合崩解剂体系的口服固体制剂 |
| CA3178291A1 (en) | 2016-08-05 | 2018-04-12 | Estetra Srl | Method for the management of dysmenorrhea and menstrual pain |
| TWI801561B (zh) | 2018-04-19 | 2023-05-11 | 比利時商依思特拉私人有限責任公司 | 化合物及其用於緩解絕經相關症狀的用途 |
| CR20200486A (es) | 2018-04-19 | 2021-01-27 | Estetra Sprl | Compuestos y sus usos para aliviar los síntomas asociados a la menopausa |
| CN109276550B (zh) * | 2018-11-27 | 2021-01-12 | 西安圣雪沙药物开发有限公司 | 一种左炔诺孕酮片及其制备方法 |
| CN110917154A (zh) * | 2019-12-12 | 2020-03-27 | 上海信谊天平药业有限公司 | 一种左炔诺孕酮片的制备方法 |
| TWI893101B (zh) | 2020-04-16 | 2025-08-11 | 比利時商埃斯特拉有限責任公司 | 具有降低之副作用之避孕組成物 |
| AU2021351921A1 (en) | 2020-09-29 | 2023-04-06 | Millicent Pharma Limited | Orodispersible formulations |
| WO2022225986A1 (en) * | 2021-04-19 | 2022-10-27 | Archer David Fitzgerald | On demand female contraceptive |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IE61236B1 (en) * | 1986-07-15 | 1994-10-19 | American Home Prod | Combination dosage form for pre-menopausal women |
| US5633011A (en) * | 1994-08-04 | 1997-05-27 | Alza Corporation | Progesterone replacement therapy |
| GB9603699D0 (en) * | 1996-02-21 | 1996-04-17 | Boots Co Plc | Therapeutic composition |
| CA2253289A1 (en) * | 1996-05-16 | 1997-11-20 | Roderick L. Mackenzie | Emergency contraceptive kit |
| JPH1171268A (ja) * | 1997-08-28 | 1999-03-16 | Kayaku:Kk | 性ホルモン含有錠剤 |
| FR2772617B1 (fr) * | 1997-12-19 | 2001-03-09 | Besins Iscovesco Lab | Comprime de progesterone et son procede de preparation |
| US6368625B1 (en) * | 1998-08-12 | 2002-04-09 | Cima Labs Inc. | Orally disintegrable tablet forming a viscous slurry |
| EP1161941A4 (en) | 1999-03-15 | 2002-08-28 | Kaken Pharma Co Ltd | QUICKLY DISMANTLING TABLETS AND METHOD FOR THE PRODUCTION THEREOF |
| US6667050B1 (en) * | 1999-04-06 | 2003-12-23 | Galen (Chemicals) Limited | Chewable oral contraceptive |
| US6316029B1 (en) * | 2000-05-18 | 2001-11-13 | Flak Pharma International, Ltd. | Rapidly disintegrating solid oral dosage form |
| PT1355644E (pt) * | 2001-01-26 | 2006-11-30 | Schering Corp | Utilização de compostos azetidinona substituídos para o tratamento de sitosterolemia |
| HU227198B1 (en) * | 2001-11-27 | 2010-10-28 | Richter Gedeon Nyrt | Pharmaceutical composition for emergency contraception containing levonorgestrel |
| US6962908B2 (en) * | 2001-12-21 | 2005-11-08 | Warner Chilcott Company Inc. | Oral pharmaceutical products containing 17 β-estradiol-3-lower alkanoate, method of administering the same and process of preparation |
| CN1819819B (zh) * | 2003-05-07 | 2011-03-09 | 株式会社三养社 | 用于制备速熔片的高度可塑性颗粒 |
| KR101159617B1 (ko) * | 2003-10-15 | 2012-06-27 | 후지카가쿠고교가부시키가이샤 | 구강내 속붕해성 정제 |
| JP4519444B2 (ja) * | 2003-10-31 | 2010-08-04 | ライオン株式会社 | 口腔内崩壊錠 |
| WO2005055945A2 (en) * | 2003-12-08 | 2005-06-23 | Gel-Del Technologies, Inc. | Mucoadhesive drug delivery devices and methods of making and using thereof |
| EP1625849A1 (en) * | 2004-08-09 | 2006-02-15 | Liconsa, Liberacion Controlada de Sustancias Activas, S.A. | Pharmaceutical composition comprising drospirenone and ethynylestradiol |
| CN1634077A (zh) * | 2004-11-18 | 2005-07-06 | 王立强 | 左炔诺孕酮口腔崩解片制剂及其制备方法 |
| JP2008536922A (ja) * | 2005-04-22 | 2008-09-11 | テバ・ファーマシューティカルズ・ユーエスエー・インコーポレイテッド | オランザピンの医薬用経口崩壊錠 |
| US8663681B2 (en) * | 2005-05-26 | 2014-03-04 | Teva Women's Health, Inc. | Oral dosage forms comprising progesterone and methods of making and using the same |
| ES2531929T3 (es) * | 2006-12-20 | 2015-03-20 | Teva Women's Health, Inc. | Formas de dosificación solidas que se disgregan en la boca que comprenden progestina y métodos para hacer y usar las mismas |
| EA201070715A1 (ru) * | 2007-12-20 | 2011-02-28 | Тева Вимен'С Хелс, Инк. | Режимы дозирования, фармацевтические композиции и упаковки для экстренной контрацепции |
-
2007
- 2007-12-20 ES ES07863134.8T patent/ES2531929T3/es active Active
- 2007-12-20 EP EP07863134.8A patent/EP2124900B1/en active Active
- 2007-12-20 BR BRPI0719486-2A2A patent/BRPI0719486A2/pt not_active IP Right Cessation
- 2007-12-20 AU AU2007338843A patent/AU2007338843B2/en not_active Ceased
- 2007-12-20 CA CA002674776A patent/CA2674776A1/en not_active Abandoned
- 2007-12-20 WO PCT/US2007/025974 patent/WO2008079245A2/en not_active Ceased
- 2007-12-20 JP JP2009542901A patent/JP5649305B2/ja not_active Expired - Fee Related
- 2007-12-20 US US12/003,234 patent/US7867515B2/en not_active Expired - Fee Related
- 2007-12-20 MX MX2009006823A patent/MX2009006823A/es active IP Right Grant
- 2007-12-20 RU RU2009125972/15A patent/RU2465907C2/ru not_active IP Right Cessation
-
2009
- 2009-06-21 IL IL199472A patent/IL199472A0/en unknown
-
2010
- 2010-12-02 US US12/958,975 patent/US8226980B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP2124900A4 (en) | 2013-04-03 |
| US8226980B2 (en) | 2012-07-24 |
| JP5649305B2 (ja) | 2015-01-07 |
| JP2010513514A (ja) | 2010-04-30 |
| WO2008079245A2 (en) | 2008-07-03 |
| RU2465907C2 (ru) | 2012-11-10 |
| WO2008079245A3 (en) | 2008-12-04 |
| ES2531929T3 (es) | 2015-03-20 |
| CA2674776A1 (en) | 2008-07-03 |
| AU2007338843B2 (en) | 2013-05-09 |
| MX2009006823A (es) | 2009-07-03 |
| US20080175906A1 (en) | 2008-07-24 |
| EP2124900B1 (en) | 2014-12-03 |
| IL199472A0 (en) | 2010-03-28 |
| AU2007338843A1 (en) | 2008-07-03 |
| EP2124900A2 (en) | 2009-12-02 |
| RU2009125972A (ru) | 2011-01-27 |
| US20110136771A1 (en) | 2011-06-09 |
| US7867515B2 (en) | 2011-01-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 9A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] | ||
| B25E | Requested change of name of applicant rejected |
Owner name: DURAMED PHARMACEUTICALS, INC (US) |